JP2018522929A5 - - Google Patents

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Publication number
JP2018522929A5
JP2018522929A5 JP2018507023A JP2018507023A JP2018522929A5 JP 2018522929 A5 JP2018522929 A5 JP 2018522929A5 JP 2018507023 A JP2018507023 A JP 2018507023A JP 2018507023 A JP2018507023 A JP 2018507023A JP 2018522929 A5 JP2018522929 A5 JP 2018522929A5
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JP
Japan
Prior art keywords
methyl
oxaspiro
methoxy
carboxylate
octane
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
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JP2018507023A
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English (en)
Japanese (ja)
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JP2018522929A (ja
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Publication date
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Priority claimed from PCT/US2016/046511 external-priority patent/WO2017027684A1/en
Publication of JP2018522929A publication Critical patent/JP2018522929A/ja
Publication of JP2018522929A5 publication Critical patent/JP2018522929A5/ja
Withdrawn legal-status Critical Current

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JP2018507023A 2015-08-11 2016-08-11 フマギロール複素環化合物ならびにその作製および使用方法 Withdrawn JP2018522929A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562203742P 2015-08-11 2015-08-11
US62/203,742 2015-08-11
PCT/US2016/046511 WO2017027684A1 (en) 2015-08-11 2016-08-11 Fumagillol heterocyclic compounds and methods of making and using same

Publications (2)

Publication Number Publication Date
JP2018522929A JP2018522929A (ja) 2018-08-16
JP2018522929A5 true JP2018522929A5 (https=) 2019-08-29

Family

ID=56799580

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018507023A Withdrawn JP2018522929A (ja) 2015-08-11 2016-08-11 フマギロール複素環化合物ならびにその作製および使用方法

Country Status (15)

Country Link
US (5) US20180230137A1 (https=)
EP (1) EP3334728A1 (https=)
JP (1) JP2018522929A (https=)
KR (1) KR20180035907A (https=)
CN (1) CN108026085A (https=)
AR (1) AR105671A1 (https=)
AU (1) AU2016306558A1 (https=)
CA (1) CA2995366A1 (https=)
EA (1) EA201890449A1 (https=)
IL (1) IL257443A (https=)
MA (1) MA42612A (https=)
MX (1) MX2018001733A (https=)
PH (1) PH12018500315A1 (https=)
TW (1) TW201718550A (https=)
WO (1) WO2017027684A1 (https=)

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* Cited by examiner, † Cited by third party
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CN106432255A (zh) 2015-08-11 2017-02-22 扎夫根公司 烟曲霉素醇螺环化合物和制备和使用其的方法
WO2018148638A1 (en) * 2017-02-10 2018-08-16 Zafgen, Inc. Pharmaceutical compositions of metap-2 inhibitors
WO2019118612A1 (en) * 2017-12-12 2019-06-20 Zafgen, Inc. Targeting compounds
WO2019173505A1 (en) * 2018-03-06 2019-09-12 Zafgen, Inc. Methods of treating disorders related to glycemic control
CN109180551A (zh) * 2018-07-17 2019-01-11 宜春学院 一种四元氮杂环中间体的制备方法
CN113453721B (zh) 2018-10-26 2025-09-16 辛德弗雷克斯公司 Metap2抑制剂的生物标志物及其应用
CN111606836B (zh) * 2020-06-12 2021-01-15 上海馨远医药科技有限公司 一种R-N-Boc-3-吡咯烷乙酸的制备方法
GB202011996D0 (en) 2020-07-31 2020-09-16 Adorx Therapeutics Ltd Antagonist compounds

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