JP2013509423A5 - - Google Patents
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- Publication number
- JP2013509423A5 JP2013509423A5 JP2012537052A JP2012537052A JP2013509423A5 JP 2013509423 A5 JP2013509423 A5 JP 2013509423A5 JP 2012537052 A JP2012537052 A JP 2012537052A JP 2012537052 A JP2012537052 A JP 2012537052A JP 2013509423 A5 JP2013509423 A5 JP 2013509423A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- methyl
- alkyl
- group
- oxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 **(C(NCC#CC(CCCC1)CCC1(*)I)=O)N Chemical compound **(C(NCC#CC(CCCC1)CCC1(*)I)=O)N 0.000 description 3
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25617109P | 2009-10-29 | 2009-10-29 | |
| US61/256,171 | 2009-10-29 | ||
| PCT/US2010/054445 WO2011059731A1 (en) | 2009-10-29 | 2010-10-28 | Alkynyl derivatives useful as dpp-1 inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013509423A JP2013509423A (ja) | 2013-03-14 |
| JP2013509423A5 true JP2013509423A5 (https=) | 2013-12-19 |
| JP5815542B2 JP5815542B2 (ja) | 2015-11-17 |
Family
ID=43503067
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012537052A Expired - Fee Related JP5815542B2 (ja) | 2009-10-29 | 2010-10-28 | Ｄｐｐ−１阻害剤として有用なアルキニル誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US8633322B2 (https=) |
| EP (1) | EP2493571B1 (https=) |
| JP (1) | JP5815542B2 (https=) |
| CN (1) | CN102596321B (https=) |
| AU (1) | AU2010319927B2 (https=) |
| ES (1) | ES2513291T3 (https=) |
| WO (1) | WO2011059731A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012119941A1 (en) | 2011-03-04 | 2012-09-13 | Prozymex A/S | Peptidyl nitrilcompounds as peptidase inhibitors |
| EP2825533B1 (en) | 2012-03-13 | 2016-10-19 | Basf Se | Fungicidal pyrimidine compounds |
| AR091858A1 (es) | 2012-07-25 | 2015-03-04 | Sova Pharmaceuticals Inc | INHIBIDORES DE CISTATIONIN-g-LIASA (CSE) |
| WO2015036059A1 (en) | 2013-09-16 | 2015-03-19 | Basf Se | Fungicidal pyrimidine compounds |
| CA2923101A1 (en) | 2013-09-16 | 2015-03-19 | Basf Se | Fungicidal pyrimidine compounds |
| CN115996923B (zh) | 2020-08-26 | 2025-07-18 | 海思科医药集团股份有限公司 | 一种作为二肽基肽酶1抑制剂的腈衍生物及其用途 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US548021A (en) * | 1895-10-15 | Wiiitfield potter toomee | ||
| US4847241A (en) * | 1985-08-14 | 1989-07-11 | G. D. Searle & Co. | Fluorenyl substituted tyrosyl dipeptide amides which are useful in treating pain |
| EP0574545B1 (en) | 1991-03-06 | 1994-11-30 | G.D. Searle & Co. | Phenyl amidines derivatives useful as platelet aggregation inhibitors |
| US5424334A (en) | 1991-12-19 | 1995-06-13 | G. D. Searle & Co. | Peptide mimetic compounds useful as platelet aggregation inhibitors |
| DE4321502A1 (de) | 1993-06-29 | 1995-01-12 | Bayer Ag | Alkinol-substituierte Peptide, Verfahren zu ihrer Herstellung und ihre Verwendung als antiretrovirale Mittel |
| AU6490396A (en) | 1995-07-14 | 1997-02-18 | Smithkline Beecham Corporation | Substituted-pent-4-ynoic acids |
| IL123164A (en) | 1995-08-30 | 2001-03-19 | Searle & Co | Meta-guanidine urea thiourea or azacyclic amino benzoic acid derivatives and pharmaceutical compositions containing them |
| JP2002145897A (ja) | 2000-11-10 | 2002-05-22 | Kyorin Pharmaceut Co Ltd | アミノ酸誘導体及びその製造法 |
| CN100522976C (zh) * | 2002-05-07 | 2009-08-05 | 神经研究公司 | 氮杂环乙炔基衍生物 |
| HK1079787A1 (zh) * | 2002-07-31 | 2006-04-13 | Ranbaxy Laboratories Limited | 用作毒蕈碱受体拮抗剂的3，6-二取代的氮杂双环[3．1．0]己烷衍生物 |
| WO2004071448A2 (en) * | 2003-02-12 | 2004-08-26 | Transtech Pharma Inc. | Substituted azole derivatives as inhibitors of protein tyrosine phosphatases |
| CA2514363A1 (en) * | 2003-02-12 | 2004-08-26 | Transtech Pharma, Inc. | Substituted azole derivatives as therapeutic agents |
| EP1633702B1 (en) * | 2003-05-30 | 2008-07-02 | Prozymex A/S | Protease inhibitors |
| US7638513B2 (en) * | 2004-06-02 | 2009-12-29 | Schering Corporation | Compounds for the treatment of inflammatory disorders |
| DE102005009784B4 (de) | 2005-03-03 | 2009-06-18 | Technische Universität Darmstadt | Peptid-Mimetika, Verfahren zur deren Herstellung, diese enthaltende pharmazeutische Zusammensetzung und deren Verwendung als Inhibitoren von Proteasomen und zur Induktion von Apoptose |
| AU2006230447A1 (en) * | 2005-03-30 | 2006-10-05 | Conforma Therapeutics Corporation | Alkynyl pyrrolopyrimidines and related analogs as HSP90-inhibitors |
| US7807699B2 (en) | 2006-03-21 | 2010-10-05 | Joyant Pharmaceuticals, Inc. | Dimeric pyrrolidine amide-containing small molecule apoptosis promoters |
| US7678894B2 (en) | 2007-05-18 | 2010-03-16 | Helicos Biosciences Corporation | Nucleotide analogs |
| US20090264431A1 (en) | 2007-08-20 | 2009-10-22 | Palovich Michael R | Novel cathepsin c inhibitors and their use |
| US7902181B2 (en) | 2007-12-12 | 2011-03-08 | Astrazeneca Ab | Compounds 010 |
-
2010
- 2010-10-28 CN CN201080049814.4A patent/CN102596321B/zh not_active Expired - Fee Related
- 2010-10-28 ES ES10774098.7T patent/ES2513291T3/es active Active
- 2010-10-28 JP JP2012537052A patent/JP5815542B2/ja not_active Expired - Fee Related
- 2010-10-28 US US12/914,244 patent/US8633322B2/en not_active Expired - Fee Related
- 2010-10-28 AU AU2010319927A patent/AU2010319927B2/en not_active Ceased
- 2010-10-28 WO PCT/US2010/054445 patent/WO2011059731A1/en not_active Ceased
- 2010-10-28 EP EP10774098.7A patent/EP2493571B1/en active Active
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