JP2013541513A5 - - Google Patents

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Publication number
JP2013541513A5
JP2013541513A5 JP2013526466A JP2013526466A JP2013541513A5 JP 2013541513 A5 JP2013541513 A5 JP 2013541513A5 JP 2013526466 A JP2013526466 A JP 2013526466A JP 2013526466 A JP2013526466 A JP 2013526466A JP 2013541513 A5 JP2013541513 A5 JP 2013541513A5
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JP
Japan
Prior art keywords
alkyl
group
heterocycle
carbocycle
optionally substituted
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JP2013526466A
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English (en)
Japanese (ja)
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JP6048406B2 (ja
JP2013541513A (ja
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Priority claimed from PCT/EP2011/065080 external-priority patent/WO2012028676A1/en
Publication of JP2013541513A publication Critical patent/JP2013541513A/ja
Publication of JP2013541513A5 publication Critical patent/JP2013541513A5/ja
Application granted granted Critical
Publication of JP6048406B2 publication Critical patent/JP6048406B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2013526466A 2010-09-02 2011-09-01 新規化合物、医薬組成物及びこれらの使用 Expired - Fee Related JP6048406B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10175100.6 2010-09-02
EP10175100 2010-09-02
PCT/EP2011/065080 WO2012028676A1 (en) 2010-09-02 2011-09-01 New compounds, pharmaceutical compositions and uses thereof

Publications (3)

Publication Number Publication Date
JP2013541513A JP2013541513A (ja) 2013-11-14
JP2013541513A5 true JP2013541513A5 (https=) 2014-10-23
JP6048406B2 JP6048406B2 (ja) 2016-12-21

Family

ID=44583007

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013526466A Expired - Fee Related JP6048406B2 (ja) 2010-09-02 2011-09-01 新規化合物、医薬組成物及びこれらの使用

Country Status (4)

Country Link
US (1) US8835472B2 (https=)
EP (1) EP2611771B1 (https=)
JP (1) JP6048406B2 (https=)
WO (1) WO2012028676A1 (https=)

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CA2835332C (en) * 2011-05-10 2019-03-26 Sandoz Ag Polymorph of linagliptin benzoate
US8530460B2 (en) 2011-12-19 2013-09-10 Boehringer Ingelheim International Gmbh Azetidine derivatives
FR3000491B1 (fr) * 2012-09-27 2015-08-28 Univ Lille Ii Droit & Sante Composes utilisables dans le traitement des infections mycobacteriennes
US9371282B2 (en) 2013-05-17 2016-06-21 Centrexion Therapeutics Corporation Somatostatin receptor subtype 4 (SSTR4) agonists
HK1217448A1 (zh) 2013-09-12 2017-01-13 辉瑞大药厂 乙酰辅酶a羧化酶抑制剂用於治疗寻常痤疮的用途
JPWO2015125824A1 (ja) 2014-02-18 2017-03-30 日産化学工業株式会社 アルキニルピリジン置換アミド化合物及び有害生物防除剤
KR20180011843A (ko) * 2015-06-11 2018-02-02 바실리어 파마슈티카 인터내셔널 리미티드 유출-펌프 억제제 및 이의 치료적 용도
AR105392A1 (es) 2015-07-20 2017-09-27 Genzyme Corp Inhibidores del receptor del factor estimulador de colonias 1 (csf-1r)
WO2017117708A1 (en) * 2016-01-05 2017-07-13 Hua Medicine (Shanghai) Ltd. Pyrazole derivatives
WO2018003924A1 (ja) * 2016-06-29 2018-01-04 日産化学工業株式会社 アルキニルピリジン置換アミド化合物及び有害生物防除剤
UY38687A (es) * 2019-05-17 2023-05-15 Novartis Ag Inhibidores del inflamasoma nlrp3, composiciones, combinaciones de los mismos y métodos para su uso
CN112979612B (zh) * 2021-02-21 2022-09-09 苏州大学 一种室温制备2-碘代杂环芳醚的方法
US12371413B2 (en) 2021-02-22 2025-07-29 Soochow University Method for preparing 2-iodoheterocyclic aryl ether at room temperature
EP4151616A4 (en) * 2021-04-26 2023-12-20 Mitsubishi Gas Chemical Company, Inc. Compound and method for producing same
TWI860849B (zh) 2021-09-14 2024-11-01 美商美國禮來大藥廠 Sstr4促效劑鹽
CA3247765A1 (en) * 2022-01-27 2025-07-10 Vivozon,Inc. PHARMACEUTICAL COMPOSITION FOR THE PREVENTION OR TREATMENT OF A MENTAL DISORDER
US20250270173A1 (en) * 2022-04-19 2025-08-28 Gilgamesh Pharmaceuticals, Inc. Pyridine derivatives for treating psychiatric disorders
UY40374A (es) 2022-08-03 2024-02-15 Novartis Ag Inhibidores de inflamasoma nlrp3

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CA2176854A1 (en) * 1995-06-07 1996-12-08 Daniel J. Keavy N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics
US6284796B1 (en) * 1998-08-06 2001-09-04 Abbott Laboratories Ukokinase inhibitors
AU2003221322A1 (en) * 2002-03-07 2003-09-16 Sds Biotech K.K. Substituted isoxazole alkylamine derivative and agri- and horticultural fungicide
US7915424B2 (en) 2004-03-22 2011-03-29 Eli Lilly And Company Pyridyl derivatives and their use as mGlu5 antagonists
WO2006016548A1 (ja) * 2004-08-09 2006-02-16 Eisai R & D Management Co., Ltd. ヘテロ環化合物を含有する新規な抗マラリア剤
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DK1794163T3 (da) 2004-09-22 2010-04-12 Pfizer Fremgangsmåde til fremstilling af poly(ADP-ribose)polymeraseinhibitorer
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