JP2015523337A5 - - Google Patents

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Publication number
JP2015523337A5
JP2015523337A5 JP2015514142A JP2015514142A JP2015523337A5 JP 2015523337 A5 JP2015523337 A5 JP 2015523337A5 JP 2015514142 A JP2015514142 A JP 2015514142A JP 2015514142 A JP2015514142 A JP 2015514142A JP 2015523337 A5 JP2015523337 A5 JP 2015523337A5
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JP
Japan
Prior art keywords
compound
contacted
solution
tms
acetonitrile
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2015514142A
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English (en)
Japanese (ja)
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JP2015523337A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2013/042150 external-priority patent/WO2013177243A1/en
Publication of JP2015523337A publication Critical patent/JP2015523337A/ja
Publication of JP2015523337A5 publication Critical patent/JP2015523337A5/ja
Pending legal-status Critical Current

Links

JP2015514142A 2012-05-23 2013-05-22 フェスチナビルを製造するためのスルフィリミンおよびスルホキシド方法 Pending JP2015523337A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261650553P 2012-05-23 2012-05-23
US61/650,553 2012-05-23
PCT/US2013/042150 WO2013177243A1 (en) 2012-05-23 2013-05-22 Sulfilimine and sulphoxide methods for producing festinavir

Publications (2)

Publication Number Publication Date
JP2015523337A JP2015523337A (ja) 2015-08-13
JP2015523337A5 true JP2015523337A5 (enExample) 2016-07-07

Family

ID=48534517

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015514142A Pending JP2015523337A (ja) 2012-05-23 2013-05-22 フェスチナビルを製造するためのスルフィリミンおよびスルホキシド方法

Country Status (5)

Country Link
US (1) US9249171B2 (enExample)
EP (1) EP2852583A1 (enExample)
JP (1) JP2015523337A (enExample)
CN (1) CN104379571A (enExample)
WO (1) WO2013177243A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014172264A1 (en) 2013-04-16 2014-10-23 Bristol-Myers Squibb Company Method for producing festinavir using 5-methyluridine as starting material
EP3008060A1 (en) 2013-06-13 2016-04-20 Bristol-Myers Squibb Company Tert-butyl-sulphoxide method for producing festinavir
EP3161159B1 (en) 2014-06-25 2020-08-05 The General Hospital Corporation Targeting human satellite ii (hsatii)
WO2020032152A1 (ja) * 2018-08-09 2020-02-13 ヤマサ醤油株式会社 4'-置換ヌクレオシド誘導体の立体選択的合成法
MX2021008751A (es) 2019-01-25 2021-11-12 Univ Brown Composiciones y metodos para tratar, prevenir o revertir la inflamacion y los trastornos asociados a la edad.
CA3250054A1 (en) * 2022-04-22 2023-10-26 Rome Therapeutics, Inc. DIDEHYDRO-3'-DESOXY-4'-ETHYNYLTHYMIDINES, RELATED COMPOUNDS AND THEIR USE IN THE TREATMENT OF MEDICAL CONDITIONS

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0454193A (ja) * 1990-05-25 1992-02-21 Japan Tobacco Inc 2’,3’―ジデオキシ―2’,3’―ジデヒドロ―β―リボヌクレオシドの製造方法
KR20110079783A (ko) 2003-02-19 2011-07-07 예일 유니버시티 항-바이러스 뉴클레오시드 유사체 및 바이러스 감염, 특히 에이치아이브이 감염의 치료방법
EA200800932A1 (ru) 2005-09-26 2008-10-30 Фармассет, Инк. Модифицированные 4`-нуклеозиды в качестве противовирусных агентов
CN101784532B (zh) 2007-06-29 2014-10-22 韩国化学研究院 Hiv逆转录酶抑制剂
US20090318380A1 (en) 2007-11-20 2009-12-24 Pharmasset, Inc. 2',4'-substituted nucleosides as antiviral agents
EP2228373B1 (en) * 2007-12-27 2017-02-08 Oncolys BioPharma, Inc. METHOD FOR PRODUCING 4'-ETHYNYL d4T
JP5485138B2 (ja) 2008-03-28 2014-05-07 浜理薬品工業株式会社 エチニルチミジン化合物の精製方法
JP5485140B2 (ja) 2008-04-10 2014-05-07 浜理薬品工業株式会社 5−メチルウリジンを出発原料とするエチニルチミジン化合物の製造方法
DE102009034346B4 (de) 2009-07-23 2013-01-24 Kone Corp. Antriebssystem für eine Personenförderanlage
KR20130008546A (ko) 2010-02-15 2013-01-22 닛산 가가쿠 고교 가부시키 가이샤 β-글리코사이드 화합물의 제조 방법
EP2537839B1 (en) 2010-02-15 2016-12-14 Nissan Chemical Industries, Ltd. B-dihydrofuran deriving compound, method for producing b-dihydrofuran deriving compound or b-tetrahydrofuran deriving compound, b -glycoside compound, method for producing b-glycoside compound, and method for producing 4'-ethynyl d4t and analogue compounds thereof

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