JP2013541513A5 - - Google Patents
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- Publication number
- JP2013541513A5 JP2013541513A5 JP2013526466A JP2013526466A JP2013541513A5 JP 2013541513 A5 JP2013541513 A5 JP 2013541513A5 JP 2013526466 A JP2013526466 A JP 2013526466A JP 2013526466 A JP2013526466 A JP 2013526466A JP 2013541513 A5 JP2013541513 A5 JP 2013541513A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- heterocycle
- carbocycle
- optionally substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10175100 | 2010-09-02 | ||
| EP10175100.6 | 2010-09-02 | ||
| PCT/EP2011/065080 WO2012028676A1 (en) | 2010-09-02 | 2011-09-01 | New compounds, pharmaceutical compositions and uses thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013541513A JP2013541513A (ja) | 2013-11-14 |
| JP2013541513A5 true JP2013541513A5 (https=) | 2014-10-23 |
| JP6048406B2 JP6048406B2 (ja) | 2016-12-21 |
Family
ID=44583007
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013526466A Expired - Fee Related JP6048406B2 (ja) | 2010-09-02 | 2011-09-01 | 新規化合物、医薬組成物及びこれらの使用 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US8835472B2 (https=) |
| EP (1) | EP2611771B1 (https=) |
| JP (1) | JP6048406B2 (https=) |
| WO (1) | WO2012028676A1 (https=) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2835332C (en) * | 2011-05-10 | 2019-03-26 | Sandoz Ag | Polymorph of linagliptin benzoate |
| US8530460B2 (en) | 2011-12-19 | 2013-09-10 | Boehringer Ingelheim International Gmbh | Azetidine derivatives |
| FR3000491B1 (fr) | 2012-09-27 | 2015-08-28 | Univ Lille Ii Droit & Sante | Composes utilisables dans le traitement des infections mycobacteriennes |
| US9371282B2 (en) | 2013-05-17 | 2016-06-21 | Centrexion Therapeutics Corporation | Somatostatin receptor subtype 4 (SSTR4) agonists |
| US20160220557A1 (en) | 2013-09-12 | 2016-08-04 | Pfizer Inc. | Use of acetyl-coa carboxylase inhibitors for treating acne vulgaris |
| AU2015219902B2 (en) | 2014-02-18 | 2018-11-22 | Nissan Chemical Corporation | Alkynyl pyridine-substituted amide compound and pesticide |
| CN107709314A (zh) * | 2015-06-11 | 2018-02-16 | 巴斯利尔药物国际股份公司 | 外排泵抑制剂及其治疗性用途 |
| CA3217238A1 (en) | 2015-07-20 | 2017-01-26 | Genzyme Corporation | Colony stimulating factor-1 receptor (csf-1r) inhibitors |
| EP3400220B1 (en) * | 2016-01-05 | 2021-03-24 | Hua Medicine (Shanghai) Ltd. | Pyrazole derivatives |
| WO2018003924A1 (ja) * | 2016-06-29 | 2018-01-04 | 日産化学工業株式会社 | アルキニルピリジン置換アミド化合物及び有害生物防除剤 |
| AR119731A1 (es) * | 2019-05-17 | 2022-01-05 | Novartis Ag | Inhibidores del inflamasoma nlrp3 |
| CN112979612B (zh) * | 2021-02-21 | 2022-09-09 | 苏州大学 | 一种室温制备2-碘代杂环芳醚的方法 |
| WO2022174468A1 (zh) * | 2021-02-22 | 2022-08-25 | 苏州大学 | 一种室温制备2-碘代杂环芳醚的方法 |
| CN115605457B (zh) * | 2021-04-26 | 2025-03-18 | 三菱瓦斯化学株式会社 | 化合物及其制造方法 |
| TWI860849B (zh) | 2021-09-14 | 2024-11-01 | 美商美國禮來大藥廠 | Sstr4促效劑鹽 |
| CA3247765A1 (en) * | 2022-01-27 | 2025-07-10 | Vivozon,Inc. | PHARMACEUTICAL COMPOSITION FOR THE PREVENTION OR TREATMENT OF A MENTAL DISORDER |
| WO2023205116A1 (en) * | 2022-04-19 | 2023-10-26 | Gilgamesh Pharmaceuticals, Inc. | Pyridine derivatives for treating psychiatric disorders |
| UY40374A (es) | 2022-08-03 | 2024-02-15 | Novartis Ag | Inhibidores de inflamasoma nlrp3 |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2176854A1 (en) * | 1995-06-07 | 1996-12-08 | Daniel J. Keavy | N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics |
| US6284796B1 (en) * | 1998-08-06 | 2001-09-04 | Abbott Laboratories | Ukokinase inhibitors |
| JP4471262B2 (ja) * | 2002-03-07 | 2010-06-02 | 株式会社エス・ディー・エス バイオテック | 置換イソキサゾールアルキルアミン誘導体及び農園芸用殺菌剤 |
| DE602005017129D1 (de) | 2004-03-22 | 2009-11-26 | Lilly Co Eli | Pyridyl-derivate und ihre verwendung als mglu5-rezeptorantagonisten |
| EP1782811A4 (en) * | 2004-08-09 | 2010-09-01 | Eisai R&D Man Co Ltd | INNOVATIVE ANTIPALUDITIC AGENT CONTAINING A HETEROCYCLIC COMPOUND |
| TWI366438B (en) * | 2004-08-12 | 2012-06-21 | Ishihara Sangyo Kaisha | Fungicidal composition containing acid amide derivative |
| PT1794163E (pt) | 2004-09-22 | 2010-03-01 | Pfizer | Método para a preparação de inibidores de poli(adpribose)- polimerases |
| WO2006094800A2 (en) * | 2005-03-04 | 2006-09-14 | Synthon B.V. | Cascade reaction process |
| JP2008534565A (ja) * | 2005-03-31 | 2008-08-28 | アストラゼネカ アクチボラグ | Tie2阻害活性のあるアミノピリミジン誘導体 |
| AR061243A1 (es) * | 2006-06-08 | 2008-08-13 | Syngenta Ltd | Derivados de n-2-feniletil-carboxamidas, composiciones para el control de mocroorganismos fitopatogenicos que los comprenden y un metodo de control o prevencion de infestacion de plantas utiles que los emplea. |
| WO2008027466A1 (en) * | 2006-08-31 | 2008-03-06 | Schering Corporation | Hydantoin derivatives useful as antibacterial agents |
| TWI519508B (zh) * | 2007-06-12 | 2016-02-01 | Achaogen Inc | 抗菌劑 |
| JP2010529971A (ja) * | 2007-06-15 | 2010-09-02 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | 新規殺微生物剤 |
| WO2009024342A2 (en) * | 2007-08-23 | 2009-02-26 | Syngenta Participations Ag | Novel microbiocides |
| MY156662A (en) * | 2007-11-01 | 2016-03-15 | Acucela Inc | Amine derivative compounds for treating ophthalmic diseases and disorders |
| JP2011510004A (ja) | 2008-01-22 | 2011-03-31 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング | タンパク質キナーゼ阻害剤及びその使用 |
| GB0807140D0 (en) * | 2008-04-18 | 2008-05-21 | Syngenta Participations Ag | Novel microbiocides |
| WO2010050445A1 (ja) | 2008-10-27 | 2010-05-06 | 武田薬品工業株式会社 | 二環性化合物 |
| JP2012162460A (ja) * | 2009-05-27 | 2012-08-30 | Nippon Soda Co Ltd | 含窒素ヘテロアリール誘導体および農園芸用殺菌剤 |
| EP2448928B1 (en) | 2009-07-01 | 2014-08-13 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
| US8389536B2 (en) | 2009-10-27 | 2013-03-05 | Hoffmann-La Roche Inc. | Positive allosteric modulators (PAM) |
-
2011
- 2011-08-17 US US13/211,472 patent/US8835472B2/en active Active
- 2011-09-01 JP JP2013526466A patent/JP6048406B2/ja not_active Expired - Fee Related
- 2011-09-01 EP EP11752529.5A patent/EP2611771B1/en active Active
- 2011-09-01 WO PCT/EP2011/065080 patent/WO2012028676A1/en not_active Ceased
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