JP2016500653A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2016500653A5 JP2016500653A5 JP2015533704A JP2015533704A JP2016500653A5 JP 2016500653 A5 JP2016500653 A5 JP 2016500653A5 JP 2015533704 A JP2015533704 A JP 2015533704A JP 2015533704 A JP2015533704 A JP 2015533704A JP 2016500653 A5 JP2016500653 A5 JP 2016500653A5
- Authority
- JP
- Japan
- Prior art keywords
- meleu
- leu
- methyl
- methylamino
- meval
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- CCHDRLLWDRWYAN-QMMMGPOBSA-N CC(C)C[C@@H](C(C)=O)N=C Chemical compound CC(C)C[C@@H](C(C)=O)N=C CCHDRLLWDRWYAN-QMMMGPOBSA-N 0.000 description 1
- 0 CC(C)C[C@@](C(C)=*)NC Chemical compound CC(C)C[C@@](C(C)=*)NC 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB1217560.0A GB201217560D0 (en) | 2012-10-02 | 2012-10-02 | Novel cyclic depsipeptide compounds and their uses |
| GB1217560.0 | 2012-10-02 | ||
| PCT/GB2013/052570 WO2014053834A1 (en) | 2012-10-02 | 2013-10-02 | Cyclic depsipeptide compounds and their uses |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2016500653A JP2016500653A (ja) | 2016-01-14 |
| JP2016500653A5 true JP2016500653A5 (https=) | 2016-10-06 |
| JP6263541B2 JP6263541B2 (ja) | 2018-01-17 |
Family
ID=47225510
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015533704A Expired - Fee Related JP6263541B2 (ja) | 2012-10-02 | 2013-10-02 | 環状デプシペプチド化合物およびそれらの用途 |
Country Status (8)
| Country | Link |
|---|---|
| US (3) | US9382295B2 (https=) |
| EP (1) | EP2904001A1 (https=) |
| JP (1) | JP6263541B2 (https=) |
| CN (1) | CN104768968B (https=) |
| AU (1) | AU2013326231B2 (https=) |
| CA (1) | CA2885940A1 (https=) |
| GB (1) | GB201217560D0 (https=) |
| WO (1) | WO2014053834A1 (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9914755B2 (en) | 2015-01-08 | 2018-03-13 | Allergan, Inc. | Cyclosporin derivatives wherein the MeBmt sidechain has been cyclized |
| US11046730B2 (en) | 2016-04-15 | 2021-06-29 | The Regents Of The University Of California | Antimicrobial compositions |
| CN111449050A (zh) | 2019-01-20 | 2020-07-28 | 睿诺医疗科技（上海）有限公司 | 环孢菌素类似物及其用途 |
| CN109821020B (zh) * | 2019-01-28 | 2021-07-30 | 温州医科大学 | 一种制备干眼症药物的应用及治疗干眼症的方法 |
| CA3152922A1 (en) | 2019-10-12 | 2021-04-15 | Michael Peel | Treatment and prevention of nephrotoxin-induced kidney injuries |
| PE20221323A1 (es) * | 2019-11-07 | 2022-09-09 | Chugai Pharmaceutical Co Ltd | Compuesto de peptidos ciclicos que tiene accion inhibidora de kras |
| IL296586B1 (en) | 2020-03-26 | 2026-04-01 | Farsight Medical Tech Shanghai Co Ltd | Cyclophilin inhibitors and their uses |
| US12465629B2 (en) | 2020-04-15 | 2025-11-11 | Farsight Medical Technology (Shanghai) Co., Ltd. | Prevention and treatment of organ injuries |
| CN121824695A (zh) * | 2022-06-24 | 2026-04-10 | 中国农业科学院生物技术研究所 | 一种抗寄生虫环肽及其应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0296123B1 (en) * | 1987-06-19 | 1994-08-31 | Sandoz Ag | Cyclic peptolides |
| US5595756A (en) * | 1993-12-22 | 1997-01-21 | Inex Pharmaceuticals Corporation | Liposomal compositions for enhanced retention of bioactive agents |
| PT1853296E (pt) | 2005-01-10 | 2012-09-26 | Debiopharm Sa | Utilização de um undecapeptídeo cíclico para a preparação de um medicamento para administração em situações de miocardia isquêmica |
| AU2009312535B2 (en) * | 2008-11-06 | 2015-03-26 | Debio Recherche Pharmaceutique S.A. | Cycloundecadepsipeptide compounds and use of said compounds as a medicament |
| US8623814B2 (en) | 2010-02-23 | 2014-01-07 | Enanta Pharmaceuticals, Inc. | Antiviral agents |
| WO2011141891A1 (en) | 2010-05-12 | 2011-11-17 | Debio Recherche Pharmaceutique S.A. | Use of cycloundecadepsipeptide compounds |
-
2012
- 2012-10-02 GB GBGB1217560.0A patent/GB201217560D0/en not_active Ceased
-
2013
- 2013-10-02 JP JP2015533704A patent/JP6263541B2/ja not_active Expired - Fee Related
- 2013-10-02 AU AU2013326231A patent/AU2013326231B2/en not_active Ceased
- 2013-10-02 EP EP13771583.5A patent/EP2904001A1/en not_active Withdrawn
- 2013-10-02 US US14/433,327 patent/US9382295B2/en not_active Expired - Fee Related
- 2013-10-02 WO PCT/GB2013/052570 patent/WO2014053834A1/en not_active Ceased
- 2013-10-02 CN CN201380056072.1A patent/CN104768968B/zh not_active Expired - Fee Related
- 2013-10-02 CA CA2885940A patent/CA2885940A1/en not_active Abandoned
-
2016
- 2016-06-20 US US15/187,039 patent/US9895412B2/en not_active Expired - Fee Related
-
2018
- 2018-01-29 US US15/882,510 patent/US20180153958A1/en not_active Abandoned
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2016500653A5 (https=) | ||
| EA200970656A1 (ru) | Вич-ингибирующие 5,6-замещенные пиримидины | |
| AR059622A1 (es) | Quinolonas utiles como inhibidores de la sintetasa del oxido nitrico inducibles | |
| JP2013530176A5 (https=) | ||
| JP2018537413A5 (ja) | 化合物、医薬的に許容される塩又はその立体異性体及び医薬組成物 | |
| JP2012140432A5 (https=) | ||
| JP2013537203A5 (https=) | ||
| ES2640911T3 (es) | Cicloalquilnitrilpirazolcarboxamidas como inhibidores de la quinasa Janus | |
| JP2019513778A5 (https=) | ||
| WO2011004162A3 (en) | 1, 2, 4-thiazolidin-3-one derivatives and their use in the treatment of cancer | |
| JP2012523457A5 (https=) | ||
| HUP0401784A2 (hu) | Heterobiciklikus szerkezetû virális polimeráz inhibitorok, eljárás az elõállításukra, köztitermékek és ezeket tartalmazó gyógyszerkészítmények | |
| WO2010089510A3 (fr) | Dérivés d'azaspiranyl-alkylcarbamates d'hétérocycles à 5 chaînons, leur préparation et leur application en thérapeutique | |
| AR081587A1 (es) | DERIVADOS DE 5,6-DIHIDRO-2H-[1,4]OXAZIN-3-IL-AMINA UTILES COMO INHIBIDORES DE LA b-SECRETASA (BACE) | |
| JP2011219498A5 (https=) | ||
| JP2013509392A5 (https=) | ||
| SMT201300085B (it) | Composti di pirrolo | |
| AR057915A1 (es) | Compuesto con estructura de cinamida de dos ciclos con actividad inhibitoria de la produccion de abeta40 y abeta42, un agente farmaceutico que lo comprende y el uso de este en el tratamiento de enfermedades mentales y neurodegenerativas. | |
| RU2017123114A (ru) | 3-оксо-3-(ариламино)пропионаты, способ их получения и их применение в получении пирролидинонов | |
| MX2013004407A (es) | Derivado de piridina y agente medicinal. | |
| MX2009008509A (es) | Compuesto de anillo puenteado-aza. | |
| AR085615A1 (es) | Derivados de fluoropiridinona utiles como agentes antibacterianos y composiciones farmaceuticas que los contienen | |
| JP2015537008A5 (https=) | ||
| WO2008126901A1 (ja) | 含窒素複素環化合物およびそれを含有する医薬組成物 | |
| DK2868660T3 (da) | Anti-tumoreffekt-potentiator omfattende en imidazooxazin-forbindelse |