JP2013533241A - 食物効果が減少した制御放出組成物 - Google Patents
食物効果が減少した制御放出組成物 Download PDFInfo
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- JP2013533241A JP2013533241A JP2013516682A JP2013516682A JP2013533241A JP 2013533241 A JP2013533241 A JP 2013533241A JP 2013516682 A JP2013516682 A JP 2013516682A JP 2013516682 A JP2013516682 A JP 2013516682A JP 2013533241 A JP2013533241 A JP 2013533241A
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- metformin
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/28—Insulins
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
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- Gastroenterology & Hepatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
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- General Chemical & Material Sciences (AREA)
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| US35725110P | 2010-06-22 | 2010-06-22 | |
| US61/357,251 | 2010-06-22 | ||
| PCT/US2011/041218 WO2011163206A2 (en) | 2010-06-22 | 2011-06-21 | Controlled release compositions with reduced food effect |
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| JP2013533241A true JP2013533241A (ja) | 2013-08-22 |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12018090B2 (en) | 2014-05-15 | 2024-06-25 | Rani Therapeutics, Llc | PCSK9 antibody preparations for delivery into a lumen of the intestinal tract using a swallowable drug delivery device |
| US12214019B2 (en) | 2014-05-15 | 2025-02-04 | Rani Therapeutics, Llc | Pharmaceutical compositions and methods for fabrication of solid masses comprising polypeptides and/or proteins |
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| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
| DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
| EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
| PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
| JP5323684B2 (ja) | 2006-05-04 | 2013-10-23 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 多形体 |
| PE20091730A1 (es) | 2008-04-03 | 2009-12-10 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
| BRPI0916997A2 (pt) | 2008-08-06 | 2020-12-15 | Boehringer Ingelheim International Gmbh | Inibidor de dpp-4 e seu uso |
| US20200155558A1 (en) | 2018-11-20 | 2020-05-21 | Boehringer Ingelheim International Gmbh | Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug |
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| MX366325B (es) | 2010-05-05 | 2019-07-05 | Boehringer Ingelheim Int | Terapia de combinacion. |
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| JP6218811B2 (ja) | 2012-05-14 | 2017-10-25 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｓｉｒｓ及び／又は敗血症の治療に用いるｄｐｐ−４阻害薬としてのキサンチン誘導体 |
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| CN105496970A (zh) * | 2015-12-18 | 2016-04-20 | 北京华禧联合科技发展有限公司 | 含有利格列汀的组合物及其制备方法 |
| CN106924208A (zh) * | 2015-12-30 | 2017-07-07 | 深圳翰宇药业股份有限公司 | 一种复方达格列净二甲双胍缓释片及其制备方法 |
| WO2017153939A1 (en) * | 2016-03-10 | 2017-09-14 | Aurobindo Pharma Limited | Pharmaceutical composition comprising canagliflozin, process of preparation and use thereof |
| BR112018072401A2 (pt) | 2016-06-10 | 2019-02-19 | Boehringer Ingelheim International Gmbh | combinações de linagliptina e metformina |
| JP2021521270A (ja) | 2018-04-06 | 2021-08-26 | アンマ セラピューティクス インコーポレイテッドＡｍｍａ Ｔｈｅｒａｐｅｕｔｉｃｓ， Ｉｎｃ． | 治療剤の制御放出用組成物 |
| IT201800011119A1 (it) | 2018-12-14 | 2020-06-14 | Dpl Pharma S P A | Composizioni farmaceutiche orali solide per la somministrazione cronotropica di sitagliptin |
| TR201916829A2 (tr) * | 2019-10-31 | 2021-05-21 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Dapagli̇flozi̇n ve metformi̇n i̇çeren çi̇ft katmanli tablet formülasyonlari |
| CN110974792A (zh) * | 2019-12-26 | 2020-04-10 | 南京亿华药业有限公司 | 一种结晶性药物片剂及其制备方法 |
| WO2022073151A1 (en) * | 2020-10-05 | 2022-04-14 | Theracos Sub, Llc | Pharmaceutical formulations |
| KR20250154775A (ko) * | 2024-04-22 | 2025-10-29 | 제이피바이오 주식회사 | 다파글리플로진, 리나글립틴 및 메트포르민을 포함하는 안정성이 향상된 약제학적 제제 |
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- 2011-06-21 MX MX2012015188A patent/MX2012015188A/es active IP Right Grant
- 2011-06-21 RU RU2012155890/15A patent/RU2012155890A/ru not_active Application Discontinuation
- 2011-06-21 AR ARP110102144A patent/AR084698A1/es unknown
- 2011-06-21 CN CN201180031366XA patent/CN103037849A/zh active Pending
- 2011-06-21 EP EP11798742.0A patent/EP2585052A4/en not_active Withdrawn
- 2011-06-21 AU AU2011271124A patent/AU2011271124A1/en not_active Abandoned
- 2011-06-21 US US13/164,995 patent/US8486453B2/en not_active Expired - Fee Related
- 2011-06-21 BR BR112012032816A patent/BR112012032816A2/pt not_active IP Right Cessation
- 2011-06-21 WO PCT/US2011/041218 patent/WO2011163206A2/en not_active Ceased
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- 2011-06-21 CA CA2802335A patent/CA2802335A1/en not_active Abandoned
- 2011-06-21 KR KR1020127033481A patent/KR20140007247A/ko not_active Withdrawn
- 2011-06-22 TW TW100121863A patent/TW201206503A/zh unknown
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12018090B2 (en) | 2014-05-15 | 2024-06-25 | Rani Therapeutics, Llc | PCSK9 antibody preparations for delivery into a lumen of the intestinal tract using a swallowable drug delivery device |
| US12214019B2 (en) | 2014-05-15 | 2025-02-04 | Rani Therapeutics, Llc | Pharmaceutical compositions and methods for fabrication of solid masses comprising polypeptides and/or proteins |
Also Published As
| Publication number | Publication date |
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| KR20140007247A (ko) | 2014-01-17 |
| CA2802335A1 (en) | 2011-12-29 |
| TW201206503A (en) | 2012-02-16 |
| BR112012032816A2 (pt) | 2016-11-08 |
| EP2585052A4 (en) | 2014-10-01 |
| AU2011271124A1 (en) | 2013-01-10 |
| AR084698A1 (es) | 2013-06-05 |
| RU2012155890A (ru) | 2014-07-27 |
| WO2011163206A3 (en) | 2012-03-01 |
| WO2011163206A4 (en) | 2012-04-26 |
| US8486453B2 (en) | 2013-07-16 |
| WO2011163206A2 (en) | 2011-12-29 |
| US20110311594A1 (en) | 2011-12-22 |
| EP2585052A2 (en) | 2013-05-01 |
| CN103037849A (zh) | 2013-04-10 |
| MX2012015188A (es) | 2013-05-20 |
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