JP2018515550A5 - - Google Patents

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Publication number
JP2018515550A5
JP2018515550A5 JP2017560135A JP2017560135A JP2018515550A5 JP 2018515550 A5 JP2018515550 A5 JP 2018515550A5 JP 2017560135 A JP2017560135 A JP 2017560135A JP 2017560135 A JP2017560135 A JP 2017560135A JP 2018515550 A5 JP2018515550 A5 JP 2018515550A5
Authority
JP
Japan
Prior art keywords
alkyl
hydrazinocarbonyl
pyridin
chloro
methylbenzoyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2017560135A
Other languages
English (en)
Japanese (ja)
Other versions
JP2018515550A (ja
JP6689887B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IN2016/050142 external-priority patent/WO2016185490A1/en
Publication of JP2018515550A publication Critical patent/JP2018515550A/ja
Publication of JP2018515550A5 publication Critical patent/JP2018515550A5/ja
Application granted granted Critical
Publication of JP6689887B2 publication Critical patent/JP6689887B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2017560135A 2015-05-18 2016-05-18 新規アミドヘテロアリールアロイルヒドラジドエチン Expired - Fee Related JP6689887B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN1953MU2015 2015-05-18
IN1953/MUM/2015 2015-05-18
PCT/IN2016/050142 WO2016185490A1 (en) 2015-05-18 2016-05-18 Novel amidoheteroaryl aroyl hydrazide ethynes

Publications (3)

Publication Number Publication Date
JP2018515550A JP2018515550A (ja) 2018-06-14
JP2018515550A5 true JP2018515550A5 (https=) 2019-05-09
JP6689887B2 JP6689887B2 (ja) 2020-04-28

Family

ID=57319598

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017560135A Expired - Fee Related JP6689887B2 (ja) 2015-05-18 2016-05-18 新規アミドヘテロアリールアロイルヒドラジドエチン

Country Status (13)

Country Link
US (1) US10150733B2 (https=)
EP (1) EP3297991B1 (https=)
JP (1) JP6689887B2 (https=)
KR (1) KR20180011772A (https=)
CN (1) CN107709300A (https=)
AU (1) AU2016263311A1 (https=)
BR (1) BR112017024633A2 (https=)
CA (1) CA2985161A1 (https=)
EA (1) EA032697B1 (https=)
ES (1) ES2774501T3 (https=)
MX (1) MX2017014752A (https=)
WO (1) WO2016185490A1 (https=)
ZA (1) ZA201707664B (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11201810294QA (en) 2016-06-02 2018-12-28 Sun Pharma Advanced Res Co Ltd Treatment for parkinson's disease
EA037697B1 (ru) * 2016-06-02 2021-05-12 Сан Фарма Адвансед Ресёрч Компани Лимитед Лечение болезни паркинсона
RU2768887C2 (ru) * 2017-03-15 2022-03-25 Сан Фарма Эдвансд Рисёч Компани Лимитед Новая аморфная дисперсия (5-{ 5-[n'-(2-хлор-6-метилбензоил)гидразинокарбонил]-2-метил-фенилэтинил} -пиридин-2-ил)амида циклопропанкарбоновой кислоты
CN113292537B (zh) 2018-06-15 2024-04-05 汉达癌症医药责任有限公司 激酶抑制剂的盐类及其组合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2007249924B2 (en) * 2006-05-08 2013-07-04 Ariad Pharmaceuticals, Inc. Acetylenic heteroaryl compounds
WO2012089106A1 (zh) * 2010-12-27 2012-07-05 Sun Shuping 作为蛋白激酶抑制剂的芳炔类衍生物及其医疗用途
CN103502217B (zh) * 2011-01-21 2015-11-25 太阳医药高级研究有限公司 包含酪氨酸激酶抑制剂的二芳基乙炔酰肼
US8859541B2 (en) * 2012-02-27 2014-10-14 Boehringer Ingelheim International Gmbh 6-alkynylpyridines

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