JP2013531640A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2013531640A5 JP2013531640A5 JP2013513621A JP2013513621A JP2013531640A5 JP 2013531640 A5 JP2013531640 A5 JP 2013531640A5 JP 2013513621 A JP2013513621 A JP 2013513621A JP 2013513621 A JP2013513621 A JP 2013513621A JP 2013531640 A5 JP2013531640 A5 JP 2013531640A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- weight
- ooc
- butyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- -1 ester amide compound Chemical class 0.000 claims 20
- 238000000034 method Methods 0.000 claims 13
- 150000001412 amines Chemical class 0.000 claims 7
- 150000007514 bases Chemical class 0.000 claims 6
- 125000004432 carbon atom Chemical group C* 0.000 claims 5
- 239000000203 mixture Substances 0.000 claims 5
- WYURNTSHIVDZCO-UHFFFAOYSA-N Tetrahydrofuran Chemical compound C1CCOC1 WYURNTSHIVDZCO-UHFFFAOYSA-N 0.000 claims 4
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 claims 3
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical compound OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 claims 3
- 150000001875 compounds Chemical class 0.000 claims 3
- CDBYLPFSWZWCQE-UHFFFAOYSA-L Sodium Carbonate Chemical compound [Na+].[Na+].[O-]C([O-])=O CDBYLPFSWZWCQE-UHFFFAOYSA-L 0.000 claims 2
- WQDUMFSSJAZKTM-UHFFFAOYSA-N Sodium methoxide Chemical compound [Na+].[O-]C WQDUMFSSJAZKTM-UHFFFAOYSA-N 0.000 claims 2
- 125000002947 alkylene group Chemical group 0.000 claims 2
- 238000006243 chemical reaction Methods 0.000 claims 2
- 125000000113 cyclohexyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 claims 2
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 2
- 125000001183 hydrocarbyl group Chemical group 0.000 claims 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 2
- 125000000959 isobutyl group Chemical group [H]C([H])([H])C([H])(C([H])([H])[H])C([H])([H])* 0.000 claims 2
- 125000001972 isopentyl group Chemical group [H]C([H])([H])C([H])(C([H])([H])[H])C([H])([H])C([H])([H])* 0.000 claims 2
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
- 125000004108 n-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 2
- 125000000740 n-pentyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 2
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 2
- BWHMMNNQKKPAPP-UHFFFAOYSA-L potassium carbonate Chemical compound [K+].[K+].[O-]C([O-])=O BWHMMNNQKKPAPP-UHFFFAOYSA-L 0.000 claims 2
- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 claims 2
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 claims 2
- 125000006219 1-ethylpentyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C([H])([H])[H] 0.000 claims 1
- 125000006176 2-ethylbutyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(C([H])([H])*)C([H])([H])C([H])([H])[H] 0.000 claims 1
- 125000003229 2-methylhexyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])(C([H])([H])[H])C([H])([H])* 0.000 claims 1
- 125000004337 3-ethylpentyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(C([H])([H])C([H])([H])[H])C([H])([H])C([H])([H])* 0.000 claims 1
- 125000003469 3-methylhexyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])(C([H])([H])[H])C([H])([H])C([H])([H])* 0.000 claims 1
- 125000005917 3-methylpentyl group Chemical group 0.000 claims 1
- GAWIXWVDTYZWAW-UHFFFAOYSA-N C[CH]O Chemical group C[CH]O GAWIXWVDTYZWAW-UHFFFAOYSA-N 0.000 claims 1
- ZLMJMSJWJFRBEC-UHFFFAOYSA-N Potassium Chemical compound [K] ZLMJMSJWJFRBEC-UHFFFAOYSA-N 0.000 claims 1
- GHVZOJONCUEWAV-UHFFFAOYSA-N [K].CCO Chemical compound [K].CCO GHVZOJONCUEWAV-UHFFFAOYSA-N 0.000 claims 1
- 150000001298 alcohols Chemical class 0.000 claims 1
- 229910052783 alkali metal Inorganic materials 0.000 claims 1
- 150000001340 alkali metals Chemical class 0.000 claims 1
- 229910052784 alkaline earth metal Inorganic materials 0.000 claims 1
- 125000001511 cyclopentyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 claims 1
- 150000002170 ethers Chemical class 0.000 claims 1
- 125000005842 heteroatom Chemical group 0.000 claims 1
- 125000004051 hexyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 1
- 125000004491 isohexyl group Chemical group C(CCC(C)C)* 0.000 claims 1
- 125000001421 myristyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
- 125000003136 n-heptyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 1
- 125000001280 n-hexyl group Chemical group C(CCCCC)* 0.000 claims 1
- 229910052757 nitrogen Inorganic materials 0.000 claims 1
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 1
- 239000003960 organic solvent Substances 0.000 claims 1
- 125000002958 pentadecyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
- 229910052700 potassium Inorganic materials 0.000 claims 1
- 239000011591 potassium Substances 0.000 claims 1
- 229910000027 potassium carbonate Inorganic materials 0.000 claims 1
- 125000002914 sec-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 1
- 125000003548 sec-pentyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 1
- 229910000029 sodium carbonate Inorganic materials 0.000 claims 1
- QDRKDTQENPPHOJ-UHFFFAOYSA-N sodium ethoxide Chemical compound [Na+].CC[O-] QDRKDTQENPPHOJ-UHFFFAOYSA-N 0.000 claims 1
- 125000002889 tridecyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
- 125000002948 undecyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR1054536A FR2961206B1 (fr) | 2010-06-09 | 2010-06-09 | Procede de preparation de composes esteramides |
| FR1054536 | 2010-06-09 | ||
| PCT/EP2011/058985 WO2011154292A1 (fr) | 2010-06-09 | 2011-05-31 | Procede de preparation de composes estaramides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013531640A JP2013531640A (ja) | 2013-08-08 |
| JP2013531640A5 true JP2013531640A5 (https=) | 2014-07-17 |
Family
ID=42782066
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013513621A Ceased JP2013531640A (ja) | 2010-06-09 | 2011-05-31 | エステルアミド化合物を調製する方法 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US9296683B2 (https=) |
| EP (1) | EP2580185B1 (https=) |
| JP (1) | JP2013531640A (https=) |
| CN (1) | CN103140472B (https=) |
| BR (1) | BR112012031312B1 (https=) |
| ES (1) | ES2513565T3 (https=) |
| FR (1) | FR2961206B1 (https=) |
| WO (1) | WO2011154292A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2957596B1 (fr) * | 2010-03-18 | 2013-07-12 | Rhodia Operations | Nouveaux composes de type esteramide, leurs procedes de preparation et leurs utilisations |
| FR2961205B1 (fr) * | 2010-06-09 | 2012-06-29 | Rhodia Operations | Procede de preparation de composes esteramides |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3288794A (en) | 1962-09-12 | 1966-11-29 | C P Hall Company Of Illinois | Method of making amides of dimethylamine and piperazine |
| US3417114A (en) | 1965-07-20 | 1968-12-17 | C P Hall Company Of Illinois | Method of making amides from moisture and acid-gas containing esters |
| EP0143303A3 (de) | 1983-10-29 | 1986-04-30 | Bayer Ag | Verfahren zur Herstellung von substituierten Bernsteinsäureamiden |
| CA2036996A1 (en) * | 1990-02-26 | 1991-08-27 | William Vanderlinde | Process for preparing metal-free fatty peroxyacid precursors having amide moieties in the fatty chain |
| GB2255681B (en) * | 1991-05-08 | 1994-09-07 | Sony Corp | Analog-to-digital converter |
| US5235093A (en) * | 1992-01-27 | 1993-08-10 | Monsanto Company | Process for preparing carboxylic amide ester |
| US5166407A (en) * | 1992-01-27 | 1992-11-24 | Monsanto Company | Process for preparing fatty peroxyacid precursors having amide moieties in the fatty chain |
| CN100537552C (zh) * | 2007-05-16 | 2009-09-09 | 江苏豪森药业股份有限公司 | 一种制备瑞格列奈的方法 |
| CA2712318C (fr) * | 2008-01-25 | 2015-12-08 | Rhodia Operations | Utilisation d'esteramides a titre de solvants, esteramides en tant que tels et procede de preparation d'esteramides |
| CN102625799A (zh) * | 2009-06-25 | 2012-08-01 | 安姆根有限公司 | 杂环化合物及其用途 |
| FR2961205B1 (fr) * | 2010-06-09 | 2012-06-29 | Rhodia Operations | Procede de preparation de composes esteramides |
-
2010
- 2010-06-09 FR FR1054536A patent/FR2961206B1/fr not_active Expired - Fee Related
-
2011
- 2011-05-31 JP JP2013513621A patent/JP2013531640A/ja not_active Ceased
- 2011-05-31 EP EP11722108.5A patent/EP2580185B1/fr active Active
- 2011-05-31 WO PCT/EP2011/058985 patent/WO2011154292A1/fr not_active Ceased
- 2011-05-31 US US13/702,453 patent/US9296683B2/en active Active
- 2011-05-31 ES ES11722108.5T patent/ES2513565T3/es active Active
- 2011-05-31 BR BR112012031312A patent/BR112012031312B1/pt not_active IP Right Cessation
- 2011-05-31 CN CN201180031817.XA patent/CN103140472B/zh active Active
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2013528200A5 (https=) | ||
| PE20091033A1 (es) | Derivados de nicotinamida como agentes anticancerosos y su preparacion | |
| PH12012502223A1 (en) | Composition , method and use | |
| UA109883C2 (uk) | Спосіб отримання сполук для застосування як інгібіторів sglt2 | |
| MX2009012885A (es) | Nuevo derivado de 1,2,3,4-tetrahidroquinoxalina que tiene, como sustituyente, grupo fenilo que tiene estructura de ester de acido sulfonico o estructura de amida de acido sulfonico introducida en este, y tiene actividad de enlace al receptor de gluco | |
| JO3098B1 (ar) | مركبات داي فينيل- بيرازول بيريدين وطريقة تحضيرها واستخدامها كمعدلات المستقبل النووي not | |
| MX2010004893A (es) | Compuesto heterociclico y composicion farmaceutica del mismo. | |
| PE20100487A1 (es) | Nuevo procedimiento de sintesis de la ivabradina y de sus sales de adicion a un acido farmaceuticamente aceptable | |
| MY148930A (en) | Process for the preparation of functionalised benzocyclobutenes, and application in the synthesis of ivabradine and addition salts thereof with a pharmaceutically acceptable acid | |
| JP2013528200A (ja) | エステルアミド化合物を調製する方法 | |
| UA101482C2 (ru) | Способ получения 2'-дезокси-5-азацитидина (децитабина) | |
| MX2013000288A (es) | Metodo para fabricar quinolina-3-carboxamidas. | |
| HRP20141004T1 (hr) | Novi postupak pripreme estera skopina | |
| AR051373A1 (es) | Procedimiento para la preparacion de analogos aciclicos de nucleotidos de fosfonatos | |
| JP2013531640A5 (https=) | ||
| RU2010115566A (ru) | Ускоренное восстановление амидов и сложных эфиров аминоборанами и добавками | |
| CO6341560A2 (es) | Proceso para la preparacion de derivados de pirimidina sustituidos. | |
| RU2012142223A (ru) | Пространственно-затрудненные амины | |
| MX2013008595A (es) | Procedimiento mejorado para la preparacion de 2,2-difluoroetilamina. | |
| PH12013500001A1 (en) | Formulations | |
| RU2013110311A (ru) | Синтез соединений тиазолидиндиона | |
| AR051936A1 (es) | Proceso para la preparacion de pirazoles | |
| MX2011008751A (es) | Proceso quimico para la produccion de eteres de haloalquenona. | |
| TW200700419A (en) | 5,6-dialkyl-7-aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds | |
| RU2016146200A (ru) | Способ производства эфира (мет)акриловой кислоты и способ производства ароматического эфира карбоновой кислоты |