GT201400062A - Composiciones farmacéuticas que comprenden 40-o-(2-hidroxi) etil-rapamicina - Google Patents

Composiciones farmacéuticas que comprenden 40-o-(2-hidroxi) etil-rapamicina

Info

Publication number
GT201400062A
GT201400062A GT201400062A GT201400062A GT201400062A GT 201400062 A GT201400062 A GT 201400062A GT 201400062 A GT201400062 A GT 201400062A GT 201400062 A GT201400062 A GT 201400062A GT 201400062 A GT201400062 A GT 201400062A
Authority
GT
Guatemala
Prior art keywords
rapamycin
hidroxi
etil
pharmaceutical compositions
diseases
Prior art date
Application number
GT201400062A
Other languages
English (en)
Spanish (es)
Inventor
Diederich Anke
Liechti Kurt
Kuehl Peter
Cheung Wing
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46968222&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT201400062(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT201400062A publication Critical patent/GT201400062A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
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    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
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    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
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    • A61K9/7007—Drug-containing films, membranes or sheets
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    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Transplantation (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
GT201400062A 2011-10-06 2014-04-04 Composiciones farmacéuticas que comprenden 40-o-(2-hidroxi) etil-rapamicina GT201400062A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161544026P 2011-10-06 2011-10-06

Publications (1)

Publication Number Publication Date
GT201400062A true GT201400062A (es) 2015-06-02

Family

ID=46968222

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201400062A GT201400062A (es) 2011-10-06 2014-04-04 Composiciones farmacéuticas que comprenden 40-o-(2-hidroxi) etil-rapamicina

Country Status (24)

Country Link
US (3) US20140242162A1 (enExample)
EP (1) EP2763663B1 (enExample)
JP (1) JP6368242B2 (enExample)
KR (1) KR101643219B1 (enExample)
CN (1) CN103874484B (enExample)
AR (1) AR088232A1 (enExample)
AU (1) AU2012320563B2 (enExample)
BR (1) BR112014007902A2 (enExample)
CA (1) CA2850995A1 (enExample)
CL (1) CL2014000844A1 (enExample)
CO (1) CO6930364A2 (enExample)
EA (1) EA025595B1 (enExample)
ES (1) ES2663744T3 (enExample)
GT (1) GT201400062A (enExample)
IL (1) IL231648A0 (enExample)
MA (1) MA35513B1 (enExample)
MX (1) MX2014004166A (enExample)
PE (1) PE20141649A1 (enExample)
PH (1) PH12014500746A1 (enExample)
SG (1) SG11201400730VA (enExample)
TN (1) TN2014000114A1 (enExample)
TW (1) TWI475993B (enExample)
WO (1) WO2013050419A1 (enExample)
ZA (1) ZA201401961B (enExample)

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TW201503912A (zh) * 2013-03-19 2015-02-01 Novartis Ag 包含癌莫事(everolimus)之醫藥組合物
US10709700B2 (en) * 2014-09-15 2020-07-14 Orphazyme A/S Arimoclomol formulation
AU2016225026A1 (en) 2015-02-27 2017-09-07 Canopy Growth Corporation Compositions comprising combinations of purified cannabinoids, with at least one flavonoid, terpene, or mineral
US10576076B2 (en) 2015-05-20 2020-03-03 Novartis Ag Pharmaceutical combination of everolimus with dactolisib
JP6762158B2 (ja) * 2015-07-28 2020-09-30 日本化薬株式会社 ラパマイシン又はその誘導体を含有する医薬組成物
WO2017018433A1 (ja) * 2015-07-28 2017-02-02 日本化薬株式会社 ラパマイシン又はその誘導体を含有する医薬組成物及びその製造方法
US20190022073A1 (en) * 2015-09-03 2019-01-24 Nippon Kayaku Kabushiki Kaisha Pharmaceutical composition comprising rapamycin or derivative thereof
JP6854639B2 (ja) * 2016-01-06 2021-04-07 日本化薬株式会社 ラパマイシン誘導体を含有する医薬組成物及びその製造方法
BR112019003815A2 (pt) 2016-08-29 2019-05-21 Canopy Growth Corporation composições solúveis em água compreendendo canabinoides purificados
US12485129B2 (en) 2016-08-29 2025-12-02 Canopy Growth Corporation Water soluble compositions comprising purified cannabinoids
JP2020500930A (ja) 2016-11-23 2020-01-16 ノバルティス アーゲー エベロリムス、ダクトリシブまたは両方で免疫応答を増強する方法
US20200093804A1 (en) * 2017-02-06 2020-03-26 Intas Pharmaceuticals Ltd. Pharmaceutical composition of everolimus
KR102051806B1 (ko) * 2018-01-12 2019-12-04 주식회사 종근당 에베로리무스를 포함하는 안정화된 약제학적 제제
WO2019157516A1 (en) 2018-02-12 2019-08-15 resTORbio, Inc. Combination therapies
JP7891740B2 (ja) * 2020-03-30 2026-07-17 イエール ユニバーシティ チロシンキナーゼ阻害剤の小児用製剤
WO2022219652A1 (en) * 2021-04-17 2022-10-20 Bdr Pharmaceuticals International Private Limited Novel sublingual pharmaceutical formulations for everolimus
KR102336007B1 (ko) * 2021-06-23 2021-12-07 주식회사 진성이앤지 콘크리트용 우레탄계 방수·방식 도막재 및 이를 이용한 방수·방식 도장 공법
WO2023044024A1 (en) * 2021-09-17 2023-03-23 Novelstar Pharmaceuticals Inc. Novel ph dependent coating drug delivery system
GB202415232D0 (en) 2024-10-16 2024-11-27 Nacamed As Composition

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CA2937492C (en) * 2008-11-11 2019-08-13 The Board Of Regents Of The University Of Texas System Inhibition of mammalian target of rapamycin
CN101862297B (zh) * 2009-04-14 2012-07-25 上海医药工业研究院 一种非水溶性药物的缓释微丸、其缓释口腔崩解片及其制备方法

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TW201318625A (zh) 2013-05-16
EA025595B1 (ru) 2017-01-30
EP2763663B1 (en) 2017-12-27
CO6930364A2 (es) 2014-04-28
TN2014000114A1 (en) 2015-07-01
CN103874484A (zh) 2014-06-18
CN103874484B (zh) 2016-09-21
EA201490743A1 (ru) 2014-07-30
BR112014007902A2 (pt) 2017-04-18
IL231648A0 (en) 2014-05-28
KR20140058670A (ko) 2014-05-14
US20180214424A1 (en) 2018-08-02
CA2850995A1 (en) 2013-04-11
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KR101643219B1 (ko) 2016-07-27
AU2012320563B2 (en) 2016-05-12
PE20141649A1 (es) 2014-11-14
EP2763663A1 (en) 2014-08-13
JP6368242B2 (ja) 2018-08-01
TWI475993B (zh) 2015-03-11
AU2012320563A1 (en) 2014-04-24
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