AU2010319927B2 - Alkynyl derivatives useful as DPP-1 inhibitors - Google Patents

Alkynyl derivatives useful as DPP-1 inhibitors Download PDF

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Publication number
AU2010319927B2
AU2010319927B2 AU2010319927A AU2010319927A AU2010319927B2 AU 2010319927 B2 AU2010319927 B2 AU 2010319927B2 AU 2010319927 A AU2010319927 A AU 2010319927A AU 2010319927 A AU2010319927 A AU 2010319927A AU 2010319927 B2 AU2010319927 B2 AU 2010319927B2
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Prior art keywords
phenyl
group
methyl
oxy
alkyl
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AU2010319927A
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AU2010319927A1 (en
Inventor
Shyamali Ghosh
Dennis J. Hlasta
Yifang Huang
Edward C. Lawson
Michael H. Parker
Allen B. Reitz
Carsten Shubert
Eric Strobel
Brett Tounge
Kimberly White
Michael P. Winters
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Janssen Pharmaceutica NV
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Janssen Pharmaceutica NV
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    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/16—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and unsaturated
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AU2010319927A 2009-10-29 2010-10-28 Alkynyl derivatives useful as DPP-1 inhibitors Ceased AU2010319927B2 (en)

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Application Number Priority Date Filing Date Title
US25617109P 2009-10-29 2009-10-29
US61/256,171 2009-10-29
PCT/US2010/054445 WO2011059731A1 (en) 2009-10-29 2010-10-28 Alkynyl derivatives useful as dpp-1 inhibitors

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AU2010319927A1 AU2010319927A1 (en) 2012-05-17
AU2010319927B2 true AU2010319927B2 (en) 2015-01-22

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US (1) US8633322B2 (https=)
EP (1) EP2493571B1 (https=)
JP (1) JP5815542B2 (https=)
CN (1) CN102596321B (https=)
AU (1) AU2010319927B2 (https=)
ES (1) ES2513291T3 (https=)
WO (1) WO2011059731A1 (https=)

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WO2012119941A1 (en) 2011-03-04 2012-09-13 Prozymex A/S Peptidyl nitrilcompounds as peptidase inhibitors
EP2825533B1 (en) 2012-03-13 2016-10-19 Basf Se Fungicidal pyrimidine compounds
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