IN2014KN00865A - - Google Patents

Info

Publication number
IN2014KN00865A
IN2014KN00865A IN865KON2014A IN2014KN00865A IN 2014KN00865 A IN2014KN00865 A IN 2014KN00865A IN 865KON2014 A IN865KON2014 A IN 865KON2014A IN 2014KN00865 A IN2014KN00865 A IN 2014KN00865A
Authority
IN
India
Prior art keywords
compounds
substituted
prophylaxis
pain
disorders
Prior art date
Application number
Inventor
Foltyn Robert Frank
Thomas Christoph
Nils Damann
Bernhard Lesch
Gregor Bahrenberg
Derek John Saunders
Hannelore Stockhausen
Yong Soo Kim
Myeong Seop Kim
Jeewoo Lee
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of IN2014KN00865A publication Critical patent/IN2014KN00865A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36—Opioid-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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Abstract

2The invention relates to substituted pyrazolyl based carboxamide and urea derivatives bearing a phenyl moiety substituted with a S0 containing group as vanilloid receptor ligands to pharmaceutical compositions containing these compounds and also to these compounds for use in the treatment and/or prophylaxis of pain and further diseases and/or disorders.
IN865KON2014 2011-11-09 2012-11-08 IN2014KN00865A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP11008927 2011-11-09
PCT/EP2012/072143 WO2013068464A1 (en) 2011-11-09 2012-11-08 Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands

Publications (1)

Publication Number Publication Date
IN2014KN00865A true IN2014KN00865A (en) 2015-10-02

Family

ID=47143914

Family Applications (1)

Application Number Title Priority Date Filing Date
IN865KON2014 IN2014KN00865A (en) 2011-11-09 2012-11-08

Country Status (13)

Country Link
EP (1) EP2776401A1 (en)
JP (1) JP2014532744A (en)
KR (1) KR20140091041A (en)
CN (1) CN104066720A (en)
AR (1) AR088799A1 (en)
AU (1) AU2012334068A1 (en)
BR (1) BR112014011108A2 (en)
CA (1) CA2854424A1 (en)
HK (1) HK1202117A1 (en)
IN (1) IN2014KN00865A (en)
MX (1) MX2014005233A (en)
TW (1) TW201326135A (en)
WO (1) WO2013068464A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ724250A (en) 2014-03-07 2022-02-25 Biocryst Pharm Inc Human plasma kallikrein inhibitors
ES2713700T3 (en) 2014-11-24 2019-05-23 Medifron Dbt Inc Derivatives of carboxamide and urea based on oxazole and thiazole substituted as ligands of the vanilloid II receptor
CN114920697A (en) * 2022-05-16 2022-08-19 河南应用技术职业学院 Heterocyclic group substituted indan propionamide compound and application thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI491595B (en) * 2009-05-07 2015-07-11 歌林達股份有限公司 Substituted phenylureas and phenylamides as vanilloid receptor ligands
US8334315B2 (en) 2009-05-07 2012-12-18 Gruenenthal Gmbh Substituted aromatic carboxamide and urea derivatives as vanilloid receptor ligands

Also Published As

Publication number Publication date
WO2013068464A1 (en) 2013-05-16
CA2854424A1 (en) 2013-05-16
AU2012334068A1 (en) 2014-05-22
BR112014011108A2 (en) 2017-05-16
TW201326135A (en) 2013-07-01
CN104066720A (en) 2014-09-24
MX2014005233A (en) 2014-08-22
HK1202117A1 (en) 2015-09-18
AR088799A1 (en) 2014-07-10
KR20140091041A (en) 2014-07-18
EP2776401A1 (en) 2014-09-17
JP2014532744A (en) 2014-12-08

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