JP2013509435A - 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン - Google Patents
長時間作用型注入可能パリペリドンエステルに関連した投与レジメン Download PDFInfo
- Publication number
- JP2013509435A JP2013509435A JP2012537131A JP2012537131A JP2013509435A JP 2013509435 A JP2013509435 A JP 2013509435A JP 2012537131 A JP2012537131 A JP 2012537131A JP 2012537131 A JP2012537131 A JP 2012537131A JP 2013509435 A JP2013509435 A JP 2013509435A
- Authority
- JP
- Japan
- Prior art keywords
- dose
- patient
- paliperidone
- paliperidone palmitate
- palmitate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Images
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Neurology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25669609P | 2009-10-30 | 2009-10-30 | |
| US61/256,696 | 2009-10-30 | ||
| PCT/US2010/054807 WO2011053829A1 (en) | 2009-10-30 | 2010-10-29 | Dosing regimen associated with long-acting injectable paliperidone esters |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015237117A Division JP2016102123A (ja) | 2009-10-30 | 2015-12-04 | 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013509435A true JP2013509435A (ja) | 2013-03-14 |
| JP2013509435A5 JP2013509435A5 (enExample) | 2013-12-19 |
Family
ID=43302985
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012537131A Pending JP2013509435A (ja) | 2009-10-30 | 2010-10-29 | 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン |
| JP2015237117A Pending JP2016102123A (ja) | 2009-10-30 | 2015-12-04 | 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015237117A Pending JP2016102123A (ja) | 2009-10-30 | 2015-12-04 | 長時間作用型注入可能パリペリドンエステルに関連した投与レジメン |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US20110105536A1 (enExample) |
| EP (1) | EP2493473A1 (enExample) |
| JP (2) | JP2013509435A (enExample) |
| KR (1) | KR20120116401A (enExample) |
| CN (1) | CN102802631A (enExample) |
| AU (2) | AU2010313290A1 (enExample) |
| BR (1) | BR112012010195A2 (enExample) |
| CA (1) | CA2742393A1 (enExample) |
| CL (1) | CL2012001110A1 (enExample) |
| MX (1) | MX2012005083A (enExample) |
| NZ (1) | NZ599558A (enExample) |
| WO (1) | WO2011053829A1 (enExample) |
Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018510894A (ja) * | 2015-04-07 | 2018-04-19 | ヤンセン ファーマシューティカルズ,インコーポレーテッド | 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン |
| JP2023551009A (ja) * | 2020-11-30 | 2023-12-06 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
| JP2023552149A (ja) * | 2020-11-30 | 2023-12-14 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
| JP2023552329A (ja) * | 2020-11-30 | 2023-12-15 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
| JP7792409B2 (ja) | 2020-11-30 | 2025-12-25 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA72189C2 (uk) | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
| SI2234617T2 (sl) | 2007-12-19 | 2025-05-30 | Janssen Pharmaceutica Nv | Režim odmerjanja v zvezi z dolgodelujočimi paliperidonijevimi estri za injiciranje |
| US9271939B2 (en) | 2010-03-15 | 2016-03-01 | Inventia Healthcare Private Limited | Stabilized prolonged release pharmaceutical composition comprising atypical antipsychotic |
| FI3156056T3 (fi) | 2011-03-18 | 2024-03-01 | Alkermes Pharma Ireland Ltd | Sorbitaaniestereitä käsittäviä farmaseuttisia koostumuksia |
| CN102993200B (zh) * | 2011-09-10 | 2016-02-03 | 鲁翠涛 | 帕潘立酮氨基酸酯及其制备方法 |
| ES2950418T3 (es) | 2012-03-19 | 2023-10-09 | Alkermes Pharma Ireland Ltd | Composiciones farmacéuticas que comprenden alcohol bencílico |
| US10004807B2 (en) | 2012-03-19 | 2018-06-26 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising fatty acid esters |
| WO2013142202A1 (en) | 2012-03-19 | 2013-09-26 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising glycerol esters |
| CA2885196C (en) | 2012-09-19 | 2021-06-22 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions having improved storage stability |
| CN106132415A (zh) | 2014-03-20 | 2016-11-16 | 奥克梅斯制药爱尔兰有限公司 | 具有增加的注射速度的阿立哌唑制剂 |
| ITUB20155193A1 (it) * | 2015-11-03 | 2017-05-03 | Italfarmaco Spa | Sospensioni orali di Givinostat fisicamente e chimicamente stabili |
| US11273158B2 (en) | 2018-03-05 | 2022-03-15 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
| US12431230B2 (en) | 2019-09-25 | 2025-09-30 | Janssen Pharmaceuticals, Inc. | Interconnection of drug administration systems |
| EP4208217A1 (en) * | 2020-09-02 | 2023-07-12 | Janssen Pharmaceutica NV | Pre-filled syringe with optimized stopper placement |
| EP4308077A1 (en) * | 2021-03-17 | 2024-01-24 | MedinCell S.A. | Long acting injectable formulation comprising risperidone and biodegradable polymers |
| CA3229731A1 (en) | 2021-08-20 | 2023-02-23 | Janssen Pharmaceutica Nv | Dosing regimens associated with extended release paliperidone injectable formulations |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2008074852A (ja) * | 2006-09-22 | 2008-04-03 | Janssen Pharmaceut Nv | 肝機能が低下した精神医学上の患者をパリペリドンで治療 |
| JP2009524685A (ja) * | 2006-08-14 | 2009-07-02 | テバ ファーマシューティカル インダストリーズ リミティド | 9−ヒドロキシ−リスペリドン(パリペリドン)の結晶型 |
| WO2009080651A1 (en) * | 2007-12-19 | 2009-07-02 | Janssen Pharmaceutica Nv | Dosing regimen associated with long acting injectable paliperidone esters |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5254556A (en) | 1988-11-07 | 1993-10-19 | Janssen Pharmaceutica N.V. | 3-piperidinyl-1,2-benzisoxazoles |
| TW487572B (en) | 1996-05-20 | 2002-05-21 | Janssen Pharmaceutica Nv | Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters |
| UA72189C2 (uk) | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
| KR100338776B1 (ko) | 2000-07-11 | 2002-05-31 | 윤종용 | 멀티 로우 어드레스 테스트 가능한 반도체 메모리 장치 및그 테스트 방법 |
| EP1879890A1 (en) | 2005-04-25 | 2008-01-23 | Janssen Pharmaceutica N.V. | Preparation of aseptic 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4h-pyridio[1,2-a]pyrimidin-4-one palmitate ester |
-
2010
- 2010-10-29 CA CA2742393A patent/CA2742393A1/en not_active Abandoned
- 2010-10-29 NZ NZ599558A patent/NZ599558A/en not_active IP Right Cessation
- 2010-10-29 CN CN2010800504164A patent/CN102802631A/zh active Pending
- 2010-10-29 KR KR1020127013546A patent/KR20120116401A/ko not_active Ceased
- 2010-10-29 AU AU2010313290A patent/AU2010313290A1/en not_active Abandoned
- 2010-10-29 WO PCT/US2010/054807 patent/WO2011053829A1/en not_active Ceased
- 2010-10-29 MX MX2012005083A patent/MX2012005083A/es not_active Application Discontinuation
- 2010-10-29 JP JP2012537131A patent/JP2013509435A/ja active Pending
- 2010-10-29 BR BR112012010195A patent/BR112012010195A2/pt not_active IP Right Cessation
- 2010-10-29 EP EP10773821A patent/EP2493473A1/en not_active Withdrawn
- 2010-11-01 US US12/916,910 patent/US20110105536A1/en not_active Abandoned
-
2012
- 2012-04-27 CL CL2012001110A patent/CL2012001110A1/es unknown
-
2013
- 2013-05-28 US US13/903,638 patent/US20130331402A1/en not_active Abandoned
-
2015
- 2015-10-16 AU AU2015243103A patent/AU2015243103A1/en not_active Abandoned
- 2015-12-04 JP JP2015237117A patent/JP2016102123A/ja active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009524685A (ja) * | 2006-08-14 | 2009-07-02 | テバ ファーマシューティカル インダストリーズ リミティド | 9−ヒドロキシ−リスペリドン(パリペリドン)の結晶型 |
| JP2008074852A (ja) * | 2006-09-22 | 2008-04-03 | Janssen Pharmaceut Nv | 肝機能が低下した精神医学上の患者をパリペリドンで治療 |
| WO2009080651A1 (en) * | 2007-12-19 | 2009-07-02 | Janssen Pharmaceutica Nv | Dosing regimen associated with long acting injectable paliperidone esters |
Cited By (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018510894A (ja) * | 2015-04-07 | 2018-04-19 | ヤンセン ファーマシューティカルズ,インコーポレーテッド | 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン |
| JP2020090498A (ja) * | 2015-04-07 | 2020-06-11 | ヤンセン ファーマシューティカルズ,インコーポレーテッド | 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン |
| JP2021130680A (ja) * | 2015-04-07 | 2021-09-09 | ヤンセン ファーマシューティカルズ,インコーポレーテッド | 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン |
| JP7228503B2 (ja) | 2015-04-07 | 2023-02-24 | ヤンセン ファーマシューティカルズ,インコーポレーテッド | 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン |
| JP7422277B2 (ja) | 2015-04-07 | 2024-01-26 | ヤンセン ファーマシューティカ エヌ.ベー. | 長時間作用型注射可能パリペリドンエステルの抜かした投与量のための投与レジメン |
| JP2023551009A (ja) * | 2020-11-30 | 2023-12-06 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
| JP2023552149A (ja) * | 2020-11-30 | 2023-12-14 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
| JP2023552329A (ja) * | 2020-11-30 | 2023-12-15 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
| JP7792409B2 (ja) | 2020-11-30 | 2025-12-25 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
| JP7792959B2 (ja) | 2020-11-30 | 2025-12-26 | ヤンセン ファーマシューティカ エヌ.ベー. | 持続放出パリペリドン注射可能製剤に関連する投与レジメン |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2015243103A1 (en) | 2015-11-05 |
| EP2493473A1 (en) | 2012-09-05 |
| NZ599558A (en) | 2014-09-26 |
| CA2742393A1 (en) | 2011-05-05 |
| CN102802631A (zh) | 2012-11-28 |
| BR112012010195A2 (pt) | 2016-04-26 |
| CL2012001110A1 (es) | 2012-10-19 |
| MX2012005083A (es) | 2012-09-28 |
| WO2011053829A1 (en) | 2011-05-05 |
| AU2010313290A1 (en) | 2012-05-17 |
| US20110105536A1 (en) | 2011-05-05 |
| US20130331402A1 (en) | 2013-12-12 |
| JP2016102123A (ja) | 2016-06-02 |
| KR20120116401A (ko) | 2012-10-22 |
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Legal Events
| Date | Code | Title | Description |
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