JP2014528431A5 - - Google Patents

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Publication number
JP2014528431A5
JP2014528431A5 JP2014533869A JP2014533869A JP2014528431A5 JP 2014528431 A5 JP2014528431 A5 JP 2014528431A5 JP 2014533869 A JP2014533869 A JP 2014533869A JP 2014533869 A JP2014533869 A JP 2014533869A JP 2014528431 A5 JP2014528431 A5 JP 2014528431A5
Authority
JP
Japan
Prior art keywords
sustained
coating
release pharmaceutical
water
release
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2014533869A
Other languages
English (en)
Japanese (ja)
Other versions
JP2014528431A (ja
JP6368242B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2012/069541 external-priority patent/WO2013050419A1/en
Publication of JP2014528431A publication Critical patent/JP2014528431A/ja
Publication of JP2014528431A5 publication Critical patent/JP2014528431A5/ja
Application granted granted Critical
Publication of JP6368242B2 publication Critical patent/JP6368242B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2014533869A 2011-10-06 2012-10-03 40−o−(2−ヒドロキシ)エチル−ラパマイシンを含む医薬組成物 Expired - Fee Related JP6368242B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161544026P 2011-10-06 2011-10-06
US61/544,026 2011-10-06
PCT/EP2012/069541 WO2013050419A1 (en) 2011-10-06 2012-10-03 Pharmaceutical compositions comprising 40 - o - ( 2 - hydroxy) ethyl - rapamycin

Publications (3)

Publication Number Publication Date
JP2014528431A JP2014528431A (ja) 2014-10-27
JP2014528431A5 true JP2014528431A5 (enExample) 2015-11-12
JP6368242B2 JP6368242B2 (ja) 2018-08-01

Family

ID=46968222

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014533869A Expired - Fee Related JP6368242B2 (ja) 2011-10-06 2012-10-03 40−o−(2−ヒドロキシ)エチル−ラパマイシンを含む医薬組成物

Country Status (24)

Country Link
US (3) US20140242162A1 (enExample)
EP (1) EP2763663B1 (enExample)
JP (1) JP6368242B2 (enExample)
KR (1) KR101643219B1 (enExample)
CN (1) CN103874484B (enExample)
AR (1) AR088232A1 (enExample)
AU (1) AU2012320563B2 (enExample)
BR (1) BR112014007902A2 (enExample)
CA (1) CA2850995A1 (enExample)
CL (1) CL2014000844A1 (enExample)
CO (1) CO6930364A2 (enExample)
EA (1) EA025595B1 (enExample)
ES (1) ES2663744T3 (enExample)
GT (1) GT201400062A (enExample)
IL (1) IL231648A0 (enExample)
MA (1) MA35513B1 (enExample)
MX (1) MX2014004166A (enExample)
PE (1) PE20141649A1 (enExample)
PH (1) PH12014500746A1 (enExample)
SG (1) SG11201400730VA (enExample)
TN (1) TN2014000114A1 (enExample)
TW (1) TWI475993B (enExample)
WO (1) WO2013050419A1 (enExample)
ZA (1) ZA201401961B (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201503912A (zh) * 2013-03-19 2015-02-01 Novartis Ag 包含癌莫事(everolimus)之醫藥組合物
US10709700B2 (en) 2014-09-15 2020-07-14 Orphazyme A/S Arimoclomol formulation
US20160250270A1 (en) 2015-02-27 2016-09-01 Ebbu, LLC Compositions comprising combinations of purified cannabinoids, with at least one flavonoid, terpene, or mineral
EP3297629A1 (en) 2015-05-20 2018-03-28 Novartis AG Pharmaceutical combination of everolimus with dactolisib
EP3329916A4 (en) 2015-07-28 2019-03-20 Nippon Kayaku Kabushiki Kaisha PHARMACEUTICAL COMPOSITION COMPRISING RAPAMYCIN OR A DERIVATIVE THEREOF, AND PROCESS FOR PRODUCING THE SAME
JP6762158B2 (ja) * 2015-07-28 2020-09-30 日本化薬株式会社 ラパマイシン又はその誘導体を含有する医薬組成物
WO2017038925A1 (ja) * 2015-09-03 2017-03-09 日本化薬株式会社 ラパマイシン又はその誘導体を含有する医薬組成物
JP6854639B2 (ja) * 2016-01-06 2021-04-07 日本化薬株式会社 ラパマイシン誘導体を含有する医薬組成物及びその製造方法
CA3034004C (en) 2016-08-29 2021-08-03 Canopy Growth Corporation Water soluble compositions comprising purified cannabinoids
US12485129B2 (en) 2016-08-29 2025-12-02 Canopy Growth Corporation Water soluble compositions comprising purified cannabinoids
BR112019010470A2 (pt) 2016-11-23 2019-09-10 Novartis Ag métodos de realce de resposta imune com everolimo, dactolisib ou ambos
EP3576735A4 (en) * 2017-02-06 2020-07-22 Intas Pharmaceuticals Limited PHARMACEUTICAL COMPOSITION OF EVEROLIMUS
KR102051806B1 (ko) * 2018-01-12 2019-12-04 주식회사 종근당 에베로리무스를 포함하는 안정화된 약제학적 제제
US10596165B2 (en) 2018-02-12 2020-03-24 resTORbio, Inc. Combination therapies
JP2023520021A (ja) * 2020-03-30 2023-05-15 アイジーアイエー ファーマシューティカルズ インコーポレイテッド チロシンキナーゼ阻害剤の小児用製剤
WO2022219652A1 (en) * 2021-04-17 2022-10-20 Bdr Pharmaceuticals International Private Limited Novel sublingual pharmaceutical formulations for everolimus
KR102336007B1 (ko) * 2021-06-23 2021-12-07 주식회사 진성이앤지 콘크리트용 우레탄계 방수·방식 도막재 및 이를 이용한 방수·방식 도장 공법
WO2023044024A1 (en) * 2021-09-17 2023-03-23 Novelstar Pharmaceuticals Inc. Novel ph dependent coating drug delivery system
GB202415232D0 (en) 2024-10-16 2024-11-27 Nacamed As Composition

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5472712A (en) * 1991-12-24 1995-12-05 Euroceltique, S.A. Controlled-release formulations coated with aqueous dispersions of ethylcellulose
GB9221220D0 (en) 1992-10-09 1992-11-25 Sandoz Ag Organic componds
FR2736550B1 (fr) 1995-07-14 1998-07-24 Sandoz Sa Composition pharmaceutique sous la forme d'une dispersion solide comprenant un macrolide et un vehicule
PT2198858E (pt) * 1998-03-26 2011-09-01 Astellas Pharma Inc Composição farmacêutica de libertação constante que contém um macrólido como o tacrolimus
GB0123400D0 (en) 2001-09-28 2001-11-21 Novartis Ag Organic compounds
AR045957A1 (es) * 2003-10-03 2005-11-16 Novartis Ag Composicion farmaceutica y combinacion
GB0419355D0 (en) * 2004-08-31 2004-09-29 Novartis Ag Organic compounds
EP1902708A1 (de) * 2006-09-25 2008-03-26 Losan Pharma GmbH Wirkstoff enthaltende stabilisierte feste Arzneimittelformen und Verfahren zu ihrer Herstellung
PT2365802T (pt) * 2008-11-11 2017-11-14 Univ Texas Microcápsulas de rapamicina e utilização para o tratamento de cancro
CN101862297B (zh) * 2009-04-14 2012-07-25 上海医药工业研究院 一种非水溶性药物的缓释微丸、其缓释口腔崩解片及其制备方法

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