JP2020531487A5 - - Google Patents

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Publication number
JP2020531487A5
JP2020531487A5 JP2020510099A JP2020510099A JP2020531487A5 JP 2020531487 A5 JP2020531487 A5 JP 2020531487A5 JP 2020510099 A JP2020510099 A JP 2020510099A JP 2020510099 A JP2020510099 A JP 2020510099A JP 2020531487 A5 JP2020531487 A5 JP 2020531487A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020510099A
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Japanese (ja)
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JP7199738B2 (ja
JPWO2019038384A5 (https=
JP2020531487A (ja
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Priority claimed from PCT/EP2018/072785 external-priority patent/WO2019038384A1/en
Publication of JP2020531487A publication Critical patent/JP2020531487A/ja
Publication of JPWO2019038384A5 publication Critical patent/JPWO2019038384A5/ja
Publication of JP2020531487A5 publication Critical patent/JP2020531487A5/ja
Priority to JP2022198545A priority Critical patent/JP2023021277A/ja
Application granted granted Critical
Publication of JP7199738B2 publication Critical patent/JP7199738B2/ja
Active legal-status Critical Current
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JP2020510099A 2017-08-23 2018-08-23 アザインドリルピリドンおよびジアザインドリルピリドン化合物 Active JP7199738B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2022198545A JP2023021277A (ja) 2017-08-23 2022-12-13 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP17187519.8 2017-08-23
EP17187519 2017-08-23
PCT/EP2018/072785 WO2019038384A1 (en) 2017-08-23 2018-08-23 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022198545A Division JP2023021277A (ja) 2017-08-23 2022-12-13 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Publications (4)

Publication Number Publication Date
JP2020531487A JP2020531487A (ja) 2020-11-05
JPWO2019038384A5 JPWO2019038384A5 (https=) 2022-10-20
JP2020531487A5 true JP2020531487A5 (https=) 2022-10-20
JP7199738B2 JP7199738B2 (ja) 2023-01-06

Family

ID=59686871

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020510099A Active JP7199738B2 (ja) 2017-08-23 2018-08-23 アザインドリルピリドンおよびジアザインドリルピリドン化合物
JP2022198545A Ceased JP2023021277A (ja) 2017-08-23 2022-12-13 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2022198545A Ceased JP2023021277A (ja) 2017-08-23 2022-12-13 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Country Status (20)

Country Link
US (2) US11498919B2 (https=)
EP (2) EP3672967B1 (https=)
JP (2) JP7199738B2 (https=)
KR (1) KR102731945B1 (https=)
CN (3) CN116589461A (https=)
AU (1) AU2018321135B2 (https=)
CY (1) CY1124818T1 (https=)
DK (1) DK3672967T3 (https=)
ES (1) ES2902346T3 (https=)
HR (1) HRP20211999T1 (https=)
HU (1) HUE057818T2 (https=)
IL (3) IL302355A (https=)
LT (1) LT3672967T (https=)
PL (1) PL3672967T3 (https=)
PT (1) PT3672967T (https=)
RS (1) RS62785B1 (https=)
SI (1) SI3672967T1 (https=)
SM (1) SMT202100718T1 (https=)
TW (2) TW202325708A (https=)
WO (1) WO2019038384A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7199738B2 (ja) * 2017-08-23 2023-01-06 スプリント バイオサイエンス アクティエボラーグ アザインドリルピリドンおよびジアザインドリルピリドン化合物
CA3200038A1 (en) * 2020-11-25 2022-06-02 Deciphera Pharmaceuticals, Llc Anti-viral activity of vps34 inhibitors
WO2022115562A1 (en) 2020-11-25 2022-06-02 Deciphera Pharmaceuticals, Llc Morpholino derivatives as vsp34 inhibitors for use in the treatment of a viral infection

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1154024B (it) * 1982-09-22 1987-01-21 Lepetit Spa Derivati pridinici e procedimento per la loro produzione
WO2006127587A1 (en) 2005-05-20 2006-11-30 Vertex Pharmaceuticals Incorporated Pyrrolopyridines useful as inhibitors of protein kinase
CN102143746A (zh) * 2008-07-03 2011-08-03 埃克塞利希斯股份有限公司 Cdk 调节剂
CA2795422A1 (en) * 2010-04-19 2011-10-27 Abbvie Inc. Pyrrolopyridine inhibitors of kinases
AU2011346567A1 (en) 2010-12-21 2013-07-25 Novartis Ag Bi-heteroaryl compounds as Vps34 inhibitors
DK2655375T3 (en) 2010-12-23 2015-03-09 Sanofi Sa PYRIMIDINON DERIVATIVES, PREPARATION AND PHARMACEUTICAL USE THEREOF
GB201120317D0 (en) 2011-11-24 2012-01-04 Queen Mary & Westfield College Screening method
CN103450152B (zh) 2012-06-04 2015-11-18 济南海乐医药技术开发有限公司 基于吲唑、吲哚或氮杂吲唑、氮杂吲哚的双芳基脲类结构抗肿瘤药物
FR2992314B1 (fr) 2012-06-22 2015-10-16 Sanofi Sa Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one et 1,2,3,4-tetrahydro-pyrimido{1,2-a}pyrimidin-6-one comportant une morpholine substituee, leur preparation et leur utilisation pharmaceutique
AU2015206652A1 (en) 2014-01-14 2016-08-04 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
WO2015108881A1 (en) * 2014-01-14 2015-07-23 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
MA39823A (fr) 2014-04-03 2018-01-09 Janssen Pharmaceutica Nv Dérivés de pyridine macrocyclique
MA39822A (fr) 2014-04-03 2018-02-06 Janssen Pharmaceutica Nv Dérivés de pyrimidine bicycle
AU2017219846B2 (en) 2016-02-19 2021-05-13 Sprint Bioscience Ab 6-aryl-4-morpholin-1-ylpyridone compounds useful for the treatment of cancer and diabetes
DK3416957T3 (da) 2016-02-19 2020-09-21 Sprint Bioscience Ab 6-heterocyclyl-4-morpholin-4-ylpyridin-2-on-forbindelser anvendelige ved behandlingen af cancer og diabetes
JP7199738B2 (ja) * 2017-08-23 2023-01-06 スプリント バイオサイエンス アクティエボラーグ アザインドリルピリドンおよびジアザインドリルピリドン化合物

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