JP2013521288A5 - - Google Patents
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- Publication number
- JP2013521288A5 JP2013521288A5 JP2012556126A JP2012556126A JP2013521288A5 JP 2013521288 A5 JP2013521288 A5 JP 2013521288A5 JP 2012556126 A JP2012556126 A JP 2012556126A JP 2012556126 A JP2012556126 A JP 2012556126A JP 2013521288 A5 JP2013521288 A5 JP 2013521288A5
- Authority
- JP
- Japan
- Prior art keywords
- hydroxy
- aryl
- alkyl
- heterocyclyl
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 *C(N=C(*)N(*)C1=O)=C1O Chemical compound *C(N=C(*)N(*)C1=O)=C1O 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US31038610P | 2010-03-04 | 2010-03-04 | |
| US61/310,386 | 2010-03-04 | ||
| PCT/US2011/026424 WO2011109267A1 (en) | 2010-03-04 | 2011-02-28 | Inhibitors of catechol o-methyl transferase and their use in the treatment of psychotic disorders |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013521288A JP2013521288A (ja) | 2013-06-10 |
| JP2013521288A5 true JP2013521288A5 (https=) | 2014-04-17 |
| JP5937971B2 JP5937971B2 (ja) | 2016-06-22 |
Family
ID=44542514
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012556126A Expired - Fee Related JP5937971B2 (ja) | 2010-03-04 | 2011-02-28 | カテコールｏ−メチルトランスフェラーゼの阻害剤および精神障害の治療におけるその使用 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US8969364B2 (https=) |
| EP (1) | EP2542084B1 (https=) |
| JP (1) | JP5937971B2 (https=) |
| KR (1) | KR101761963B1 (https=) |
| CN (1) | CN102858177B (https=) |
| AU (1) | AU2011223888B2 (https=) |
| BR (1) | BR112012021656A2 (https=) |
| CA (1) | CA2789475C (https=) |
| DK (1) | DK2542084T3 (https=) |
| ES (1) | ES2662332T3 (https=) |
| HU (1) | HUE036431T2 (https=) |
| MX (1) | MX336711B (https=) |
| NO (1) | NO2542084T3 (https=) |
| PL (1) | PL2542084T3 (https=) |
| PT (1) | PT2542084T (https=) |
| RU (1) | RU2572624C2 (https=) |
| WO (1) | WO2011109267A1 (https=) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201111704D0 (en) | 2011-07-07 | 2011-08-24 | Takeda Pharmaceutical | Novel compounds |
| GB201111705D0 (en) | 2011-07-07 | 2011-08-24 | Takeda Pharmaceutical | Compounds and their use |
| JO3115B1 (ar) | 2011-08-22 | 2017-09-20 | Takeda Pharmaceuticals Co | مركبات بيريدازينون واستخدامها كمثبطات daao |
| AU2012337781B2 (en) | 2011-11-15 | 2017-07-06 | Takeda Pharmaceutical Company Limited | Dihydroxy aromatic heterocyclic compound |
| TWI638802B (zh) | 2012-05-24 | 2018-10-21 | 芬蘭商奧利安公司 | 兒茶酚ｏ－甲基轉移酶活性抑制化合物 |
| BR112014030284B1 (pt) | 2012-07-18 | 2021-11-30 | Sunshine Lake Pharma Co., Ltd | Composto, composição farmacêutica, e, uso de um composto ou de uma composição farmacêutica |
| WO2014043252A2 (en) * | 2012-09-11 | 2014-03-20 | Rutgers, The State University Of New Jersey | Therapeutic hydroxypyridinones, hydroxypyrimidinones and hydroxypyridazinones |
| GB201222711D0 (en) | 2012-12-17 | 2013-01-30 | Takeda Pharmaceutical | Novel compounds |
| KR101685862B1 (ko) | 2012-12-27 | 2016-12-20 | 에프. 호프만-라 로슈 아게 | Comt 억제제 |
| DK3013813T3 (da) | 2013-06-27 | 2019-06-03 | Pfizer | Heteroaromatiske forbindelser og anvendelse deraf som dopamin-d1-ligander |
| US9902712B2 (en) | 2013-12-19 | 2018-02-27 | Sunshine Lake Pharma Co., Ltd. | Nitrogenous heterocyclic derivatives and their application in drugs |
| PL236355B1 (pl) | 2015-04-02 | 2021-01-11 | Celon Pharma Spolka Akcyjna | Pochodne 7-(morfolin-4-ylo)pirazolo[1,5-α]pirymidyny jako inhibitory kinazy PI3 |
| EP3733188B1 (en) * | 2015-06-08 | 2023-01-25 | The Regents of the University of California | Use of h3k9me3 modulation for enhancing cognitive function |
| AU2019395201A1 (en) | 2018-12-06 | 2021-05-20 | Daiichi Sankyo Company, Limited | Cycloalkane-1,3-diamine derivative |
| CN113499525A (zh) * | 2021-08-25 | 2021-10-15 | 骆艳 | 一种针对发展性阅读障碍儿童的训练系统 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3631045A (en) * | 1969-11-04 | 1971-12-28 | American Home Prod | 4 5-diamino-7h-pyrrolo(2 3-d)pyrimidine derivatives |
| US3910913A (en) * | 1969-11-04 | 1975-10-07 | American Home Prod | 4,5-Diamino-7H-pyrrolo{8 2,3-d{9 pyrimidine derivatives |
| DOP1981004033A (es) * | 1980-12-23 | 1990-12-29 | Ciba Geigy Ag | Procedimiento para proteger plantas de cultivo de la accion fitotoxica de herbicidas. |
| US5726124A (en) * | 1992-07-17 | 1998-03-10 | Rohm And Haas Company | 2-arylpyrimidines and herbicidal use thereof |
| CA2416248A1 (en) | 2000-07-18 | 2002-01-24 | Neurogen Corporation | 5-substituted 2-aryl-4-pyrimidinones |
| SE0004053D0 (sv) * | 2000-11-06 | 2000-11-06 | Astrazeneca Ab | N-type calcium channel antagonists for the treatment of pain |
| IL161337A0 (en) * | 2001-10-26 | 2004-09-27 | Angeletti P Ist Richerche Bio | N-substituted hydroxypyrimidinone carboxamide inhibitors of hiv integrase |
| RU2004135554A (ru) * | 2002-05-09 | 2006-01-20 | Цитокинетикс, Инк. (Us) | Пиримидиноны, композиции на их основе и способы их использования |
| US6930117B2 (en) | 2002-11-09 | 2005-08-16 | The Procter & Gamble Company | N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones |
| US8455489B2 (en) * | 2003-11-10 | 2013-06-04 | Exelixis, Inc. | Substituted pyrimidine compositions and methods of use |
| TW200526635A (en) * | 2003-12-22 | 2005-08-16 | Shionogi & Co | Hydroxypyrimidinone derivative having HIV integrase inhibitory activity |
| GB0515327D0 (en) * | 2005-07-26 | 2005-08-31 | Portela & Ca Sa | Comt inhibitors |
| JP2009007273A (ja) * | 2007-06-27 | 2009-01-15 | Ajinomoto Co Inc | ジアミノピリミジン化合物の製造方法 |
| CN101747282A (zh) * | 2008-12-10 | 2010-06-23 | 上海特化医药科技有限公司 | 一类含有嘧啶酮苯基的化合物、其药物组合物及其制备方法和用途 |
| JP5442852B2 (ja) * | 2009-08-13 | 2014-03-12 | 田辺三菱製薬株式会社 | タウプロテインキナーゼ１阻害剤としてのピリミドン誘導体 |
| US9328075B2 (en) * | 2011-05-05 | 2016-05-03 | St. Jude Children's Research Hospital | Pyrimidinone compounds and methods for treating influenza |
-
2011
- 2011-02-28 US US13/582,637 patent/US8969364B2/en active Active
- 2011-02-28 AU AU2011223888A patent/AU2011223888B2/en not_active Ceased
- 2011-02-28 PT PT117511295T patent/PT2542084T/pt unknown
- 2011-02-28 PL PL11751129T patent/PL2542084T3/pl unknown
- 2011-02-28 CN CN201180012339.8A patent/CN102858177B/zh not_active Expired - Fee Related
- 2011-02-28 RU RU2012142171/04A patent/RU2572624C2/ru not_active IP Right Cessation
- 2011-02-28 ES ES11751129.5T patent/ES2662332T3/es active Active
- 2011-02-28 DK DK11751129.5T patent/DK2542084T3/en active
- 2011-02-28 CA CA2789475A patent/CA2789475C/en active Active
- 2011-02-28 EP EP11751129.5A patent/EP2542084B1/en active Active
- 2011-02-28 WO PCT/US2011/026424 patent/WO2011109267A1/en not_active Ceased
- 2011-02-28 BR BR112012021656A patent/BR112012021656A2/pt active Search and Examination
- 2011-02-28 NO NO11751129A patent/NO2542084T3/no unknown
- 2011-02-28 JP JP2012556126A patent/JP5937971B2/ja not_active Expired - Fee Related
- 2011-02-28 MX MX2012010189A patent/MX336711B/es unknown
- 2011-02-28 KR KR1020127023050A patent/KR101761963B1/ko not_active Expired - Fee Related
- 2011-02-28 HU HUE11751129A patent/HUE036431T2/hu unknown