JP2014527043A - Ｓｒｃホモロジー２プロテインチロシンホスファターゼ−１を含むアゴニスト及びその治療方法 - Google Patents

Ｓｒｃホモロジー２プロテインチロシンホスファターゼ−１を含むアゴニスト及びその治療方法 Download PDF

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JP2014527043A
JP2014527043A JP2014523113A JP2014523113A JP2014527043A JP 2014527043 A JP2014527043 A JP 2014527043A JP 2014523113 A JP2014523113 A JP 2014523113A JP 2014523113 A JP2014523113 A JP 2014523113A JP 2014527043 A JP2014527043 A JP 2014527043A
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チョン−ワイ シアオ
クエン−フェン チェン
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DCB USA LLC
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    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/59—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton the carbon skeleton being further substituted by singly-bound oxygen atoms
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    • C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
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    • C07C275/36—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with at least one of the oxygen atoms further bound to a carbon atom of a six-membered aromatic ring, e.g. N-aryloxyphenylureas
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JP2014523113A 2011-08-03 2012-08-03 Ｓｒｃホモロジー２プロテインチロシンホスファターゼ−１を含むアゴニスト及びその治療方法 Pending JP2014527043A (ja)

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US201161514555P 2011-08-03 2011-08-03
US61/514,555 2011-08-03
PCT/US2012/049446 WO2013020014A1 (en) 2011-08-03 2012-08-03 Agonists of src homology-2 containing protein tyrosine phosphatase-1 and treatment methods using the same

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Cited By (1)

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JP2019528279A (ja) * 2016-08-17 2019-10-10 アイカーン スクール オブ メディシン アット マウント サイナイ キナーゼ阻害物質化合物、組成物、及びがんの治療方法

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CA2883172A1 (en) * 2012-08-29 2014-03-06 Merck Patent Gmbh Ddr2 inhibitors for the treatment of osteoarthritis
EP2989466B1 (en) * 2013-04-25 2018-10-31 CBS Bioscience, Co., Ltd Analytical method for increasing susceptibility of molecular targeted therapy in hepatocellular carcinoma
WO2015051149A1 (en) * 2013-10-04 2015-04-09 The Trustees Of Columbia University In The City Of New York Sorafenib analogs and uses thereof
KR20180043199A (ko) 2015-08-31 2018-04-27 도레이 카부시키가이샤 요소 유도체 및 그 용도
US10745346B2 (en) * 2015-09-02 2020-08-18 Kuen-Feng Chen Agonists of protein tyrosine phosphatase SHP-1
CN109789116B (zh) * 2016-09-22 2022-02-01 陈昆锋 Sc-43用于改善纤维化的用途
MX2019009200A (es) * 2017-02-03 2019-10-21 Univ California Composiciones y métodos para inhibir el reticulón 4.
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