JP2016535033A5 - - Google Patents

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Publication number
JP2016535033A5
JP2016535033A5 JP2016526839A JP2016526839A JP2016535033A5 JP 2016535033 A5 JP2016535033 A5 JP 2016535033A5 JP 2016526839 A JP2016526839 A JP 2016526839A JP 2016526839 A JP2016526839 A JP 2016526839A JP 2016535033 A5 JP2016535033 A5 JP 2016535033A5
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JP
Japan
Prior art keywords
boronic acid
chiral
represented
formula
primary
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2016526839A
Other languages
English (en)
Japanese (ja)
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JP2016535033A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2014/063692 external-priority patent/WO2015066612A2/en
Publication of JP2016535033A publication Critical patent/JP2016535033A/ja
Publication of JP2016535033A5 publication Critical patent/JP2016535033A5/ja
Pending legal-status Critical Current

Links

JP2016526839A 2013-11-03 2014-11-03 活性化されていない第二級ボロン酸のクロスカップリング Pending JP2016535033A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361899296P 2013-11-03 2013-11-03
US61/899,296 2013-11-03
PCT/US2014/063692 WO2015066612A2 (en) 2013-11-03 2014-11-03 Cross-coupling of unactivated secondary boronic acids

Publications (2)

Publication Number Publication Date
JP2016535033A JP2016535033A (ja) 2016-11-10
JP2016535033A5 true JP2016535033A5 (enExample) 2018-02-08

Family

ID=51952004

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016526839A Pending JP2016535033A (ja) 2013-11-03 2014-11-03 活性化されていない第二級ボロン酸のクロスカップリング

Country Status (4)

Country Link
US (1) US10072028B2 (enExample)
EP (1) EP3063154B1 (enExample)
JP (1) JP2016535033A (enExample)
WO (1) WO2015066612A2 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6866583B2 (ja) * 2016-07-05 2021-04-28 Dic株式会社 液晶化合物
US10370393B2 (en) 2017-04-21 2019-08-06 The Board Of Trustees Of The University Of Illinois Stereoretentive cross-coupling of boronic acids
WO2021199310A1 (ja) * 2020-03-31 2021-10-07 エヌ・イーケムキャット株式会社 芳香族化合物の製造方法
WO2022032007A2 (en) * 2020-08-05 2022-02-10 Skyhawk Therapeutics, Inc. Process for the preparation of intermediates useful in the preparation of compounds that modulate splicing
WO2022031998A2 (en) * 2020-08-05 2022-02-10 Skyhawk Therapeutics, Inc. Process for the preparation of intermediates useful in the preparation of compounds that modulate splicing

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2694068C (en) 2007-07-23 2016-08-30 The Board Of Trustees Of The University Of Illinois System for controlling the reactivity of boronic acids
JP5501656B2 (ja) * 2008-05-16 2014-05-28 株式会社半導体エネルギー研究所 組成物、薄膜の作製方法、及び発光素子の作製方法
US8338601B2 (en) 2008-09-26 2012-12-25 Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
WO2011103435A2 (en) 2010-02-18 2011-08-25 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
EP2596000B1 (en) 2010-07-23 2016-04-20 The Board of Trustees of the University of Illionis Apparatus and methods for the automated synthesis of small molecules
US9012658B2 (en) 2011-04-27 2015-04-21 The Board Of Trustees Of The University Of Illinois Automated synthesis of small molecules using chiral, non-racemic boronates
EP2647628A1 (en) 2012-04-02 2013-10-09 Almirall, S.A. Substituted tricyclic compounds with activity towards ep1 receptors

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