JP2013522273A5 - - Google Patents
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- Publication number
- JP2013522273A5 JP2013522273A5 JP2012557537A JP2012557537A JP2013522273A5 JP 2013522273 A5 JP2013522273 A5 JP 2013522273A5 JP 2012557537 A JP2012557537 A JP 2012557537A JP 2012557537 A JP2012557537 A JP 2012557537A JP 2013522273 A5 JP2013522273 A5 JP 2013522273A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- alkyl
- oxo
- quin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10156681.8 | 2010-03-16 | ||
| EP10156681 | 2010-03-16 | ||
| PCT/EP2011/053957 WO2011113859A1 (en) | 2010-03-16 | 2011-03-16 | Processes and intermediates for preparing a macrocyclic protease inhibitor of hcv |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016021576A Division JP2016164143A (ja) | 2010-03-16 | 2016-02-08 | Ｈｃｖの大環状プロテアーゼ阻害剤の製造のための方法及び中間体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013522273A JP2013522273A (ja) | 2013-06-13 |
| JP2013522273A5 true JP2013522273A5 (https=) | 2014-06-19 |
Family
ID=42342793
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012557537A Withdrawn JP2013522273A (ja) | 2010-03-16 | 2011-03-16 | Ｈｃｖの大環状プロテアーゼ阻害剤の製造のための方法及び中間体 |
| JP2016021576A Pending JP2016164143A (ja) | 2010-03-16 | 2016-02-08 | Ｈｃｖの大環状プロテアーゼ阻害剤の製造のための方法及び中間体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016021576A Pending JP2016164143A (ja) | 2010-03-16 | 2016-02-08 | Ｈｃｖの大環状プロテアーゼ阻害剤の製造のための方法及び中間体 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US9586893B2 (https=) |
| EP (2) | EP2547645B1 (https=) |
| JP (2) | JP2013522273A (https=) |
| KR (1) | KR20130034012A (https=) |
| CN (1) | CN103249708A (https=) |
| AU (1) | AU2011229164B2 (https=) |
| BR (1) | BR112012023296B1 (https=) |
| CA (1) | CA2793129A1 (https=) |
| IL (1) | IL221242A (https=) |
| MX (1) | MX2012010678A (https=) |
| RU (1) | RU2628081C2 (https=) |
| WO (1) | WO2011113859A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9586893B2 (en) * | 2010-03-16 | 2017-03-07 | Janssen Pharmaceuticals | Processes and intermediates for preparing a macrocyclic protease inhibitor of HCV |
| CA2845720A1 (en) | 2011-09-22 | 2013-03-28 | Janssen Pharmaceuticals, Inc. | Processes and intermediates for preparing a macrocyclic protease inhibitor of hcv |
| WO2016105333A1 (en) * | 2014-12-22 | 2016-06-30 | Colgate-Palmolive Company | Unit dose fabric softener |
| MA41812A (fr) | 2015-03-27 | 2018-01-30 | Janssen Pharmaceuticals Inc | Procédés et intermédiaires pour la préparation d'un inhibiteur de protéase macrocyclique du vhc |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL8300536A (nl) | 1983-02-14 | 1984-09-03 | Oce Andeno Bv | Optisch actief alfa-azido-p-hydroxyfenylazijnzuur en zijn zouten alsmede de bereiding daarvan. |
| JPS6124539A (ja) * | 1984-07-11 | 1986-02-03 | Sagami Chem Res Center | 光学活性（ｒ）−２，５，１２−トリヒドロキシ−１，２，３，４−テトラヒドロナフタセン−６，１１−ジオン−２−カルボン酸の取得方法 |
| JPH06124539A (ja) | 1992-10-08 | 1994-05-06 | Sony Corp | ディジタルｖｔｒ |
| JPH08231469A (ja) | 1995-02-23 | 1996-09-10 | Nippon Kayaku Co Ltd | シクロペンタンカルボン酸誘導体及びその製造法 |
| JPH11180930A (ja) * | 1997-12-22 | 1999-07-06 | Sumitomo Chem Co Ltd | 光学活性ｔｒａｎｓ−シクロブタンジカルボン酸類の製造方法 |
| DE10029139A1 (de) * | 2000-06-14 | 2002-01-03 | Sueddeutsche Kalkstickstoff | Verfahren zur Herstellung von Amiden oder Estern |
| PL1713822T3 (pl) | 2004-01-30 | 2010-08-31 | Medivir Ab | Inhibitory proteazy serynowej HCV NS-3 |
| PE20070211A1 (es) | 2005-07-29 | 2007-05-12 | Medivir Ab | Compuestos macrociclicos como inhibidores del virus de hepatitis c |
| BRPI0614620A2 (pt) * | 2005-07-29 | 2011-04-12 | Tibotec Pharm Ltd | compostos inibidores macrocìclicos do vìrus da hepatite c, uso dos mesmos, processo para preparar os referidos compostos, combinação e composição farmacêutica |
| US20070185346A1 (en) * | 2006-02-03 | 2007-08-09 | Vaidya Niteen A | Kit for automated resolving agent selection and method thereof |
| DE602008001251D1 (de) * | 2007-02-01 | 2010-06-24 | Tibotec Pharm Ltd | Verfahren und zwischenprodukte zur herstellung eines makrozyklischen proteasehemmers von hcv |
| US9586893B2 (en) * | 2010-03-16 | 2017-03-07 | Janssen Pharmaceuticals | Processes and intermediates for preparing a macrocyclic protease inhibitor of HCV |
-
2011
- 2011-03-16 US US13/634,996 patent/US9586893B2/en not_active Expired - Fee Related
- 2011-03-16 BR BR112012023296-7A patent/BR112012023296B1/pt not_active IP Right Cessation
- 2011-03-16 WO PCT/EP2011/053957 patent/WO2011113859A1/en not_active Ceased
- 2011-03-16 CN CN2011800140694A patent/CN103249708A/zh active Pending
- 2011-03-16 RU RU2012143977A patent/RU2628081C2/ru not_active IP Right Cessation
- 2011-03-16 CA CA2793129A patent/CA2793129A1/en not_active Abandoned
- 2011-03-16 EP EP11709692.5A patent/EP2547645B1/en active Active
- 2011-03-16 MX MX2012010678A patent/MX2012010678A/es active IP Right Grant
- 2011-03-16 EP EP17166514.4A patent/EP3239129A1/en not_active Withdrawn
- 2011-03-16 KR KR1020127024789A patent/KR20130034012A/ko not_active Ceased
- 2011-03-16 JP JP2012557537A patent/JP2013522273A/ja not_active Withdrawn
- 2011-03-16 AU AU2011229164A patent/AU2011229164B2/en not_active Ceased
-
2012
- 2012-08-01 IL IL221242A patent/IL221242A/en not_active IP Right Cessation
-
2016
- 2016-02-08 JP JP2016021576A patent/JP2016164143A/ja active Pending
-
2017
- 2017-02-10 US US15/429,250 patent/US20170152253A1/en not_active Abandoned
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