JP2013538230A - 抗ウイルス治療用の２’−フルオロ置換カルバヌクレオシド類似体 - Google Patents
抗ウイルス治療用の２’−フルオロ置換カルバヌクレオシド類似体 Download PDFInfo
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- JP2013538230A JP2013538230A JP2013529139A JP2013529139A JP2013538230A JP 2013538230 A JP2013538230 A JP 2013538230A JP 2013529139 A JP2013529139 A JP 2013529139A JP 2013529139 A JP2013529139 A JP 2013529139A JP 2013538230 A JP2013538230 A JP 2013538230A
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Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/4164—1,3-Diazoles
- A61K31/4188—1,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
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- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/7056—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
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| JP2017523169A (ja) * | 2014-07-28 | 2017-08-17 | ギリアード サイエンシーズ， インコーポレイテッド | 呼吸器合胞体ウイルス感染の処置のために有用な、チエノ［３，２−ｄ］ピリミジン、フロ［３，２−ｄ］ピリミジン、およびピロロ［３，２−ｄ］ピリミジン |
| KR20230057411A (ko) * | 2020-08-27 | 2023-04-28 | 길리애드 사이언시즈, 인코포레이티드 | 바이러스 감염 치료를 위한 화합물 및 방법 |
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| EA025311B1 (ru) | 2010-07-19 | 2016-12-30 | Гайлид Сайэнсиз, Инк. | Способы получения диастереомерно чистых фосфорамидатных пролекарств |
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2011
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- 2011-03-22 KR KR1020137010012A patent/KR101879887B1/ko active Active
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- 2013-03-18 CL CL2013000727A patent/CL2013000727A1/es unknown
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2016
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| JP2017523169A (ja) * | 2014-07-28 | 2017-08-17 | ギリアード サイエンシーズ， インコーポレイテッド | 呼吸器合胞体ウイルス感染の処置のために有用な、チエノ［３，２−ｄ］ピリミジン、フロ［３，２−ｄ］ピリミジン、およびピロロ［３，２−ｄ］ピリミジン |
| JP2020023590A (ja) * | 2014-07-28 | 2020-02-13 | ギリアード サイエンシーズ， インコーポレイテッド | 呼吸器合胞体ウイルス感染の処置のために有用な、チエノ［３，２−ｄ］ピリミジン、フロ［３，２−ｄ］ピリミジン、およびピロロ［３，２−ｄ］ピリミジン |
| JP6991188B2 (ja) | 2014-07-28 | 2022-01-12 | ギリアード サイエンシーズ， インコーポレイテッド | 呼吸器合胞体ウイルス感染の処置のために有用な、チエノ［３，２－ｄ］ピリミジン、フロ［３，２－ｄ］ピリミジン、およびピロロ［３，２－ｄ］ピリミジン |
| KR20230057411A (ko) * | 2020-08-27 | 2023-04-28 | 길리애드 사이언시즈, 인코포레이티드 | 바이러스 감염 치료를 위한 화합물 및 방법 |
| JP2023540225A (ja) * | 2020-08-27 | 2023-09-22 | ギリアード サイエンシーズ， インコーポレイテッド | ウイルス感染症の治療のための化合物及び方法 |
| JP7560659B2 (ja) | 2020-08-27 | 2024-10-02 | ギリアード サイエンシーズ， インコーポレイテッド | ウイルス感染症の治療のための化合物及び方法 |
| JP2024178294A (ja) * | 2020-08-27 | 2024-12-24 | ギリアード サイエンシーズ， インコーポレイテッド | ウイルス感染症の治療のための化合物及び方法 |
| KR102833881B1 (ko) | 2020-08-27 | 2025-07-15 | 길리애드 사이언시즈, 인코포레이티드 | 바이러스 감염 치료를 위한 화합물 및 방법 |
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|---|---|
| CN103108876A (zh) | 2013-05-15 |
| JP2017119726A (ja) | 2017-07-06 |
| PH12013500311A1 (en) | 2013-04-22 |
| CA2807496C (en) | 2019-01-22 |
| EA201390141A1 (ru) | 2013-09-30 |
| EA026523B1 (ru) | 2017-04-28 |
| KR20130110168A (ko) | 2013-10-08 |
| CO6680669A2 (es) | 2013-05-31 |
| BR112013008017A2 (pt) | 2016-06-14 |
| JP6475280B2 (ja) | 2019-02-27 |
| PE20131165A1 (es) | 2013-10-14 |
| JP2016074732A (ja) | 2016-05-12 |
| EP2619206A1 (en) | 2013-07-31 |
| MX2013003179A (es) | 2013-04-24 |
| CR20130172A (es) | 2013-05-29 |
| CL2013000727A1 (es) | 2013-08-23 |
| ZA201301042B (en) | 2014-07-30 |
| AP3699A (en) | 2016-05-31 |
| AU2011306066A1 (en) | 2013-02-28 |
| ECSP13012560A (es) | 2013-06-28 |
| IL225221A0 (en) | 2013-06-27 |
| KR101879887B1 (ko) | 2018-07-18 |
| CA2807496A1 (en) | 2012-03-29 |
| MA34593B1 (fr) | 2013-10-02 |
| NZ608070A (en) | 2015-11-27 |
| WO2012039791A1 (en) | 2012-03-29 |
| AP2013006767A0 (en) | 2013-03-31 |
| PH12013500311B1 (en) | 2017-11-08 |
| JP2019014726A (ja) | 2019-01-31 |
| PE20230684A1 (es) | 2023-04-21 |
| AU2011306066B2 (en) | 2015-01-29 |
| SG188223A1 (en) | 2013-04-30 |
| PE20171624A1 (es) | 2017-11-02 |
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