JP2009534358A5 - - Google Patents

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Publication number
JP2009534358A5
JP2009534358A5 JP2009505894A JP2009505894A JP2009534358A5 JP 2009534358 A5 JP2009534358 A5 JP 2009534358A5 JP 2009505894 A JP2009505894 A JP 2009505894A JP 2009505894 A JP2009505894 A JP 2009505894A JP 2009534358 A5 JP2009534358 A5 JP 2009534358A5
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JP
Japan
Prior art keywords
alkyl
optionally
group
substituted
nitrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2009505894A
Other languages
English (en)
Japanese (ja)
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JP2009534358A (ja
Filing date
Publication date
Priority claimed from GBGB0607944.6A external-priority patent/GB0607944D0/en
Application filed filed Critical
Publication of JP2009534358A publication Critical patent/JP2009534358A/ja
Publication of JP2009534358A5 publication Critical patent/JP2009534358A5/ja
Pending legal-status Critical Current

Links

JP2009505894A 2006-04-21 2007-04-19 アデノシンａ３受容体アゴニスト Pending JP2009534358A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0607944.6A GB0607944D0 (en) 2006-04-21 2006-04-21 Organic compounds
PCT/EP2007/053847 WO2007147659A1 (en) 2006-04-21 2007-04-19 Adenosine a3 receptor agonists

Publications (2)

Publication Number Publication Date
JP2009534358A JP2009534358A (ja) 2009-09-24
JP2009534358A5 true JP2009534358A5 (https=) 2011-03-10

Family

ID=36581041

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009505894A Pending JP2009534358A (ja) 2006-04-21 2007-04-19 アデノシンａ３受容体アゴニスト

Country Status (12)

Country Link
US (1) US20090281126A1 (https=)
EP (1) EP2013199A1 (https=)
JP (1) JP2009534358A (https=)
KR (1) KR20080110845A (https=)
CN (1) CN101426785A (https=)
AU (1) AU2007263237B2 (https=)
BR (1) BRPI0710514A2 (https=)
CA (1) CA2649648A1 (https=)
GB (1) GB0607944D0 (https=)
MX (1) MX2008013520A (https=)
RU (1) RU2008145708A (https=)
WO (1) WO2007147659A1 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500281A (es) * 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
GB0500785D0 (en) * 2005-01-14 2005-02-23 Novartis Ag Organic compounds
GB0607945D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607950D0 (en) 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607953D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607948D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
PT2322525E (pt) 2006-04-21 2013-12-26 Novartis Ag Derivados de purina para utilização como agonistas do recetor de adenosina a2a
GB0607954D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
EP1889846A1 (en) 2006-07-13 2008-02-20 Novartis AG Purine derivatives as A2a agonists
EP1903044A1 (en) 2006-09-14 2008-03-26 Novartis AG Adenosine Derivatives as A2A Receptor Agonists
CN101553459A (zh) * 2006-11-10 2009-10-07 诺瓦提斯公司 环戊烯二醇单乙酸酯衍生物
BRPI0818578A2 (pt) * 2007-10-17 2015-07-21 Novartis Ag Derivados de purina como ligantes receptores de adenosina a1
AU2009231978C1 (en) 2008-03-31 2014-01-30 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Purine derivatives as A3 adenosine receptor- selective agonists
US8916570B2 (en) 2008-03-31 2014-12-23 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services A3 adenosine receptor agonists and antagonists
EP2331542B1 (en) 2008-08-01 2016-07-27 The United States of America, as Represented by The Secretary, Department of Health and Human Services A3 adenosine receptor antagonists and partial agonists
US9181253B2 (en) 2008-08-01 2015-11-10 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Adenosine receptor agonists, partial agonists, and antagonists

Family Cites Families (39)

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JP2000502709A (ja) * 1996-01-02 2000-03-07 ローヌ―プーラン ローラー ファーマシューティカルズ インコーポレイテッド ２，４―ジヒドロキシピリジン及び２，４―ジヒドロキシ―３―ニトロピリジンの製造方法
US6376472B1 (en) * 1996-07-08 2002-04-23 Aventis Pharmaceuticals, Inc. Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties
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US6586413B2 (en) * 1999-11-05 2003-07-01 The United States Of America As Represented By The Department Of Health And Human Services Methods and compositions for reducing ischemic injury of the heart by administering adenosine receptor agonists and antagonists
US7589075B2 (en) * 2001-01-16 2009-09-15 Can-Fite Biopharma Ltd. Use of an adenosine A3 receptor agonist for inhibition of viral replication
US20040162422A1 (en) * 2001-03-20 2004-08-19 Adrian Hall Chemical compounds
EP1258247A1 (en) * 2001-05-14 2002-11-20 Aventis Pharma Deutschland GmbH Adenosine analogues for the treatment of insulin resistance syndrome and diabetes
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JP2007517019A (ja) * 2003-12-29 2007-06-28 カン−フィテ・バイオファーマ・リミテッド 多発性硬化症の治療方法
PL1778239T3 (pl) * 2004-07-28 2014-01-31 Can Fite Biopharma Ltd Agoniści receptora adenozynowego A3 do leczenia zaburzeń suchego oka w tym zespołu Sjogrena
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GT200500281A (es) * 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
US7176172B2 (en) * 2004-10-25 2007-02-13 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Quaternary ammonium polyol salts as anti-aging actives in personal care compositions
US20080051364A1 (en) * 2004-11-08 2008-02-28 Pninna Fishman Therapeutic Treatment of Accelerated Bone Resorption
GB0500785D0 (en) * 2005-01-14 2005-02-23 Novartis Ag Organic compounds
PT1848718E (pt) * 2005-02-04 2012-10-11 Millennium Pharm Inc Inibidores de enzimas de activação e1
EP1959939B1 (en) * 2005-11-30 2012-01-11 Can-Fite Biopharma Ltd. Use of a3 adenosine receptor agonist in osteoarthritis treatment
EP1983990B1 (en) * 2006-01-26 2011-03-23 Government of the United States of America, Represented by the Secretary, Department of Health and Human Services A3 adenosine receptor allosteric modulators
KR101450535B1 (ko) * 2006-02-02 2014-10-14 밀레니엄 파머슈티컬스 인코퍼레이티드 Ｅ１ 활성화 효소의 억제제
GB0607945D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607951D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607954D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
PT2322525E (pt) * 2006-04-21 2013-12-26 Novartis Ag Derivados de purina para utilização como agonistas do recetor de adenosina a2a
GB0607950D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607948D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
EP1889846A1 (en) * 2006-07-13 2008-02-20 Novartis AG Purine derivatives as A2a agonists
US8008307B2 (en) * 2006-08-08 2011-08-30 Millennium Pharmaceuticals, Inc. Heteroaryl compounds useful as inhibitors of E1 activating enzymes
EP1903044A1 (en) * 2006-09-14 2008-03-26 Novartis AG Adenosine Derivatives as A2A Receptor Agonists
CN101553459A (zh) * 2006-11-10 2009-10-07 诺瓦提斯公司 环戊烯二醇单乙酸酯衍生物
BRPI0818578A2 (pt) * 2007-10-17 2015-07-21 Novartis Ag Derivados de purina como ligantes receptores de adenosina a1
US20090181934A1 (en) * 2007-10-17 2009-07-16 Novartis Ag Organic Compounds

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