JP2016503401A - ジアリールヨードニウム塩を製造するための方法及び試薬 - Google Patents

ジアリールヨードニウム塩を製造するための方法及び試薬 Download PDF

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JP2016503401A
JP2016503401A JP2015539844A JP2015539844A JP2016503401A JP 2016503401 A JP2016503401 A JP 2016503401A JP 2015539844 A JP2015539844 A JP 2015539844A JP 2015539844 A JP2015539844 A JP 2015539844A JP 2016503401 A JP2016503401 A JP 2016503401A
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heterocycloalkyl
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JP2016503401A5 (enExample
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スティーヴン・ジー・ディマグノ
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グランド・フルーア・ファーマスーティカルズ・インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/02—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
    • C07D475/04—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
    • C07C309/65—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00—Ethers; Compounds having groups, groups or groups
    • C07C43/02—Ethers
    • C07C43/20—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
    • C07C43/225—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C71/00—Esters of oxyacids of halogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/44—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having three double bonds between ring members or between ring members and non-ring members
    • C07D207/444—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having three double bonds between ring members or between ring members and non-ring members having two doubly-bound oxygen atoms directly attached in positions 2 and 5
    • C07D207/448—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having three double bonds between ring members or between ring members and non-ring members having two doubly-bound oxygen atoms directly attached in positions 2 and 5 with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms, e.g. maleimide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • C07D277/66—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2 with aromatic rings or ring systems directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Furan Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
JP2015539844A 2012-10-27 2013-10-25 ジアリールヨードニウム塩を製造するための方法及び試薬 Pending JP2016503401A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261719387P 2012-10-27 2012-10-27
US61/719,387 2012-10-27
PCT/US2013/066830 WO2014066772A1 (en) 2012-10-27 2013-10-25 Processes and reagents for making diaryliodonium salts

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JP2016503401A true JP2016503401A (ja) 2016-02-04
JP2016503401A5 JP2016503401A5 (enExample) 2016-12-08

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US (1) US20140121371A1 (enExample)
EP (1) EP2912011A4 (enExample)
JP (1) JP2016503401A (enExample)
AU (1) AU2013334166A1 (enExample)
CA (1) CA2889575A1 (enExample)
IL (1) IL238449A0 (enExample)
WO (1) WO2014066772A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018185503A (ja) * 2017-04-25 2018-11-22 住友化学株式会社 レジスト組成物及びレジストパターンの製造方法

Families Citing this family (6)

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Publication number Priority date Publication date Assignee Title
US9278959B2 (en) 2012-06-05 2016-03-08 Nutech Ventures Processes and reagents for making diaryliodonium salts
US10053423B2 (en) * 2014-01-03 2018-08-21 Nutech Ventures Radioiodinated compounds
WO2016201128A1 (en) * 2015-06-12 2016-12-15 Nutech Ventures Guanidinium compounds
EP3307712A4 (en) * 2015-06-12 2019-01-02 Nutech Ventures Radioiodinated bioconjugation reagents
US10703708B2 (en) * 2015-11-24 2020-07-07 Institut National De La Sante Et De La Recherche Medicale (Inserm) Method for synthesizing iodo- or astatoarenes using diaryliodonium salts
CN116675628A (zh) * 2023-05-10 2023-09-01 南通新纳希新材料有限公司 一种新型的碘鎓盐纯化方法

Citations (4)

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Publication number Priority date Publication date Assignee Title
WO2010117435A2 (en) * 2009-04-08 2010-10-14 The Regents Of The University Of California No-carrier-added nucleophilic [f-18] fluorination of aromatic compounds
US20110190505A1 (en) * 2010-02-04 2011-08-04 Dimagno Stephen Iodonium Cyclophanes for SECURE Arene Functionalization
JP2012506440A (ja) * 2008-10-21 2012-03-15 ヌテク ベンチャーズ 環系芳香族のフッ素化
JP2015523985A (ja) * 2012-06-05 2015-08-20 ニューテック・ベンチャーズ ジアリールヨードニウム塩を製造するための方法及び反応剤

Family Cites Families (3)

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SG98433A1 (en) * 1999-12-21 2003-09-19 Ciba Sc Holding Ag Iodonium salts as latent acid donors
JP4552611B2 (ja) * 2003-11-18 2010-09-29 和光純薬工業株式会社 低分子リサイクル型超原子価ヨウ素試薬
GB0329716D0 (en) * 2003-12-23 2004-01-28 Amersham Plc Radical trap

Patent Citations (4)

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Publication number Priority date Publication date Assignee Title
JP2012506440A (ja) * 2008-10-21 2012-03-15 ヌテク ベンチャーズ 環系芳香族のフッ素化
WO2010117435A2 (en) * 2009-04-08 2010-10-14 The Regents Of The University Of California No-carrier-added nucleophilic [f-18] fluorination of aromatic compounds
US20110190505A1 (en) * 2010-02-04 2011-08-04 Dimagno Stephen Iodonium Cyclophanes for SECURE Arene Functionalization
JP2015523985A (ja) * 2012-06-05 2015-08-20 ニューテック・ベンチャーズ ジアリールヨードニウム塩を製造するための方法及び反応剤

Non-Patent Citations (4)

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Title
MINKWITZ, R. ET AL., EUR. J. INORG. CHEM., JPN6017002729, 2000, pages 2387 - 2392, ISSN: 0003640154 *
TETRAHEDRON LETTERS, vol. 37(46), JPN6017002727, 1996, pages 8421 - 8424, ISSN: 0003640156 *
YE, C. ET AL., ORGANIC LETTERS, vol. 7, no. 18, JPN6017034784, 2005, pages 3961 - 3964, ISSN: 0003640153 *
ZEFIROV, N. S. ET AL.: "General method for synthesis of aryliodoso derivatives under aprotic conditions by reaction of iodos", ZHURNAL ORGANICHESKOI KHIMII, vol. 25, no. 8, JPN6017034785, 1989, pages 1807 - 1808, ISSN: 0003640155 *

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018185503A (ja) * 2017-04-25 2018-11-22 住友化学株式会社 レジスト組成物及びレジストパターンの製造方法
JP2022070893A (ja) * 2017-04-25 2022-05-13 住友化学株式会社 レジスト組成物及びレジストパターンの製造方法
JP7087490B2 (ja) 2017-04-25 2022-06-21 住友化学株式会社 レジスト組成物及びレジストパターンの製造方法
JP7193021B2 (ja) 2017-04-25 2022-12-20 住友化学株式会社 レジスト組成物及びレジストパターンの製造方法

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EP2912011A1 (en) 2015-09-02
EP2912011A4 (en) 2016-11-09
IL238449A0 (en) 2015-06-30
US20140121371A1 (en) 2014-05-01
CA2889575A1 (en) 2014-05-01
WO2014066772A1 (en) 2014-05-01
AU2013334166A1 (en) 2015-05-28

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