KR20120116401A - 장기-작용성의 주사가능한 팔리페리돈 에스테르와 관련된 투약 요법 - Google Patents
장기-작용성의 주사가능한 팔리페리돈 에스테르와 관련된 투약 요법 Download PDFInfo
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- KR20120116401A KR20120116401A KR1020127013546A KR20127013546A KR20120116401A KR 20120116401 A KR20120116401 A KR 20120116401A KR 1020127013546 A KR1020127013546 A KR 1020127013546A KR 20127013546 A KR20127013546 A KR 20127013546A KR 20120116401 A KR20120116401 A KR 20120116401A
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- paliperidone palmitate
- paliperidone
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- GFQYVLUOOAAOGM-UHFFFAOYSA-N zirconium(iv) silicate Chemical compound [Zr+4].[O-][Si]([O-])([O-])[O-] GFQYVLUOOAAOGM-UHFFFAOYSA-N 0.000 description 1
- WFPIAZLQTJBIFN-DVZOWYKESA-N zuclopenthixol Chemical compound C1CN(CCO)CCN1CC\C=C\1C2=CC(Cl)=CC=C2SC2=CC=CC=C2/1 WFPIAZLQTJBIFN-DVZOWYKESA-N 0.000 description 1
- 229960000783 zuclopenthixol decanoate Drugs 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
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- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Neurology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| Application Number | Priority Date | Filing Date | Title |
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| US25669609P | 2009-10-30 | 2009-10-30 | |
| US61/256,696 | 2009-10-30 |
Publications (1)
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|---|---|
| KR20120116401A true KR20120116401A (ko) | 2012-10-22 |
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Family Applications (1)
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| KR1020127013546A Ceased KR20120116401A (ko) | 2009-10-30 | 2010-10-29 | 장기-작용성의 주사가능한 팔리페리돈 에스테르와 관련된 투약 요법 |
Country Status (12)
| Country | Link |
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| US (2) | US20110105536A1 (enExample) |
| EP (1) | EP2493473A1 (enExample) |
| JP (2) | JP2013509435A (enExample) |
| KR (1) | KR20120116401A (enExample) |
| CN (1) | CN102802631A (enExample) |
| AU (2) | AU2010313290A1 (enExample) |
| BR (1) | BR112012010195A2 (enExample) |
| CA (1) | CA2742393A1 (enExample) |
| CL (1) | CL2012001110A1 (enExample) |
| MX (1) | MX2012005083A (enExample) |
| NZ (1) | NZ599558A (enExample) |
| WO (1) | WO2011053829A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20170134583A (ko) * | 2015-04-07 | 2017-12-06 | 얀센 파마슈티칼즈, 인코포레이티드 | 장기간 작용형 주사용 팔리페리돈 에스테르에 대한 누락된 용량에 대한 투여 계획 |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA72189C2 (uk) | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
| SI2234617T2 (sl) | 2007-12-19 | 2025-05-30 | Janssen Pharmaceutica Nv | Režim odmerjanja v zvezi z dolgodelujočimi paliperidonijevimi estri za injiciranje |
| US9271939B2 (en) | 2010-03-15 | 2016-03-01 | Inventia Healthcare Private Limited | Stabilized prolonged release pharmaceutical composition comprising atypical antipsychotic |
| FI3156056T3 (fi) | 2011-03-18 | 2024-03-01 | Alkermes Pharma Ireland Ltd | Sorbitaaniestereitä käsittäviä farmaseuttisia koostumuksia |
| CN102993200B (zh) * | 2011-09-10 | 2016-02-03 | 鲁翠涛 | 帕潘立酮氨基酸酯及其制备方法 |
| ES2950418T3 (es) | 2012-03-19 | 2023-10-09 | Alkermes Pharma Ireland Ltd | Composiciones farmacéuticas que comprenden alcohol bencílico |
| US10004807B2 (en) | 2012-03-19 | 2018-06-26 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising fatty acid esters |
| WO2013142202A1 (en) | 2012-03-19 | 2013-09-26 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising glycerol esters |
| CA2885196C (en) | 2012-09-19 | 2021-06-22 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions having improved storage stability |
| CN106132415A (zh) | 2014-03-20 | 2016-11-16 | 奥克梅斯制药爱尔兰有限公司 | 具有增加的注射速度的阿立哌唑制剂 |
| ITUB20155193A1 (it) * | 2015-11-03 | 2017-05-03 | Italfarmaco Spa | Sospensioni orali di Givinostat fisicamente e chimicamente stabili |
| US11273158B2 (en) | 2018-03-05 | 2022-03-15 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
| US12431230B2 (en) | 2019-09-25 | 2025-09-30 | Janssen Pharmaceuticals, Inc. | Interconnection of drug administration systems |
| EP4208217A1 (en) * | 2020-09-02 | 2023-07-12 | Janssen Pharmaceutica NV | Pre-filled syringe with optimized stopper placement |
| DK4025188T3 (da) | 2020-11-30 | 2024-03-04 | Janssen Pharmaceutica Nv | Doseringsregimer associeret med injicerbare paliperidonformuleringer med forlænget frigivelse |
| EP4025189B1 (en) | 2020-11-30 | 2024-06-05 | Janssen Pharmaceutica NV | Dosing regimens associated with extended release paliperidone injectable formulations |
| EP4385564A3 (en) | 2020-11-30 | 2024-10-09 | JANSSEN Pharmaceutica NV | Dosing regimens associated with extended release paliperidone injectable formulations |
| EP4308077A1 (en) * | 2021-03-17 | 2024-01-24 | MedinCell S.A. | Long acting injectable formulation comprising risperidone and biodegradable polymers |
| CA3229731A1 (en) | 2021-08-20 | 2023-02-23 | Janssen Pharmaceutica Nv | Dosing regimens associated with extended release paliperidone injectable formulations |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5254556A (en) | 1988-11-07 | 1993-10-19 | Janssen Pharmaceutica N.V. | 3-piperidinyl-1,2-benzisoxazoles |
| TW487572B (en) | 1996-05-20 | 2002-05-21 | Janssen Pharmaceutica Nv | Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters |
| UA72189C2 (uk) | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
| KR100338776B1 (ko) | 2000-07-11 | 2002-05-31 | 윤종용 | 멀티 로우 어드레스 테스트 가능한 반도체 메모리 장치 및그 테스트 방법 |
| EP1879890A1 (en) | 2005-04-25 | 2008-01-23 | Janssen Pharmaceutica N.V. | Preparation of aseptic 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4h-pyridio[1,2-a]pyrimidin-4-one palmitate ester |
| US20070197591A1 (en) * | 2005-12-12 | 2007-08-23 | Sandra Boom | Use of paliperidone for the treatment of a mental disorder in a psychiatric patient with reduced hepatic function |
| TW200825077A (en) * | 2006-08-14 | 2008-06-16 | Teva Pharma | Crystal forms of 9-hydroxy-risperidone (paliperidone) |
| SI2234617T2 (sl) | 2007-12-19 | 2025-05-30 | Janssen Pharmaceutica Nv | Režim odmerjanja v zvezi z dolgodelujočimi paliperidonijevimi estri za injiciranje |
-
2010
- 2010-10-29 CA CA2742393A patent/CA2742393A1/en not_active Abandoned
- 2010-10-29 NZ NZ599558A patent/NZ599558A/en not_active IP Right Cessation
- 2010-10-29 CN CN2010800504164A patent/CN102802631A/zh active Pending
- 2010-10-29 KR KR1020127013546A patent/KR20120116401A/ko not_active Ceased
- 2010-10-29 AU AU2010313290A patent/AU2010313290A1/en not_active Abandoned
- 2010-10-29 WO PCT/US2010/054807 patent/WO2011053829A1/en not_active Ceased
- 2010-10-29 MX MX2012005083A patent/MX2012005083A/es not_active Application Discontinuation
- 2010-10-29 JP JP2012537131A patent/JP2013509435A/ja active Pending
- 2010-10-29 BR BR112012010195A patent/BR112012010195A2/pt not_active IP Right Cessation
- 2010-10-29 EP EP10773821A patent/EP2493473A1/en not_active Withdrawn
- 2010-11-01 US US12/916,910 patent/US20110105536A1/en not_active Abandoned
-
2012
- 2012-04-27 CL CL2012001110A patent/CL2012001110A1/es unknown
-
2013
- 2013-05-28 US US13/903,638 patent/US20130331402A1/en not_active Abandoned
-
2015
- 2015-10-16 AU AU2015243103A patent/AU2015243103A1/en not_active Abandoned
- 2015-12-04 JP JP2015237117A patent/JP2016102123A/ja active Pending
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20170134583A (ko) * | 2015-04-07 | 2017-12-06 | 얀센 파마슈티칼즈, 인코포레이티드 | 장기간 작용형 주사용 팔리페리돈 에스테르에 대한 누락된 용량에 대한 투여 계획 |
| KR20230162162A (ko) * | 2015-04-07 | 2023-11-28 | 잔센파마슈티카엔.브이. | 장기간 작용형 주사용 팔리페리돈 에스테르에 대한 누락된 용량에 대한 투여 계획 |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2015243103A1 (en) | 2015-11-05 |
| EP2493473A1 (en) | 2012-09-05 |
| NZ599558A (en) | 2014-09-26 |
| CA2742393A1 (en) | 2011-05-05 |
| JP2013509435A (ja) | 2013-03-14 |
| CN102802631A (zh) | 2012-11-28 |
| BR112012010195A2 (pt) | 2016-04-26 |
| CL2012001110A1 (es) | 2012-10-19 |
| MX2012005083A (es) | 2012-09-28 |
| WO2011053829A1 (en) | 2011-05-05 |
| AU2010313290A1 (en) | 2012-05-17 |
| US20110105536A1 (en) | 2011-05-05 |
| US20130331402A1 (en) | 2013-12-12 |
| JP2016102123A (ja) | 2016-06-02 |
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