JP2014193889A5 - - Google Patents

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Publication number
JP2014193889A5
JP2014193889A5 JP2014099667A JP2014099667A JP2014193889A5 JP 2014193889 A5 JP2014193889 A5 JP 2014193889A5 JP 2014099667 A JP2014099667 A JP 2014099667A JP 2014099667 A JP2014099667 A JP 2014099667A JP 2014193889 A5 JP2014193889 A5 JP 2014193889A5
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JP
Japan
Prior art keywords
alkyl
independently
substituted
hal
alkoxy
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JP2014099667A
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English (en)
Japanese (ja)
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JP5876527B2 (ja
JP2014193889A (ja
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Publication of JP2014193889A publication Critical patent/JP2014193889A/ja
Publication of JP2014193889A5 publication Critical patent/JP2014193889A5/ja
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Publication of JP5876527B2 publication Critical patent/JP5876527B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2014099667A 2007-04-11 2014-05-13 診断用画像及び放射線治療用の葉酸複合体及び対応する金属キレート錯体 Expired - Fee Related JP5876527B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07105980.2 2007-04-11
EP07105980 2007-04-11

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2010502521A Division JP5710246B2 (ja) 2007-04-11 2008-04-11 診断用画像及び放射線治療用の葉酸複合体及び対応する金属キレート錯体

Publications (3)

Publication Number Publication Date
JP2014193889A JP2014193889A (ja) 2014-10-09
JP2014193889A5 true JP2014193889A5 (https=) 2015-03-19
JP5876527B2 JP5876527B2 (ja) 2016-03-02

Family

ID=39683755

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2010502521A Expired - Fee Related JP5710246B2 (ja) 2007-04-11 2008-04-11 診断用画像及び放射線治療用の葉酸複合体及び対応する金属キレート錯体
JP2014099667A Expired - Fee Related JP5876527B2 (ja) 2007-04-11 2014-05-13 診断用画像及び放射線治療用の葉酸複合体及び対応する金属キレート錯体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2010502521A Expired - Fee Related JP5710246B2 (ja) 2007-04-11 2008-04-11 診断用画像及び放射線治療用の葉酸複合体及び対応する金属キレート錯体

Country Status (11)

Country Link
US (2) US20100143249A1 (https=)
EP (1) EP2146995A1 (https=)
JP (2) JP5710246B2 (https=)
KR (2) KR101605426B1 (https=)
CN (1) CN101646672B (https=)
AU (1) AU2008237935B2 (https=)
CA (1) CA2670385C (https=)
EA (1) EA200901344A1 (https=)
IL (1) IL201250A0 (https=)
WO (1) WO2008125618A1 (https=)
ZA (1) ZA200903483B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008125618A1 (en) * 2007-04-11 2008-10-23 Merck Eprova Ag Folate-conjugates and corresponding metal-chelate complexes for use in diagnostic imaging and radiotherapy
US8236284B1 (en) * 2008-04-02 2012-08-07 University Of Central Florida Research Foundation, Inc. Multimodal, multifunctional polymer coated nanoparticles
FR2942227B1 (fr) * 2009-02-13 2011-04-15 Guerbet Sa Utilisation de tampons pour la complexation de radionucleides
WO2011084571A2 (en) 2009-12-16 2011-07-14 Mallinckrodt Inc. Azide derivatives for phototherapy
CN103732595B (zh) * 2011-08-17 2017-02-08 默克及其合伙人公司 叶酸的白蛋白‑结合实体缀合物
AU2013258027B2 (en) 2012-05-08 2017-11-30 Merck & Cie 18F-labelled follate/antifolate analogues
EP3253732A4 (en) * 2015-02-06 2018-08-29 Cempra Pharmaceuticals, Inc. 4-azidobutylamines and processes for preparing
WO2020256210A1 (ko) 2019-06-20 2020-12-24 주식회사 쿼드마이너 네트워크 포렌식 시스템 및 이를 이용한 네트워크 포렌식 방법

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6093382A (en) * 1998-05-16 2000-07-25 Bracco Research Usa Inc. Metal complexes derivatized with folate for use in diagnostic and therapeutic applications
ATE427948T1 (de) * 2001-04-24 2009-04-15 Purdue Research Foundation Folat-mimetika und deren folatrezeptorbindende konjugate
JP4801348B2 (ja) * 2002-05-06 2011-10-26 エンドサイト,インコーポレイテッド ビタミンを標的とした造影剤
EP1618380B1 (en) * 2003-04-29 2009-12-30 Universität Zürich N epsilon AND/OR N alpha DERIVATIZED, METAL AND ORGANIC PROTECTED L-HISTIDINE FOR COUPLING TO BIOMOLECULES FOR HIGHLY EFFICIENT LABELING WITH (M(OH2)3(CO)3)+ BY FAC COORDINATION
US9265746B2 (en) * 2006-05-31 2016-02-23 Merck & Cie Method for cell-specific targeting
WO2008125618A1 (en) * 2007-04-11 2008-10-23 Merck Eprova Ag Folate-conjugates and corresponding metal-chelate complexes for use in diagnostic imaging and radiotherapy

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