JP2017531039A5 - - Google Patents

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Publication number
JP2017531039A5
JP2017531039A5 JP2017538467A JP2017538467A JP2017531039A5 JP 2017531039 A5 JP2017531039 A5 JP 2017531039A5 JP 2017538467 A JP2017538467 A JP 2017538467A JP 2017538467 A JP2017538467 A JP 2017538467A JP 2017531039 A5 JP2017531039 A5 JP 2017531039A5
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JP
Japan
Prior art keywords
dihydro
thieno
azaspiro
oxa
carboxamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2017538467A
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English (en)
Japanese (ja)
Other versions
JP2017531039A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/GB2015/052945 external-priority patent/WO2016055792A1/en
Publication of JP2017531039A publication Critical patent/JP2017531039A/ja
Publication of JP2017531039A5 publication Critical patent/JP2017531039A5/ja
Withdrawn legal-status Critical Current

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JP2017538467A 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体 Withdrawn JP2017531039A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14188494 2014-10-10
EP14188494.0 2014-10-10
PCT/GB2015/052945 WO2016055792A1 (en) 2014-10-10 2015-10-08 Novel 5,6-dihydro-4h-benzo[b]thieno-[2,3-d]azepine derivatives

Publications (2)

Publication Number Publication Date
JP2017531039A JP2017531039A (ja) 2017-10-19
JP2017531039A5 true JP2017531039A5 (show.php) 2018-11-22

Family

ID=51842340

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2017538467A Withdrawn JP2017531039A (ja) 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体
JP2017538466A Active JP6675407B2 (ja) 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2017538466A Active JP6675407B2 (ja) 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体

Country Status (13)

Country Link
US (6) US9732098B2 (show.php)
EP (2) EP3204389B1 (show.php)
JP (2) JP2017531039A (show.php)
KR (1) KR20170058921A (show.php)
CN (1) CN106852144B (show.php)
AU (1) AU2015329789B2 (show.php)
BR (1) BR112017005104B1 (show.php)
CA (1) CA2957868C (show.php)
EA (1) EA201790796A8 (show.php)
IL (1) IL250823A0 (show.php)
MX (1) MX2017004652A (show.php)
SG (1) SG11201701184WA (show.php)
WO (2) WO2016055791A1 (show.php)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3204389B1 (en) 2014-10-10 2019-06-26 Pulmocide Limited Novel 5,6-dihydro-4h-benzo[b]thieno-[2,3-d]azepine derivative
JP6694886B2 (ja) 2014-12-18 2020-05-20 プルモシデ リミテド 4,5−ジヒドロ−6H−チエノ[3,2−d]ベンゾアゼピン誘導体及び呼吸器合胞体ウイルス(RSV)感染を治療するためのその使用
MY197231A (en) 2015-07-22 2023-06-06 Enanta Pharm Inc Benzodiazepine derivatives as rsv inhibitors
US20170226129A1 (en) 2016-01-15 2017-08-10 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
ES2877808T3 (es) * 2016-02-03 2021-11-17 Janssen Sciences Ireland Unlimited Co Producto combinado para tratar o mejorar una infección por virus respiratorio sincicial
WO2017175000A1 (en) 2016-04-08 2017-10-12 Pulmocide Limited Compounds
US10398706B2 (en) 2017-01-06 2019-09-03 Enanta Pharmaceuticals, Inc. Heteroaryldiazepine derivatives as RSV inhibitors
NZ756805A (en) 2017-02-16 2025-10-31 Enanta Pharm Inc Processes for the preparation of benzodiazepine derivatives
WO2018226801A1 (en) 2017-06-07 2018-12-13 Enanta Pharmaceuticals, Inc. Aryldiazepine derivatives as rsv inhibitors
WO2019006291A1 (en) * 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
US11091501B2 (en) 2017-06-30 2021-08-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
BR112020006334A2 (pt) 2017-09-29 2020-09-24 Enanta Pharmaceuticals, Inc. combinação de agentes farmacêuticos como inibidores de rsv
EP3710009B1 (en) 2017-11-13 2025-07-30 Enanta Pharmaceuticals, Inc. Processes for the resolution of benzodiazepin-2-one and benzoazepin-2-one derivatives
US10647711B2 (en) 2017-11-13 2020-05-12 Enanta Pharmaceuticals, Inc. Azepin-2-one derivatives as RSV inhibitors
WO2019199908A1 (en) * 2018-04-11 2019-10-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
WO2020190935A1 (en) 2019-03-18 2020-09-24 Enanta Pharmaceuticals, Inc. Benzodiazepine derivatives as rsv inhibitors
WO2020210246A1 (en) * 2019-04-09 2020-10-15 Enanta Pharmaceuticals, Inc, Heterocyclic compounds as rsv inhibitors
JP7681009B2 (ja) 2019-10-04 2025-05-21 エナンタ ファーマシューティカルズ インコーポレイテッド 抗ウイルス性複素環化合物
US11505558B1 (en) 2019-10-04 2022-11-22 Enanta Pharmaceuticals, Inc. Antiviral heterocyclic compounds
UY39032A (es) 2020-01-24 2021-07-30 Enanta Pharm Inc Compuestos heterocíclicos como agentes antivirales
WO2022010882A1 (en) * 2020-07-07 2022-01-13 Enanta Pharmaceuticals, Inc, Dihydroquinoxaline and dihydropyridopyrazine derivatives as rsv inhibitors
US11945824B2 (en) 2020-10-19 2024-04-02 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as anti-viral agents
CA3173354A1 (en) 2021-02-26 2022-09-01 Adam SZYMANIAK A 2,3-dihydrofuro[2,3-c]pyridine-3-carboxamide compound and its antiviral use
AR129003A1 (es) 2022-04-07 2024-07-03 Enanta Pharm Inc Compuestos heterocíclicos antivirales
US12162857B2 (en) 2022-04-27 2024-12-10 Enanta Pharmaceuticals, Inc. Antiviral compounds

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5693635A (en) 1993-07-29 1997-12-02 American Cyanamid Company Tricyclic benzazepine vasopressin antagonists
PL351470A1 (en) 1999-04-28 2003-04-22 Aventis Pharma Gmbh Tri-aryl acid derivatives as ppar receptor ligands
EP2240029A4 (en) * 2008-01-07 2012-08-22 Synta Pharmaceuticals Corp COMPOUNDS FOR USE AGAINST INFLAMMATORY AND IMMUNOMIC DISEASES
US8999969B2 (en) 2009-07-09 2015-04-07 Gilead Sciences, Inc. Anti-RSV compounds
KR101804588B1 (ko) 2009-10-13 2017-12-04 리간드 파마슈티칼스 인코포레이티드 조혈 성장 인자 모방체 소분자 화합물 및 이의 용도
US8791136B2 (en) 2010-07-29 2014-07-29 Rigel Pharmaceuticals, Inc. Substituted pyridine, pyridazine, pyrazine and pyrimidine compounds and methods for using the same
WO2012129562A2 (en) 2011-03-24 2012-09-27 The Scripps Research Institute Compounds and methods for inducing chondrogenesis
RU2017106742A (ru) 2014-08-05 2018-09-06 Элиос Биофарма, Инк. Комбинированная терапия для лечения парамиксовируса
EP3204389B1 (en) * 2014-10-10 2019-06-26 Pulmocide Limited Novel 5,6-dihydro-4h-benzo[b]thieno-[2,3-d]azepine derivative
US20170226129A1 (en) 2016-01-15 2017-08-10 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
ES2877808T3 (es) 2016-02-03 2021-11-17 Janssen Sciences Ireland Unlimited Co Producto combinado para tratar o mejorar una infección por virus respiratorio sincicial
WO2019006291A1 (en) 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
US11091501B2 (en) 2017-06-30 2021-08-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors

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