JP2015523337A5 - - Google Patents
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- Publication number
- JP2015523337A5 JP2015523337A5 JP2015514142A JP2015514142A JP2015523337A5 JP 2015523337 A5 JP2015523337 A5 JP 2015523337A5 JP 2015514142 A JP2015514142 A JP 2015514142A JP 2015514142 A JP2015514142 A JP 2015514142A JP 2015523337 A5 JP2015523337 A5 JP 2015523337A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- contacted
- solution
- tms
- acetonitrile
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261650553P | 2012-05-23 | 2012-05-23 | |
| US61/650,553 | 2012-05-23 | ||
| PCT/US2013/042150 WO2013177243A1 (en) | 2012-05-23 | 2013-05-22 | Sulfilimine and sulphoxide methods for producing festinavir |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2015523337A JP2015523337A (ja) | 2015-08-13 |
| JP2015523337A5 true JP2015523337A5 (enExample) | 2016-07-07 |
Family
ID=48534517
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015514142A Pending JP2015523337A (ja) | 2012-05-23 | 2013-05-22 | フェスチナビルを製造するためのスルフィリミンおよびスルホキシド方法 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US9249171B2 (enExample) |
| EP (1) | EP2852583A1 (enExample) |
| JP (1) | JP2015523337A (enExample) |
| CN (1) | CN104379571A (enExample) |
| WO (1) | WO2013177243A1 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2986602A1 (en) | 2013-04-16 | 2016-02-24 | Bristol-Myers Squibb Company | Method for producing festinavir using 5-methyluridine as starting material |
| US20160130260A1 (en) | 2013-06-13 | 2016-05-12 | Bristol-Myers Squibb Company | Tert-butyl sulphoxide method for producing festinavir |
| EP3760208B1 (en) | 2014-06-25 | 2024-05-29 | The General Hospital Corporation | Targeting human satellite ii (hsatii) |
| WO2020032152A1 (ja) * | 2018-08-09 | 2020-02-13 | ヤマサ醤油株式会社 | 4'-置換ヌクレオシド誘導体の立体選択的合成法 |
| EP3914604B1 (en) | 2019-01-25 | 2026-03-04 | Brown University | Compositions comprising censavudine or elvucitabine for treating age-associated inflammation and disorders |
| EP4511381A1 (en) * | 2022-04-22 | 2025-02-26 | Rome Therapeutics, Inc. | Didehydro-3'-deoxy-4'-ethynylthymidines and related compounds and their use in treating medical conditions |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0454193A (ja) * | 1990-05-25 | 1992-02-21 | Japan Tobacco Inc | 2’,3’―ジデオキシ―2’,3’―ジデヒドロ―β―リボヌクレオシドの製造方法 |
| CA2514466C (en) | 2003-02-19 | 2015-05-26 | Yale University | Anti-viral nucleoside analogs and methods for treating viral infections, especially hiv infections |
| CA2623522C (en) | 2005-09-26 | 2015-12-08 | Pharmasset, Inc. | Modified 4'-nucleosides as antiviral agents |
| EA200971115A1 (ru) | 2007-06-29 | 2010-04-30 | Корея Рисерч Инститьют Оф Кемикал Текнолоджи | Новые ингибиторы обратной транскриптазы вич |
| US20090318380A1 (en) | 2007-11-20 | 2009-12-24 | Pharmasset, Inc. | 2',4'-substituted nucleosides as antiviral agents |
| US9051288B2 (en) | 2007-12-27 | 2015-06-09 | Oncolys Biopharma, Inc. | Method for producing 4′-ethynyl d4T |
| JP5485138B2 (ja) | 2008-03-28 | 2014-05-07 | 浜理薬品工業株式会社 | エチニルチミジン化合物の精製方法 |
| WO2009125841A1 (ja) | 2008-04-10 | 2009-10-15 | 浜理薬品工業株式会社 | 5-メチルウリジンを出発原料とするエチニルチミジン化合物の製造方法 |
| DE102009034346B4 (de) | 2009-07-23 | 2013-01-24 | Kone Corp. | Antriebssystem für eine Personenförderanlage |
| WO2011099442A1 (ja) | 2010-02-15 | 2011-08-18 | 日産化学工業株式会社 | β-グリコシド化合物の製造方法 |
| WO2011099443A1 (ja) | 2010-02-15 | 2011-08-18 | 日産化学工業株式会社 | β-ジヒドロフラン誘導化合物、β-ジヒドロフラン誘導化合物またはβ-テトラヒドロフラン誘導化合物の製造方法、β-グリコシド化合物、β-グリコシド化合物の製造方法、並びに、4'-エチニルd4T及びその類縁化合物の製造方法 |
-
2013
- 2013-05-22 CN CN201380027023.5A patent/CN104379571A/zh active Pending
- 2013-05-22 US US14/402,231 patent/US9249171B2/en active Active
- 2013-05-22 WO PCT/US2013/042150 patent/WO2013177243A1/en not_active Ceased
- 2013-05-22 EP EP13725545.1A patent/EP2852583A1/en not_active Withdrawn
- 2013-05-22 JP JP2015514142A patent/JP2015523337A/ja active Pending
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