JP2013518812A5 - - Google Patents
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- Publication number
- JP2013518812A5 JP2013518812A5 JP2012549078A JP2012549078A JP2013518812A5 JP 2013518812 A5 JP2013518812 A5 JP 2013518812A5 JP 2012549078 A JP2012549078 A JP 2012549078A JP 2012549078 A JP2012549078 A JP 2012549078A JP 2013518812 A5 JP2013518812 A5 JP 2013518812A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- alkenyl
- aryl
- halo
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29474110P | 2010-01-13 | 2010-01-13 | |
| US61/294,741 | 2010-01-13 | ||
| PCT/US2011/021129 WO2011088209A2 (en) | 2010-01-13 | 2011-01-13 | 1-deoxy analogs of vitamin d-related compounds |
Related Child Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015136522A Division JP2015212294A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
| JP2015136520A Division JP2016006055A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
| JP2015136521A Division JP2016006056A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013518812A JP2013518812A (ja) | 2013-05-23 |
| JP2013518812A5 true JP2013518812A5 (enExample) | 2014-03-06 |
| JP5887672B2 JP5887672B2 (ja) | 2016-03-16 |
Family
ID=44010128
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012549078A Expired - Fee Related JP5887672B2 (ja) | 2010-01-13 | 2011-01-13 | ビタミンd関連化合物の1−デオキシ類似体 |
| JP2015136521A Pending JP2016006056A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
| JP2015136520A Pending JP2016006055A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
| JP2015136522A Pending JP2015212294A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015136521A Pending JP2016006056A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
| JP2015136520A Pending JP2016006055A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
| JP2015136522A Pending JP2015212294A (ja) | 2010-01-13 | 2015-07-07 | ビタミンd関連化合物の1−デオキシ類似体 |
Country Status (3)
| Country | Link |
|---|---|
| US (3) | US9775903B2 (enExample) |
| JP (4) | JP5887672B2 (enExample) |
| WO (1) | WO2011088209A2 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9775903B2 (en) * | 2010-01-13 | 2017-10-03 | Johns Hopkins University | 1-deoxy analogs of 1,25-dihydroxyvitamin D3 compounds |
| GB2512314A (en) * | 2013-03-26 | 2014-10-01 | Kartar Singh Lalvani | Statin composition |
| CN105348163B (zh) * | 2014-08-18 | 2017-06-16 | 武汉启瑞药业有限公司 | 维生素d类似物及其制备方法和医药用途 |
| WO2018230711A1 (ja) | 2017-06-16 | 2018-12-20 | 学校法人同志社 | mTORインヒビターを含む、眼の症状、障害または疾患を治療または予防するための医薬およびその応用 |
| US20230398130A1 (en) * | 2020-10-23 | 2023-12-14 | Massachusetts Institute Of Technology | Methods and compositions for differentiating stem cells |
| WO2025094144A1 (en) | 2023-11-02 | 2025-05-08 | Eirgen Pharma Ltd. | Controlling loss of kidney function |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5830885A (en) | 1992-03-12 | 1998-11-03 | The Johns Hopkins University | Antiproliferative vitamin D3 hybrids |
| DE60031666T2 (de) * | 1999-04-01 | 2007-08-30 | The Johns Hopkins University | NICHT-CALCEMISCHE, TRANSKRIPTIONELL-AKTIVE, SCHWEFELHALTIGE ANALOGA VON 1-alpha, 25-DIHYDROXYVITAMIN D3 MIT ANTIPROLIFERATIVER WIRKUNG |
| WO2001028565A1 (en) * | 1999-10-19 | 2001-04-26 | Juichiro Nakayama | Remedies for pigmentation and melanocyte proliferation inhibitors |
| JP2002104995A (ja) * | 2000-09-29 | 2002-04-10 | Masahiko Hosaka | テロメラーゼ活性抑制剤 |
| US7166585B2 (en) * | 2001-08-22 | 2007-01-23 | Cytochroma Inc. | 24-Sulfur-substituted analogs of 1α,25-dihydroxy vitamin D3 |
| ES2283593T3 (es) | 2001-10-12 | 2007-11-01 | Johns Hopkins University | Analogos de oxima poco calcemicos de 1alfa,25-dihidroxi vitamina d3. |
| AU2003233735A1 (en) | 2002-06-13 | 2003-12-31 | Cytochroma Inc. | 24-sulfoximine vitamin d3 compounds |
| TWI286554B (en) * | 2002-06-27 | 2007-09-11 | Chugai Pharmaceutical Co Ltd | Ferrocene compounds and uses thereof |
| WO2004037781A1 (en) * | 2002-10-23 | 2004-05-06 | Leo Pharma A/S | Vitamin d analogues, compositions comprising said analogues and their use |
| WO2004054968A2 (en) * | 2002-12-18 | 2004-07-01 | Johns Hopkins University | 25-so2-substituted analogs of 1alpha, 25-dihydroxyvitamin d3 (calcitriol) |
| EP1883626B1 (en) * | 2005-04-25 | 2017-10-11 | OPKO Ireland Global Holdings, Ltd. | Low-calcemic 16,23-diene 25-oxime analogs of 1alpha,25-dihydroxy vitamin d3 |
| JP4882050B2 (ja) * | 2006-03-15 | 2012-02-22 | 日本マイクロバイオファーマ株式会社 | インデン誘導体の製造方法およびその製造中間体 |
| JP2009532458A (ja) | 2006-04-06 | 2009-09-10 | ウイスコンシン アラムニ リサーチ ファンデーション | 2−メチレン−1α−ヒドロキシ−19,21−ジノルビタミンD3類縁体およびその使用 |
| US9775903B2 (en) * | 2010-01-13 | 2017-10-03 | Johns Hopkins University | 1-deoxy analogs of 1,25-dihydroxyvitamin D3 compounds |
-
2011
- 2011-01-13 US US13/521,980 patent/US9775903B2/en not_active Expired - Fee Related
- 2011-01-13 WO PCT/US2011/021129 patent/WO2011088209A2/en not_active Ceased
- 2011-01-13 JP JP2012549078A patent/JP5887672B2/ja not_active Expired - Fee Related
-
2015
- 2015-07-07 JP JP2015136521A patent/JP2016006056A/ja active Pending
- 2015-07-07 JP JP2015136520A patent/JP2016006055A/ja active Pending
- 2015-07-07 JP JP2015136522A patent/JP2015212294A/ja active Pending
-
2017
- 2017-10-02 US US15/722,694 patent/US20180117156A1/en not_active Abandoned
-
2018
- 2018-10-25 US US16/170,487 patent/US20190060456A1/en not_active Abandoned
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