JP2014532744A - バニロイド受容体リガンドとしての、ｓｏ２含有基で置換されたフェニル部分を担持する置換ピラゾリルをベースとするカルボキサミドおよび尿素誘導体 - Google Patents
バニロイド受容体リガンドとしての、ｓｏ２含有基で置換されたフェニル部分を担持する置換ピラゾリルをベースとするカルボキサミドおよび尿素誘導体 Download PDFInfo
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- JP2014532744A JP2014532744A JP2014540456A JP2014540456A JP2014532744A JP 2014532744 A JP2014532744 A JP 2014532744A JP 2014540456 A JP2014540456 A JP 2014540456A JP 2014540456 A JP2014540456 A JP 2014540456A JP 2014532744 A JP2014532744 A JP 2014532744A
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- methyl
- phenyl
- fluoro
- pyrazol
- methylsulfonyl
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- 239000000203 mixture Substances 0.000 claims description 53
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- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11008927.3 | 2011-11-09 | ||
| EP11008927 | 2011-11-09 | ||
| PCT/EP2012/072143 WO2013068464A1 (en) | 2011-11-09 | 2012-11-08 | Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2014532744A true JP2014532744A (ja) | 2014-12-08 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014540456A Withdrawn JP2014532744A (ja) | 2011-11-09 | 2012-11-08 | バニロイド受容体リガンドとしての、ｓｏ２含有基で置換されたフェニル部分を担持する置換ピラゾリルをベースとするカルボキサミドおよび尿素誘導体 |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP2776401A1 (es) |
| JP (1) | JP2014532744A (es) |
| KR (1) | KR20140091041A (es) |
| CN (1) | CN104066720A (es) |
| AR (1) | AR088799A1 (es) |
| AU (1) | AU2012334068A1 (es) |
| BR (1) | BR112014011108A2 (es) |
| CA (1) | CA2854424A1 (es) |
| HK (1) | HK1202117A1 (es) |
| IN (1) | IN2014KN00865A (es) |
| MX (1) | MX2014005233A (es) |
| TW (1) | TW201326135A (es) |
| WO (1) | WO2013068464A1 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2016011468A (es) | 2014-03-07 | 2017-01-23 | Biocryst Pharm Inc | Inhibidores de calicreína plasmática humana. |
| BR112017010402B1 (pt) * | 2014-11-24 | 2023-12-12 | Medifron Dbt Inc | Carboxamida substituída à base de tiazol e oxazol e derivados de ureia como ligantes de receptor vanilóide ii |
| CN114920697A (zh) * | 2022-05-16 | 2022-08-19 | 河南应用技术职业学院 | 杂环基取代的茚满丙酰胺类化合物及其应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| AU2010244685B2 (en) | 2009-05-07 | 2016-02-18 | Medifron Dbt Inc. | Substituted phenylureas and phenylamides as vanilloid receptor ligands |
| BRPI1011192A2 (pt) | 2009-05-07 | 2016-03-15 | Gruenenthal Gmbh | derivados de carboxamida e ureia aromáticas substituídas como ligantes de receptor de vaniloide, composição farmacêutica, uso e processo para preparação dos referidos derivados |
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2012
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- 2012-11-08 TW TW101141483A patent/TW201326135A/zh unknown
- 2012-11-08 IN IN865KON2014 patent/IN2014KN00865A/en unknown
- 2012-11-08 EP EP12783220.2A patent/EP2776401A1/en not_active Withdrawn
- 2012-11-08 CN CN201280055221.8A patent/CN104066720A/zh active Pending
- 2012-11-08 AR ARP120104205A patent/AR088799A1/es unknown
- 2012-11-08 JP JP2014540456A patent/JP2014532744A/ja not_active Withdrawn
- 2012-11-08 MX MX2014005233A patent/MX2014005233A/es not_active Application Discontinuation
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2015
- 2015-03-13 HK HK15102581.4A patent/HK1202117A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20140091041A (ko) | 2014-07-18 |
| BR112014011108A2 (pt) | 2017-05-16 |
| AU2012334068A1 (en) | 2014-05-22 |
| WO2013068464A1 (en) | 2013-05-16 |
| EP2776401A1 (en) | 2014-09-17 |
| MX2014005233A (es) | 2014-08-22 |
| HK1202117A1 (en) | 2015-09-18 |
| TW201326135A (zh) | 2013-07-01 |
| IN2014KN00865A (es) | 2015-10-02 |
| CA2854424A1 (en) | 2013-05-16 |
| AR088799A1 (es) | 2014-07-10 |
| CN104066720A (zh) | 2014-09-24 |
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