KR20140091041A - 바닐로이드 수용체 리간드로서의 so2-함유 그룹으로 치환된 페닐 모이어티를 갖는 치환된 피라졸릴계 카복사미드 및 우레아 유도체들 - Google Patents
바닐로이드 수용체 리간드로서의 so2-함유 그룹으로 치환된 페닐 모이어티를 갖는 치환된 피라졸릴계 카복사미드 및 우레아 유도체들 Download PDFInfo
- Publication number
- KR20140091041A KR20140091041A KR1020147015421A KR20147015421A KR20140091041A KR 20140091041 A KR20140091041 A KR 20140091041A KR 1020147015421 A KR1020147015421 A KR 1020147015421A KR 20147015421 A KR20147015421 A KR 20147015421A KR 20140091041 A KR20140091041 A KR 20140091041A
- Authority
- KR
- South Korea
- Prior art keywords
- phenyl
- methyl
- fluoro
- methylsulfonyl
- group
- Prior art date
Links
- 0 CC(C(NCc1cc(*)n[n]1C1=CC(C)(**)C=C(*)C(*)=C1)=O)c1cc(*)c(*(C)CC(C)(C)S(**)(=O)=O)c(*)c1 Chemical compound CC(C(NCc1cc(*)n[n]1C1=CC(C)(**)C=C(*)C(*)=C1)=O)c1cc(*)c(*(C)CC(C)(C)S(**)(=O)=O)c(*)c1 0.000 description 3
- CEAGLDAEZQNFGC-UHFFFAOYSA-N CS(CCc(c(F)c1)ccc1N)(=O)=O Chemical compound CS(CCc(c(F)c1)ccc1N)(=O)=O CEAGLDAEZQNFGC-UHFFFAOYSA-N 0.000 description 1
- ZZURNVWYIDEVLH-UHFFFAOYSA-N CS(CCc(c(F)c1)ccc1NC(NCc1cc(C2CC2)n[n]1-c1cc(Cl)ccc1)=O)(=O)=O Chemical compound CS(CCc(c(F)c1)ccc1NC(NCc1cc(C2CC2)n[n]1-c1cc(Cl)ccc1)=O)(=O)=O ZZURNVWYIDEVLH-UHFFFAOYSA-N 0.000 description 1
- PZYLYSZFZWNLRP-UHFFFAOYSA-N CS(CCc(c(F)c1)ccc1NC(Oc1ccccc1)=O)(=O)=O Chemical compound CS(CCc(c(F)c1)ccc1NC(Oc1ccccc1)=O)(=O)=O PZYLYSZFZWNLRP-UHFFFAOYSA-N 0.000 description 1
- QCMJFIOMUPUNCX-UHFFFAOYSA-N CS(CCc(ccc([N+]([O-])=O)c1)c1F)(=O)=O Chemical compound CS(CCc(ccc([N+]([O-])=O)c1)c1F)(=O)=O QCMJFIOMUPUNCX-UHFFFAOYSA-N 0.000 description 1
- DATVTDZGELNXCT-UHFFFAOYSA-N [O-][N+](c1cc(F)c(CCBr)cc1)=O Chemical compound [O-][N+](c1cc(F)c(CCBr)cc1)=O DATVTDZGELNXCT-UHFFFAOYSA-N 0.000 description 1
- HKGNZXXYXCKJHO-UHFFFAOYSA-N [O-][N+](c1ccc(CC(O)=O)c(F)c1)=O Chemical compound [O-][N+](c1ccc(CC(O)=O)c(F)c1)=O HKGNZXXYXCKJHO-UHFFFAOYSA-N 0.000 description 1
- MVVPCXHRMBDTBV-UHFFFAOYSA-N [O-][N+](c1ccc(CCO)c(F)c1)=O Chemical compound [O-][N+](c1ccc(CCO)c(F)c1)=O MVVPCXHRMBDTBV-UHFFFAOYSA-N 0.000 description 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
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- Rheumatology (AREA)
- Dermatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Virology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Urology & Nephrology (AREA)
- Hematology (AREA)
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- Anesthesiology (AREA)
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- Cardiology (AREA)
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- Communicable Diseases (AREA)
- Nutrition Science (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Ophthalmology & Optometry (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11008927 | 2011-11-09 | ||
| EP11008927.3 | 2011-11-09 | ||
| PCT/EP2012/072143 WO2013068464A1 (en) | 2011-11-09 | 2012-11-08 | Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20140091041A true KR20140091041A (ko) | 2014-07-18 |
Family
ID=47143914
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020147015421A KR20140091041A (ko) | 2011-11-09 | 2012-11-08 | 바닐로이드 수용체 리간드로서의 so2-함유 그룹으로 치환된 페닐 모이어티를 갖는 치환된 피라졸릴계 카복사미드 및 우레아 유도체들 |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP2776401A1 (es) |
| JP (1) | JP2014532744A (es) |
| KR (1) | KR20140091041A (es) |
| CN (1) | CN104066720A (es) |
| AR (1) | AR088799A1 (es) |
| AU (1) | AU2012334068A1 (es) |
| BR (1) | BR112014011108A2 (es) |
| CA (1) | CA2854424A1 (es) |
| HK (1) | HK1202117A1 (es) |
| IN (1) | IN2014KN00865A (es) |
| MX (1) | MX2014005233A (es) |
| TW (1) | TW201326135A (es) |
| WO (1) | WO2013068464A1 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4180424A1 (en) | 2014-03-07 | 2023-05-17 | BioCryst Pharmaceuticals, Inc. | Substituted pyrazoles as human plasma kallikrein inhibitors |
| TW201625568A (zh) * | 2014-11-24 | 2016-07-16 | 歌林達有限公司 | 作爲類香草素受體之配位體ｉｉ之經取代以噁唑及噻唑爲主之甲醯胺及脲衍生物 |
| CN114920697A (zh) * | 2022-05-16 | 2022-08-19 | 河南应用技术职业学院 | 杂环基取代的茚满丙酰胺类化合物及其应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2553392C2 (ru) | 2009-05-07 | 2015-06-10 | Грюненталь Гмбх | Замещенные фенилмочевины и фениламиды в качестве лигандов ваниллоидных рецепторов |
| MX2011011800A (es) | 2009-05-07 | 2012-01-27 | Gruenenthal Gmbh | Derivados de carboxamida y urea aromaticas sustituidas como ligandos del receptor de vanilloides. |
-
2012
- 2012-11-08 AR ARP120104205A patent/AR088799A1/es unknown
- 2012-11-08 AU AU2012334068A patent/AU2012334068A1/en not_active Abandoned
- 2012-11-08 CA CA2854424A patent/CA2854424A1/en not_active Abandoned
- 2012-11-08 EP EP12783220.2A patent/EP2776401A1/en not_active Withdrawn
- 2012-11-08 JP JP2014540456A patent/JP2014532744A/ja not_active Withdrawn
- 2012-11-08 KR KR1020147015421A patent/KR20140091041A/ko not_active Application Discontinuation
- 2012-11-08 MX MX2014005233A patent/MX2014005233A/es not_active Application Discontinuation
- 2012-11-08 CN CN201280055221.8A patent/CN104066720A/zh active Pending
- 2012-11-08 BR BR112014011108A patent/BR112014011108A2/pt not_active IP Right Cessation
- 2012-11-08 TW TW101141483A patent/TW201326135A/zh unknown
- 2012-11-08 IN IN865KON2014 patent/IN2014KN00865A/en unknown
- 2012-11-08 WO PCT/EP2012/072143 patent/WO2013068464A1/en active Application Filing
-
2015
- 2015-03-13 HK HK15102581.4A patent/HK1202117A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| HK1202117A1 (en) | 2015-09-18 |
| BR112014011108A2 (pt) | 2017-05-16 |
| CN104066720A (zh) | 2014-09-24 |
| IN2014KN00865A (es) | 2015-10-02 |
| JP2014532744A (ja) | 2014-12-08 |
| MX2014005233A (es) | 2014-08-22 |
| EP2776401A1 (en) | 2014-09-17 |
| WO2013068464A1 (en) | 2013-05-16 |
| AU2012334068A1 (en) | 2014-05-22 |
| TW201326135A (zh) | 2013-07-01 |
| CA2854424A1 (en) | 2013-05-16 |
| AR088799A1 (es) | 2014-07-10 |
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