JP2017505789A5 - - Google Patents
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- JP2017505789A5 JP2017505789A5 JP2016551215A JP2016551215A JP2017505789A5 JP 2017505789 A5 JP2017505789 A5 JP 2017505789A5 JP 2016551215 A JP2016551215 A JP 2016551215A JP 2016551215 A JP2016551215 A JP 2016551215A JP 2017505789 A5 JP2017505789 A5 JP 2017505789A5
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- Japan
- Prior art keywords
- aerosol formulation
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- sirolimus
- particles
- microns
- Prior art date
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201461938282P | 2014-02-11 | 2014-02-11 | |
| US61/938,282 | 2014-02-11 | ||
| US201462060970P | 2014-10-07 | 2014-10-07 | |
| US62/060,970 | 2014-10-07 | ||
| PCT/US2015/015266 WO2015123219A1 (en) | 2014-02-11 | 2015-02-10 | Rapamycin for the treatment of lymphangioleiomyomatosis |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2017505789A JP2017505789A (ja) | 2017-02-23 |
| JP2017505789A5 true JP2017505789A5 (https=) | 2020-01-23 |
Family
ID=52595442
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016551215A Pending JP2017505789A (ja) | 2014-02-11 | 2015-02-10 | リンパ脈管筋腫症の治療のためのラパマイシン |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20150265582A1 (https=) |
| EP (1) | EP3104891A1 (https=) |
| JP (1) | JP2017505789A (https=) |
| KR (1) | KR20160120739A (https=) |
| CN (1) | CN106573067A (https=) |
| AU (1) | AU2015217349A1 (https=) |
| BR (1) | BR112016018365A2 (https=) |
| CA (1) | CA2939342A1 (https=) |
| IL (1) | IL247155A0 (https=) |
| MX (1) | MX2016010373A (https=) |
| RU (1) | RU2016136348A (https=) |
| WO (1) | WO2015123219A1 (https=) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2014117035A1 (en) | 2013-01-24 | 2014-07-31 | Transderm, Inc. | COMPOSITIONS FOR TRANSDERMAL DELIVERY OF mTOR INHIBITORS |
| US10307370B2 (en) | 2013-10-08 | 2019-06-04 | AI Therapeutics, Inc. | Rapamycin for the treatment of lymphangioleiomyomatosis |
| US10307371B2 (en) | 2014-02-11 | 2019-06-04 | AI Therapeutics, Inc. | Rapamycin for the treatment of lymphangioleiomyomatosis |
| DK3125875T3 (da) | 2014-04-04 | 2023-07-24 | Ai Therapeutics Inc | Inhalerbar rapamycinformulering til behandling af aldersrelaterede tilstande |
| KR20170095807A (ko) * | 2014-10-07 | 2017-08-23 | 램 테라퓨틱스, 인코포레이티드 | 폐 고혈압의 치료를 위한 흡입가능 라파마이신 제제 |
| MA40910A (fr) * | 2014-11-07 | 2017-09-12 | Civitas Therapeutics Inc | Poudres de rapamycine pour administration pulmonaire |
| WO2016130645A1 (en) * | 2015-02-10 | 2016-08-18 | Lam Therapeutics, Inc. | Rapamycin for the treatment of lymphangioleiomyomatosis |
| US10383860B2 (en) * | 2015-07-28 | 2019-08-20 | Nippon Kayaku Kabushiki Kaisha | Pharmaceutical composition comprising rapamycin or derivative thereof, and method for producing the same |
| US11224594B2 (en) * | 2015-09-16 | 2022-01-18 | Philip Morris Products S.A. | Nicotine formulations and methods of making and using the same |
| GB201611639D0 (en) * | 2016-07-04 | 2016-08-17 | Ockham Biotech Ltd | Delivery device and formulation |
| JP7108631B2 (ja) | 2017-01-06 | 2022-07-28 | パルヴェラ セラピューティクス、インク． | ｍＴＯＲ阻害剤の無水組成物およびその使用方法 |
| PT110585B (pt) * | 2018-02-22 | 2021-04-22 | Hovione Farmaciencia Sa | Processo de produção contínua de partículas compreendendo secagem por atomização com preparação contínua da solução de atomização |
| US10350226B1 (en) * | 2018-06-27 | 2019-07-16 | Joshua O. Atiba | Therapy and prevention of prion protein complex infections |
| US11000513B2 (en) | 2018-07-02 | 2021-05-11 | Palvella Therapeutics, Inc. | Anhydrous compositions of mTOR inhibitors and methods of use |
| US20240009231A1 (en) * | 2020-09-25 | 2024-01-11 | University Of Cincinnati | Method for Pleurodesis and Delivery of Drugs to the Lung and Pleural Space |
| US12485133B2 (en) * | 2021-02-04 | 2025-12-02 | Hovione Scientia Limited | Inhaled ivermectin |
| CN114755421B (zh) * | 2022-04-07 | 2025-07-18 | 华中科技大学同济医学院附属同济医院 | 淋巴管平滑肌瘤病的蛋白质生物标志物及应用 |
| CN118615239B (zh) * | 2024-06-17 | 2025-07-22 | 明思未来(北京)科技发展有限公司 | 一种依维莫司眼局部给药制剂 |
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| US2517482A (en) * | 1949-04-09 | 1950-08-01 | Sharp & Dohme Inc | Inhaler |
| ZA737247B (en) | 1972-09-29 | 1975-04-30 | Ayerst Mckenna & Harrison | Rapamycin and process of preparation |
| US5080899A (en) | 1991-02-22 | 1992-01-14 | American Home Products Corporation | Method of treating pulmonary inflammation |
| AU688782B2 (en) * | 1993-09-30 | 1998-03-19 | Wyeth | Rapamycin formulations for oral administration |
| US5635161A (en) | 1995-06-07 | 1997-06-03 | Abbott Laboratories | Aerosol drug formulations containing vegetable oils |
| BE1009856A5 (fr) | 1995-07-14 | 1997-10-07 | Sandoz Sa | Composition pharmaceutique sous la forme d'une dispersion solide comprenant un macrolide et un vehicule. |
| GB9606452D0 (en) | 1996-03-27 | 1996-06-05 | Sandoz Ltd | Organic compounds |
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| US5989591A (en) | 1997-03-14 | 1999-11-23 | American Home Products Corporation | Rapamycin formulations for oral administration |
| US20040039047A1 (en) | 1998-08-11 | 2004-02-26 | Mark Zamoyski | Compositions and methods for treating lung cancers |
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| CA2457148A1 (en) | 2001-08-20 | 2003-02-27 | Transave, Inc. | Treatment of cancers by inhalation of stable platinum-containing formulations |
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| AU2003237863A1 (en) | 2002-05-20 | 2003-12-12 | Research Development Foundation | Aerosol drug inhibition of lung metastases |
| AR050374A1 (es) * | 2004-08-20 | 2006-10-18 | Wyeth Corp | Forma polimorfica de rafampicina |
| US20060094744A1 (en) | 2004-09-29 | 2006-05-04 | Maryanoff Cynthia A | Pharmaceutical dosage forms of stable amorphous rapamycin like compounds |
| AU2006222409A1 (en) | 2005-03-08 | 2006-09-14 | Lifecycle Pharma A/S | Pharmaceutical compositions comprising sirolimus and/or an analogue thereof |
| US20060210638A1 (en) * | 2005-03-17 | 2006-09-21 | Elan Pharma International Limited | Injectable compositions of nanoparticulate immunosuppressive compounds |
| CN1883474A (zh) * | 2005-06-22 | 2006-12-27 | 华北制药集团新药研究开发有限责任公司 | 一种含大环内酯类化合物和多孔水不溶性亲水性载体的组合物 |
| RU2008121713A (ru) * | 2005-12-20 | 2010-01-27 | Вайет (Us) | Контроль стабильности лекарственной формы cci-779 посредством контроля примесей лекарственныхого вещества |
| LT1983984T (lt) | 2006-02-02 | 2018-06-11 | Novartis Ag | Tuberozinės sklerozės gydymas |
| EP1938800A1 (en) * | 2006-12-06 | 2008-07-02 | Ranbaxy Laboratories Limited | Sirolimus nanodispersion |
| EP1952807A1 (en) | 2007-01-24 | 2008-08-06 | LEK Pharmaceuticals D.D. | Sirolimus formulation |
| US20100166869A1 (en) * | 2007-05-03 | 2010-07-01 | Desai Neil P | Methods and compositions for treating pulmonary hypertension |
| CN102292072A (zh) * | 2009-01-26 | 2011-12-21 | 特瓦制药工业有限公司 | 用微粒包衣载体的方法 |
| GB0908129D0 (en) * | 2009-05-12 | 2009-06-24 | Innovata Ltd | Composition |
| US9248110B2 (en) | 2010-03-18 | 2016-02-02 | Steven Lehrer | Compositions and methods of treating and preventing lung cancer and lymphangioleiomyomatosis |
| PT105058B (pt) | 2010-04-21 | 2013-04-17 | Hovione Farmaciencia S A | Processo para processamento de partículas de ingredientes activos farmacêuticos |
| WO2011163600A2 (en) | 2010-06-25 | 2011-12-29 | Apt Pharmaceuticals, Inc. | Tacrolimus compositions for aerosol administration |
| CA2812952A1 (en) * | 2010-09-27 | 2012-04-12 | Microdose Therapeutx, Inc. | Methods and compositions for disease treatment using inhalation |
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| US10307370B2 (en) * | 2013-10-08 | 2019-06-04 | AI Therapeutics, Inc. | Rapamycin for the treatment of lymphangioleiomyomatosis |
-
2015
- 2015-02-10 KR KR1020167023793A patent/KR20160120739A/ko not_active Withdrawn
- 2015-02-10 CA CA2939342A patent/CA2939342A1/en not_active Abandoned
- 2015-02-10 RU RU2016136348A patent/RU2016136348A/ru not_active Application Discontinuation
- 2015-02-10 JP JP2016551215A patent/JP2017505789A/ja active Pending
- 2015-02-10 BR BR112016018365A patent/BR112016018365A2/pt not_active Application Discontinuation
- 2015-02-10 AU AU2015217349A patent/AU2015217349A1/en not_active Abandoned
- 2015-02-10 WO PCT/US2015/015266 patent/WO2015123219A1/en not_active Ceased
- 2015-02-10 EP EP15706986.5A patent/EP3104891A1/en not_active Withdrawn
- 2015-02-10 US US14/618,621 patent/US20150265582A1/en not_active Abandoned
- 2015-02-10 CN CN201580019126.6A patent/CN106573067A/zh active Pending
- 2015-02-10 MX MX2016010373A patent/MX2016010373A/es unknown
-
2016
- 2016-08-07 IL IL247155A patent/IL247155A0/en unknown
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