JP2019518026A5 - - Google Patents
Info
- Publication number
- JP2019518026A5 JP2019518026A5 JP2018563619A JP2018563619A JP2019518026A5 JP 2019518026 A5 JP2019518026 A5 JP 2019518026A5 JP 2018563619 A JP2018563619 A JP 2018563619A JP 2018563619 A JP2018563619 A JP 2018563619A JP 2019518026 A5 JP2019518026 A5 JP 2019518026A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- crystal
- crystals
- solvate
- Prior art date
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2016/084300 | 2016-06-01 | ||
| CNPCT/CN2016/084300 | 2016-06-01 | ||
| PCT/CN2017/086760 WO2017206924A1 (zh) | 2016-06-01 | 2017-06-01 | 抑制蛋白激酶活性化合物的晶型及其应用 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2019518026A JP2019518026A (ja) | 2019-06-27 |
| JPWO2017206924A5 JPWO2017206924A5 (https=) | 2022-03-15 |
| JP2019518026A5 true JP2019518026A5 (https=) | 2022-03-15 |
| JP7054528B2 JP7054528B2 (ja) | 2022-04-14 |
Family
ID=60477983
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018563619A Active JP7054528B2 (ja) | 2016-06-01 | 2017-06-01 | プロテインキナーゼ活性を抑制する化合物の結晶形態、及びその適用 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US10899744B2 (https=) |
| EP (1) | EP3470410B1 (https=) |
| JP (1) | JP7054528B2 (https=) |
| KR (1) | KR102466958B1 (https=) |
| CN (1) | CN109195964B (https=) |
| AU (1) | AU2017274110B2 (https=) |
| CA (1) | CA3026142C (https=) |
| EA (1) | EA201892687A1 (https=) |
| ES (1) | ES2981015T3 (https=) |
| IL (1) | IL263356B (https=) |
| MY (1) | MY188379A (https=) |
| PH (1) | PH12018502529A1 (https=) |
| PL (1) | PL3470410T3 (https=) |
| RU (1) | RU2744264C2 (https=) |
| SG (1) | SG11201810800VA (https=) |
| TW (1) | TWI646094B (https=) |
| WO (1) | WO2017206924A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL279579B2 (en) | 2018-06-21 | 2023-02-01 | Betta Pharmaceuticals Co Ltd | Crystalline form of a compound to inhibit the activity of cdk4/6 and its use |
| EP4188922A1 (en) | 2020-08-03 | 2023-06-07 | Teva Pharmaceuticals International GmbH | Solid state forms of ensartinib and ensartinib salts |
| EP4385510A4 (en) * | 2021-08-10 | 2025-08-20 | Betta Pharmaceuticals Co Ltd | USE OF ENSARTINIB OR A CORRESPONDING SALT IN THE TREATMENT OF A DISEASE CARRYING A MET EXON 14 SKIPPING MUTATION |
| KR102851417B1 (ko) * | 2022-08-16 | 2025-08-28 | 제이투에이치바이오텍 (주) | 피리미딘-4-카복사마이드 화합물의 결정형 및 이를 포함하는 경구용 약학 제제 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL358271A1 (pl) * | 2000-03-06 | 2004-08-09 | Warner-Lambert Company | 5-alkilopirydo[2,3-D]pirymidyny jako inhibitory kinazy tyrozyny |
| CA2517256C (en) * | 2003-02-26 | 2013-04-30 | Sugen, Inc. | Aminoheteroaryl compounds as protein kinase inhibitors |
| US8414489B2 (en) | 2003-11-13 | 2013-04-09 | Medtronic Minimed, Inc. | Fabrication of multi-sensor arrays |
| ME01309B (me) * | 2004-08-26 | 2013-12-20 | Pfizer | Pirazolom supstituirani heteroarilni spojevi kao inhibitori proteinskih kinaza |
| BRPI0514687A (pt) | 2004-08-26 | 2008-06-17 | Pfizer | compostos amino heteroarila como inibidores de proteìna tirosina cinase |
| KR101146852B1 (ko) * | 2005-12-05 | 2012-05-16 | 화이자 프로덕츠 인크. | Ｃ?ｍｅｔ／ｈｇｆｒ 억제제의 다형체 |
| CN101652068A (zh) * | 2007-01-19 | 2010-02-17 | 艾科睿制药公司 | 激酶抑制物化合物 |
| ES2670665T3 (es) * | 2008-06-19 | 2018-05-31 | Xcovery Holding Company Llc | Compuestos de piridazina carboxamida sustituidos como compuestos inhibidores de quinasa |
| EA024809B1 (ru) * | 2010-10-08 | 2016-10-31 | Икскавери Холдинг Кампани, Ллс | Замещенные соединения пиридазинкарбоксамида |
| WO2012048258A2 (en) * | 2010-10-08 | 2012-04-12 | Xcovery Holding Company, Llc | Substituted pyridazine carboxamide compounds as kinase inhibitor compounds |
-
2017
- 2017-05-31 TW TW106117900A patent/TWI646094B/zh active
- 2017-06-01 WO PCT/CN2017/086760 patent/WO2017206924A1/zh not_active Ceased
- 2017-06-01 PL PL17805869.9T patent/PL3470410T3/pl unknown
- 2017-06-01 ES ES17805869T patent/ES2981015T3/es active Active
- 2017-06-01 KR KR1020187038142A patent/KR102466958B1/ko active Active
- 2017-06-01 IL IL263356A patent/IL263356B/en unknown
- 2017-06-01 EP EP17805869.9A patent/EP3470410B1/en active Active
- 2017-06-01 SG SG11201810800VA patent/SG11201810800VA/en unknown
- 2017-06-01 CN CN201780006852.3A patent/CN109195964B/zh active Active
- 2017-06-01 JP JP2018563619A patent/JP7054528B2/ja active Active
- 2017-06-01 MY MYPI2018002245A patent/MY188379A/en unknown
- 2017-06-01 CA CA3026142A patent/CA3026142C/en active Active
- 2017-06-01 US US16/306,104 patent/US10899744B2/en active Active
- 2017-06-01 RU RU2018145183A patent/RU2744264C2/ru active
- 2017-06-01 EA EA201892687A patent/EA201892687A1/ru unknown
- 2017-06-01 AU AU2017274110A patent/AU2017274110B2/en active Active
-
2018
- 2018-11-29 PH PH12018502529A patent/PH12018502529A1/en unknown
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