JP2016525533A5 - - Google Patents

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JP2016525533A5
JP2016525533A5 JP2016528538A JP2016528538A JP2016525533A5 JP 2016525533 A5 JP2016525533 A5 JP 2016525533A5 JP 2016528538 A JP2016528538 A JP 2016528538A JP 2016528538 A JP2016528538 A JP 2016528538A JP 2016525533 A5 JP2016525533 A5 JP 2016525533A5
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Japan
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group
salt
hydroxy
antagonist
methyl
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JP2016528538A
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Japanese (ja)
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JP6374962B2 (ja
JP2016525533A (ja
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Priority claimed from PCT/EP2014/065965 external-priority patent/WO2015011244A1/en
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Publication of JP2016525533A5 publication Critical patent/JP2016525533A5/ja
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JP2016528538A 2013-07-25 2014-07-24 ムスカリン受容体アンタゴニスト活性およびβ２アドレナリン受容体アゴニスト活性の両方を有する、２−アミノ−１−ヒドロキシエチル−８−ヒドロキシキノリン−２（１Ｈ）−オン誘導体の塩 Expired - Fee Related JP6374962B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13382304.7 2013-07-25
EP13382304 2013-07-25
PCT/EP2014/065965 WO2015011244A1 (en) 2013-07-25 2014-07-24 SALTS OF 2-AMINO-1-HYDROXYETHYL-8-HYDROXYQUINOLIN-2(1H)-ONE DERIVATIVES HAVING BOTH MUSCARINIC RECEPTOR ANTAGONIST AND β2 ADRENERGIC RECEPTOR AGONIST ACTIVITIES

Publications (3)

Publication Number Publication Date
JP2016525533A JP2016525533A (ja) 2016-08-25
JP2016525533A5 true JP2016525533A5 (https=) 2017-06-29
JP6374962B2 JP6374962B2 (ja) 2018-08-15

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JP2016528538A Expired - Fee Related JP6374962B2 (ja) 2013-07-25 2014-07-24 ムスカリン受容体アンタゴニスト活性およびβ２アドレナリン受容体アゴニスト活性の両方を有する、２−アミノ−１−ヒドロキシエチル−８−ヒドロキシキノリン−２（１Ｈ）−オン誘導体の塩

Country Status (36)

Country Link
US (1) US9579316B2 (https=)
EP (1) EP3024489B1 (https=)
JP (1) JP6374962B2 (https=)
KR (1) KR102338155B1 (https=)
CN (2) CN105492027A (https=)
AR (1) AR097079A1 (https=)
AU (1) AU2014295028B2 (https=)
BR (1) BR112016001295B1 (https=)
CA (1) CA2917596C (https=)
CL (1) CL2016000187A1 (https=)
CR (1) CR20160043A (https=)
CY (1) CY1122920T1 (https=)
DK (1) DK3024489T3 (https=)
DO (1) DOP2016000011A (https=)
EA (1) EA035436B1 (https=)
ES (1) ES2788627T3 (https=)
HR (1) HRP20200670T1 (https=)
HU (1) HUE049441T2 (https=)
IL (1) IL243173B (https=)
LT (1) LT3024489T (https=)
MX (1) MX360837B (https=)
MY (1) MY184681A (https=)
NI (1) NI201600012A (https=)
NZ (1) NZ715128A (https=)
PE (1) PE20160173A1 (https=)
PH (1) PH12016500125A1 (https=)
PL (1) PL3024489T3 (https=)
PT (1) PT3024489T (https=)
RS (1) RS60185B1 (https=)
SG (1) SG11201510682YA (https=)
SI (1) SI3024489T1 (https=)
SM (1) SMT202000185T1 (https=)
TW (1) TWI641373B (https=)
UY (1) UY35678A (https=)
WO (1) WO2015011244A1 (https=)
ZA (1) ZA201509203B (https=)

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TW201440768A (zh) 2013-02-27 2014-11-01 Almirall Sa 雙毒蕈鹼拮抗劑-β2腎上腺素促效劑複合物及皮質類固醇之組合物
TWI643853B (zh) 2013-02-27 2018-12-11 阿爾米雷爾有限公司 同時具有β2腎上腺素受體促效劑和M3毒蕈鹼受體拮抗劑活性之2-氨基-1-羥乙基-8-羥基喹啉-2(1H)-酮衍生物之鹽類
TWI641373B (zh) 2013-07-25 2018-11-21 阿爾米雷爾有限公司 具有蕈毒鹼受體拮抗劑和β２腎上腺素受體促效劑二者之活性的２－胺基－１－羥乙基－８－羥基喹啉－２（１Ｈ）－酮衍生物之鹽
TW201517906A (zh) 2013-07-25 2015-05-16 Almirall Sa 含有ｍａｂａ化合物和皮質類固醇之組合
TW201617343A (zh) 2014-09-26 2016-05-16 阿爾米雷爾有限公司 具有β２腎上腺素促效劑及Ｍ３蕈毒拮抗劑活性之新穎雙環衍生物

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