JP2020505432A - 耳鳴りの処置におけるガボキサドールの使用 - Google Patents

耳鳴りの処置におけるガボキサドールの使用 Download PDF

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Publication number
JP2020505432A
JP2020505432A JP2019542186A JP2019542186A JP2020505432A JP 2020505432 A JP2020505432 A JP 2020505432A JP 2019542186 A JP2019542186 A JP 2019542186A JP 2019542186 A JP2019542186 A JP 2019542186A JP 2020505432 A JP2020505432 A JP 2020505432A
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JP
Japan
Prior art keywords
gaboxadol
patient
pharmaceutically acceptable
acceptable salt
hours
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Pending
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JP2019542186A
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English (en)
Japanese (ja)
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JP2020505432A5 (enExample
Inventor
マシュー・デューリング
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Ovid Therapeutics Inc
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Ovid Therapeutics Inc
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Publication of JP2020505432A publication Critical patent/JP2020505432A/ja
Publication of JP2020505432A5 publication Critical patent/JP2020505432A5/ja
Priority to JP2022163131A priority Critical patent/JP2023011630A/ja
Priority to JP2024163596A priority patent/JP2024178317A/ja
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2019542186A 2017-02-03 2018-02-02 耳鳴りの処置におけるガボキサドールの使用 Pending JP2020505432A (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2022163131A JP2023011630A (ja) 2017-02-03 2022-10-11 耳鳴りの処置におけるガボキサドールの使用
JP2024163596A JP2024178317A (ja) 2017-02-03 2024-09-20 耳鳴りの処置におけるガボキサドールの使用

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201762454280P 2017-02-03 2017-02-03
US62/454,280 2017-02-03
US201762530528P 2017-07-10 2017-07-10
US62/530,528 2017-07-10
US201762536669P 2017-07-25 2017-07-25
US62/536,669 2017-07-25
PCT/US2018/016602 WO2018144827A1 (en) 2017-02-03 2018-02-02 Use of gaboxadol in the treatment of tinnitus

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022163131A Division JP2023011630A (ja) 2017-02-03 2022-10-11 耳鳴りの処置におけるガボキサドールの使用

Publications (2)

Publication Number Publication Date
JP2020505432A true JP2020505432A (ja) 2020-02-20
JP2020505432A5 JP2020505432A5 (enExample) 2021-03-18

Family

ID=63038963

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2019542186A Pending JP2020505432A (ja) 2017-02-03 2018-02-02 耳鳴りの処置におけるガボキサドールの使用
JP2022163131A Pending JP2023011630A (ja) 2017-02-03 2022-10-11 耳鳴りの処置におけるガボキサドールの使用
JP2024163596A Pending JP2024178317A (ja) 2017-02-03 2024-09-20 耳鳴りの処置におけるガボキサドールの使用

Family Applications After (2)

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JP2022163131A Pending JP2023011630A (ja) 2017-02-03 2022-10-11 耳鳴りの処置におけるガボキサドールの使用
JP2024163596A Pending JP2024178317A (ja) 2017-02-03 2024-09-20 耳鳴りの処置におけるガボキサドールの使用

Country Status (17)

Country Link
US (3) US10071083B2 (enExample)
EP (1) EP3576738B1 (enExample)
JP (3) JP2020505432A (enExample)
KR (1) KR20190112046A (enExample)
CN (1) CN110402140A (enExample)
AU (1) AU2018215363A1 (enExample)
BR (1) BR112019015832A2 (enExample)
CA (1) CA3051586A1 (enExample)
DK (1) DK3576738T3 (enExample)
ES (1) ES2930899T3 (enExample)
HU (1) HUE060609T2 (enExample)
IL (1) IL268210A (enExample)
MX (1) MX393900B (enExample)
PE (1) PE20191407A1 (enExample)
PL (1) PL3576738T3 (enExample)
PT (1) PT3576738T (enExample)
WO (1) WO2018144827A1 (enExample)

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MX391708B (es) 2015-07-17 2025-03-21 Ovid Therapeutics Inc Metodos para tratar trastornos del desarrollo con gaboxadol.
MX2019001669A (es) 2016-08-11 2019-09-27 Ovid Therapeutics Inc Metodos y composiciones para el tratamiento de trastornos epilepticos.
US10071083B2 (en) 2017-02-03 2018-09-11 Ovid Therapeutics Inc Use of gaboxadol in the treatment of tinnitus
KR20210062662A (ko) 2018-09-20 2021-05-31 오비드 테라퓨틱스 인크. 투렛 증후군, 틱들 및 말더듬의 치료를 위한 가복사돌의 사용
CN113395962A (zh) 2018-11-21 2021-09-14 Certego治疗公司 加波沙朵用于降低自杀风险和快速缓解抑郁症
WO2020131856A1 (en) * 2018-12-17 2020-06-25 Ovid Therapeutics Inc. Use of gaboxadol for the treatment of non-24 hour sleep-wake disorder
AU2020405060A1 (en) * 2019-12-18 2022-06-09 Ovid Therapeutics Inc. Gaboxadol for therapeutic treatment of 1p36 deletion syndrome
AU2021275863A1 (en) 2020-05-20 2023-02-02 Certego Therapeutics Inc. Ring deuterated gaboxadol and its use for the treatment of psychiatric disorders
EP4299059A1 (en) 2022-07-01 2024-01-03 Labelic Analysis, S.L. Composition for the treatment of tinnitus

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Also Published As

Publication number Publication date
US10188635B2 (en) 2019-01-29
AU2018215363A1 (en) 2019-08-15
DK3576738T3 (da) 2022-11-28
CN110402140A (zh) 2019-11-01
HUE060609T2 (hu) 2023-04-28
EP3576738A1 (en) 2019-12-11
WO2018144827A1 (en) 2018-08-09
MX2019009190A (es) 2019-09-26
US20180344709A1 (en) 2018-12-06
ES2930899T3 (es) 2022-12-22
JP2024178317A (ja) 2024-12-24
US10071083B2 (en) 2018-09-11
BR112019015832A2 (pt) 2020-03-31
IL268210A (en) 2019-09-26
PE20191407A1 (es) 2019-10-04
CA3051586A1 (en) 2018-08-09
JP2023011630A (ja) 2023-01-24
PL3576738T3 (pl) 2023-02-06
EP3576738B1 (en) 2022-10-12
MX393900B (es) 2025-03-24
KR20190112046A (ko) 2019-10-02
EP3576738A4 (en) 2021-02-17
PT3576738T (pt) 2022-11-30
US20180221355A1 (en) 2018-08-09
US20190111033A1 (en) 2019-04-18

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