JP2014514288A5 - - Google Patents
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- Publication number
- JP2014514288A5 JP2014514288A5 JP2014501606A JP2014501606A JP2014514288A5 JP 2014514288 A5 JP2014514288 A5 JP 2014514288A5 JP 2014501606 A JP2014501606 A JP 2014501606A JP 2014501606 A JP2014501606 A JP 2014501606A JP 2014514288 A5 JP2014514288 A5 JP 2014514288A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- bisphosphonic acid
- alkyl
- acid derivative
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CC(N1CCN(C)CC1)=* Chemical compound CC(N1CCN(C)CC1)=* 0.000 description 4
- RXYPXQSKLGGKOL-UHFFFAOYSA-N CN1CCN(C)CC1 Chemical compound CN1CCN(C)CC1 RXYPXQSKLGGKOL-UHFFFAOYSA-N 0.000 description 2
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR1152546A FR2973378B1 (fr) | 2011-03-28 | 2011-03-28 | Derives d'acide hydroxybisphosphonique bifonctionnels |
| FR1152546 | 2011-03-28 | ||
| PCT/EP2012/055569 WO2012130911A1 (fr) | 2011-03-28 | 2012-03-28 | Derives d'acide hydroxybisphosphonique bifonctionnels |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014514288A JP2014514288A (ja) | 2014-06-19 |
| JP2014514288A5 true JP2014514288A5 (enExample) | 2015-05-14 |
| JP6026499B2 JP6026499B2 (ja) | 2016-11-16 |
Family
ID=45926557
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014501606A Expired - Fee Related JP6026499B2 (ja) | 2011-03-28 | 2012-03-28 | 二機能性ヒドロキシ−ビスホスホン酸誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US9173946B2 (enExample) |
| EP (1) | EP2691402B1 (enExample) |
| JP (1) | JP6026499B2 (enExample) |
| CA (1) | CA2831713C (enExample) |
| ES (1) | ES2743276T3 (enExample) |
| FR (1) | FR2973378B1 (enExample) |
| WO (1) | WO2012130911A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR3028762B1 (fr) | 2014-11-20 | 2017-01-06 | Atlanthera | Derives hydroxybisphosphoniques hydrosolubles de la doxorubicine |
| TWI609875B (zh) * | 2015-04-20 | 2018-01-01 | 聚和國際股份有限公司 | 用於骨掃描的化合物及其用途 |
| JP7599176B2 (ja) * | 2019-02-06 | 2024-12-13 | オレゴン ヘルス アンド サイエンス ユニバーシティ | ビスホスホネート連結化合物 |
| EP4003201A4 (en) * | 2019-07-24 | 2023-08-23 | Brigham Young University | BONE BONDING CONNECTIONS |
| US11679099B2 (en) * | 2020-05-13 | 2023-06-20 | Seoul National University R&Db Foundation | Use of HIF-2α inhibitors for treating chondrosarcoma, or preventing recurrence and metastasis thereof |
| FR3122427B1 (fr) | 2021-04-30 | 2025-03-07 | Atlanthera | Derives hydroxybisphosphoniques de meloxicam pour traitement des maladies inflammatoires osteoarticulaires |
| KR20240116793A (ko) * | 2021-12-10 | 2024-07-30 | 피피지 인더스트리즈 오하이오 인코포레이티드 | 카바제이트 작용성 화합물 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2558373A1 (de) | 1974-12-26 | 1976-07-08 | Yoshida Kogyo Kk | Aussenfenstereinheit |
| US4830847A (en) * | 1985-06-28 | 1989-05-16 | The Procter & Gamble Company | Diphosphonate-derivatized macromolecules |
| PH26923A (en) * | 1989-03-08 | 1992-12-03 | Ciba Geigy | N-substituted amino alkanediphosphonic acids |
| IT1303672B1 (it) * | 1998-07-28 | 2001-02-23 | Nicox Sa | Sali nitrati di farmaci attivi nei disordini ossei |
| EP1615639A2 (en) * | 2003-04-03 | 2006-01-18 | Semafore Pharmaceuticals, Inc. | Targeted bone marrow protection agents |
| US8404664B2 (en) * | 2005-08-11 | 2013-03-26 | Targanta Therapeutics, Inc. | Phosphonated Rifamycins and uses thereof for the prevention and treatment of bone and joint infections |
| US8133311B2 (en) * | 2007-04-30 | 2012-03-13 | Cabot Corporation | Pigment dipsersions comprising functionalized non-polymeric dispersants |
| FR2926081B1 (fr) * | 2008-01-03 | 2010-02-19 | Univ Nantes | Derives d'acide hydroxy-bisphosphonique comme vecteur ciblant le tissu osseux |
| FR2926080B1 (fr) * | 2008-01-03 | 2010-04-02 | Univ Nantes | Procede de synthese de derives d'acide hydroxy-bisphosphonique |
| EP2289558A1 (en) * | 2009-08-25 | 2011-03-02 | KTB Tumorforschungsgesellschaft mbH | Bisphosphonate-prodrugs |
-
2011
- 2011-03-28 FR FR1152546A patent/FR2973378B1/fr not_active Expired - Fee Related
-
2012
- 2012-03-28 ES ES12711632T patent/ES2743276T3/es active Active
- 2012-03-28 WO PCT/EP2012/055569 patent/WO2012130911A1/fr not_active Ceased
- 2012-03-28 US US14/008,986 patent/US9173946B2/en active Active
- 2012-03-28 JP JP2014501606A patent/JP6026499B2/ja not_active Expired - Fee Related
- 2012-03-28 EP EP12711632.5A patent/EP2691402B1/fr active Active
- 2012-03-28 CA CA2831713A patent/CA2831713C/fr active Active
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