JP2020528907A5 - - Google Patents
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- JP2020528907A5 JP2020528907A5 JP2020504026A JP2020504026A JP2020528907A5 JP 2020528907 A5 JP2020528907 A5 JP 2020528907A5 JP 2020504026 A JP2020504026 A JP 2020504026A JP 2020504026 A JP2020504026 A JP 2020504026A JP 2020528907 A5 JP2020528907 A5 JP 2020528907A5
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023016586A JP7554300B2 (ja) | 2017-07-28 | 2023-02-07 | 大環式化合物およびその使用 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762538193P | 2017-07-28 | 2017-07-28 | |
| US62/538,193 | 2017-07-28 | ||
| US201862700990P | 2018-07-20 | 2018-07-20 | |
| US62/700,990 | 2018-07-20 | ||
| PCT/US2018/043817 WO2019023417A1 (en) | 2017-07-28 | 2018-07-26 | MACROCYCLIC COMPOUNDS AND USES THEREOF |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023016586A Division JP7554300B2 (ja) | 2017-07-28 | 2023-02-07 | 大環式化合物およびその使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020528907A JP2020528907A (ja) | 2020-10-01 |
| JP2020528907A5 true JP2020528907A5 (cg-RX-API-DMAC10.html) | 2021-09-02 |
| JP7224334B2 JP7224334B2 (ja) | 2023-02-17 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020504026A Active JP7224334B2 (ja) | 2017-07-28 | 2018-07-26 | 大環式化合物およびその使用 |
| JP2023016586A Active JP7554300B2 (ja) | 2017-07-28 | 2023-02-07 | 大環式化合物およびその使用 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023016586A Active JP7554300B2 (ja) | 2017-07-28 | 2023-02-07 | 大環式化合物およびその使用 |
Country Status (29)
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9714258B2 (en) | 2014-01-24 | 2017-07-25 | Tp Therapeutics, Inc. | Diaryl macrocycles as modulators of protein kinases |
| JP6871903B2 (ja) | 2015-07-02 | 2021-05-19 | ターニング・ポイント・セラピューティクス・インコーポレイテッドＴｕｒｎｉｎｇ Ｐｏｉｎｔ Ｔｈｅｒａｐｅｕｔｉｃｓ，Ｉｎｃ． | プロテインキナーゼのモジュレーターとしてのキラルジアリール大環状分子 |
| PT3733187T (pt) | 2015-07-21 | 2024-11-08 | Turning Point Therapeutics Inc | Macrociclo de diarilo quiral e utilização do mesmo no tratamento do cancro |
| JP2019527230A (ja) | 2016-07-28 | 2019-09-26 | ターニング・ポイント・セラピューティクス・インコーポレイテッドＴｕｒｎｉｎｇ Ｐｏｉｎｔ Ｔｈｅｒａｐｅｕｔｉｃｓ，Ｉｎｃ． | 大環状キナーゼ阻害剤 |
| TWI808958B (zh) | 2017-01-25 | 2023-07-21 | 美商特普醫葯公司 | 涉及二芳基巨環化合物之組合療法 |
| HRP20241197T1 (hr) | 2017-07-28 | 2024-11-22 | Turning Point Therapeutics, Inc. | Makrociklični spojevi i primjene istih |
| CN109516999B (zh) * | 2017-11-01 | 2021-08-17 | 郑州泰基鸿诺医药股份有限公司 | 用作蛋白质激酶调节剂的化合物及其应用 |
| PL3728271T3 (pl) | 2017-12-19 | 2023-01-23 | Turning Point Therapeutics, Inc. | Związki makrocykliczne do leczenia chorób |
| WO2019206069A1 (zh) | 2018-04-25 | 2019-10-31 | 北京普祺医药科技有限公司 | 一种二芳基巨环化合物、药物组合物以及其用途 |
| CN113490664B (zh) | 2018-10-22 | 2025-05-16 | 阿鲁米斯公司 | Tyk2抑制剂和其用途 |
| CA3132632A1 (en) * | 2019-03-11 | 2020-09-17 | Esker Therapeutics, Inc. | Tyk2 inhibitors and uses thereof |
| US12410191B2 (en) | 2019-05-21 | 2025-09-09 | Zhejiang Hisun Pharmaceutical Co., Ltd. | Macrolide derivatives, preparation method and application thereof |
| CN114423762B (zh) * | 2019-09-30 | 2024-03-29 | 浙江海正药业股份有限公司 | 大环类衍生物及其制备方法和用途 |
| EP4114530A4 (en) * | 2020-03-02 | 2024-04-17 | Turning Point Therapeutics, Inc. | THERAPEUTIC USES OF MACROCYCLIC COMPOUNDS |
| WO2021244609A1 (zh) * | 2020-06-04 | 2021-12-09 | 成都倍特药业股份有限公司 | 具有大环结构的化合物及其用途 |
| CN111620881B (zh) * | 2020-07-08 | 2023-03-31 | 浙江合聚生物医药有限公司 | 拉罗替尼衍生物及其制备方法和应用 |
| CN116635076A (zh) * | 2020-12-17 | 2023-08-22 | 荣山医药股份有限公司 | 大环化合物及其用途 |
| CN114685532A (zh) * | 2020-12-31 | 2022-07-01 | 正大天晴药业集团股份有限公司 | 大环类化合物及其医药用途 |
| CN116829562B (zh) * | 2021-02-10 | 2025-04-01 | 深圳国顺康医药科技有限公司 | 一种巨环化合物、药物组合物以及其用途 |
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