JP2018529703A - Ｎ−（１，３，４−オキサジアゾール−２−イル）アリールカルボキサミド類を合成する方法 - Google Patents

Ｎ−（１，３，４−オキサジアゾール−２−イル）アリールカルボキサミド類を合成する方法 Download PDF

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Publication number
JP2018529703A
JP2018529703A JP2018515819A JP2018515819A JP2018529703A JP 2018529703 A JP2018529703 A JP 2018529703A JP 2018515819 A JP2018515819 A JP 2018515819A JP 2018515819 A JP2018515819 A JP 2018515819A JP 2018529703 A JP2018529703 A JP 2018529703A
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JP
Japan
Prior art keywords
methyl
formula
alkyl
iii
represented
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2018515819A
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English (en)
Japanese (ja)
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JP2018529703A5 (enExample
Inventor
フンケ，クリスティアン
ネーフ，アルント
パツエノク，セルギー
ルイ，ノルベルト
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Bayer CropScience AG
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Bayer CropScience AG
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Publication date
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Publication of JP2018529703A publication Critical patent/JP2018529703A/ja
Publication of JP2018529703A5 publication Critical patent/JP2018529703A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/113—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/582—Recycling of unreacted starting or intermediate materials

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Laminated Bodies (AREA)
  • Shaping By String And By Release Of Stress In Plastics And The Like (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
JP2018515819A 2015-09-28 2016-09-23 Ｎ−（１，３，４−オキサジアゾール−２−イル）アリールカルボキサミド類を合成する方法 Pending JP2018529703A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15187023.5 2015-09-28
EP15187023 2015-09-28
PCT/EP2016/072629 WO2017055175A1 (de) 2015-09-28 2016-09-23 Verfahren zur herstellung von n-(1,3,4-oxadiazol-2-yl)arylcarboxamiden

Publications (2)

Publication Number Publication Date
JP2018529703A true JP2018529703A (ja) 2018-10-11
JP2018529703A5 JP2018529703A5 (enExample) 2019-10-31

Family

ID=54207378

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018515819A Pending JP2018529703A (ja) 2015-09-28 2016-09-23 Ｎ−（１，３，４−オキサジアゾール−２−イル）アリールカルボキサミド類を合成する方法

Country Status (10)

Country Link
US (1) US10189800B2 (enExample)
EP (1) EP3356336A1 (enExample)
JP (1) JP2018529703A (enExample)
KR (1) KR20180059456A (enExample)
CN (1) CN108137519A (enExample)
BR (1) BR112018006202A2 (enExample)
IL (1) IL258320B (enExample)
MX (1) MX2018003963A (enExample)
TW (1) TW201711566A (enExample)
WO (1) WO2017055175A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018202535A1 (de) * 2017-05-04 2018-11-08 Bayer Cropscience Aktiengesellschaft Herbizid wirksame 4-difluormethylbenzoylamide
KR102868734B1 (ko) * 2020-12-17 2025-10-02 주식회사 팜한농 N-(1-메틸-1h-테트라졸-5-일)-2-(((2-메틸-2h-테트라졸-5-일)메톡시)메틸)-6-(트리플루오로메틸)니코틴아마이드의 제조 방법

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009091267A (ja) * 2007-10-04 2009-04-30 Kyorin Pharmaceut Co Ltd アミド誘導体及びそれらを有効成分とするスフィンゴシン−１−リン酸−１（ｓ１ｐ１）受容体選択的アゴニスト
JP2012519730A (ja) * 2009-07-06 2012-08-30 アケビア セラピューティクス インコーポレイテッド がん細胞の転移を予防するための化合物、組成物および方法
JP2014510088A (ja) * 2011-03-22 2014-04-24 バイエル・インテレクチユアル・プロパテイー・ゲー・エム・ベー・ハー Ｎ−（１，３，４−オキサジアゾール−２−イル）アリールカルボキサミドおよび除草剤としてのその使用
WO2014114779A1 (en) * 2013-01-28 2014-07-31 H. Lundbeck A/S N-substituted-5-substituted phthalamic acids as sortilin inhibitors
WO2015137216A1 (ja) * 2014-03-10 2015-09-17 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 ２－アシルイミノピリジン誘導体の製造法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040077690A1 (en) * 2000-09-29 2004-04-22 Bing-Yan Zhu Quaternary amidino based inhibitors of factor xa
US20080090834A1 (en) * 2006-07-06 2008-04-17 Pfizer Inc Selective azole pde10a inhibitor compounds
JP5805767B2 (ja) * 2010-09-01 2015-11-10 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ Ｎ−（テトラゾール−５−イル）アリールカルボキサミド類及びｎ−（トリアゾール−５−イル）アリールカルボキサミド類並びに除草剤としてのそれらの使用
CN103443107B (zh) * 2011-03-28 2016-04-20 弗·哈夫曼-拉罗切有限公司 噻唑并嘧啶化合物
JP6001048B2 (ja) * 2011-03-28 2016-10-05 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ チアゾロピリミジン化合物
AU2012331283A1 (en) * 2011-11-03 2014-05-22 Bayer Intellectual Property Gmbh Herbicidally active oxime-ether-substituted benzoylamides
CN102491971B (zh) * 2011-12-19 2017-03-01 北京理工大学 手性[(4-甲基-2-丙基-1h-苯并咪唑-6-酰胺)-1-基]甲基联苯类化合物及其制备方法和用途
EP2817296B1 (de) 2012-02-21 2016-08-31 Bayer Intellectual Property GmbH Herbizid wirksame 3-(sulfin-/sulfonimidoyl)-benzamide

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009091267A (ja) * 2007-10-04 2009-04-30 Kyorin Pharmaceut Co Ltd アミド誘導体及びそれらを有効成分とするスフィンゴシン−１−リン酸−１（ｓ１ｐ１）受容体選択的アゴニスト
JP2012519730A (ja) * 2009-07-06 2012-08-30 アケビア セラピューティクス インコーポレイテッド がん細胞の転移を予防するための化合物、組成物および方法
JP2014510088A (ja) * 2011-03-22 2014-04-24 バイエル・インテレクチユアル・プロパテイー・ゲー・エム・ベー・ハー Ｎ−（１，３，４−オキサジアゾール−２−イル）アリールカルボキサミドおよび除草剤としてのその使用
WO2014114779A1 (en) * 2013-01-28 2014-07-31 H. Lundbeck A/S N-substituted-5-substituted phthalamic acids as sortilin inhibitors
WO2015137216A1 (ja) * 2014-03-10 2015-09-17 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 ２－アシルイミノピリジン誘導体の製造法

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
HIGASHI, FUKUJI ET AL, J.POLYM.SCI.POLYM.CHEM.ED., vol. 24, JPN6020032860, 1986, pages 187 - 189, ISSN: 0004336753 *

Also Published As

Publication number Publication date
TW201711566A (zh) 2017-04-01
US20180273496A1 (en) 2018-09-27
BR112018006202A2 (pt) 2018-10-09
US10189800B2 (en) 2019-01-29
KR20180059456A (ko) 2018-06-04
IL258320B (en) 2019-09-26
CN108137519A (zh) 2018-06-08
WO2017055175A1 (de) 2017-04-06
EP3356336A1 (de) 2018-08-08
IL258320A (en) 2018-05-31
MX2018003963A (es) 2018-06-08

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