JP2013509376A5 - - Google Patents
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- Publication number
- JP2013509376A5 JP2013509376A5 JP2012535821A JP2012535821A JP2013509376A5 JP 2013509376 A5 JP2013509376 A5 JP 2013509376A5 JP 2012535821 A JP2012535821 A JP 2012535821A JP 2012535821 A JP2012535821 A JP 2012535821A JP 2013509376 A5 JP2013509376 A5 JP 2013509376A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- substituted
- amino
- propanamide
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09174390.6 | 2009-10-28 | ||
| EP09174390A EP2316820A1 (en) | 2009-10-28 | 2009-10-28 | 2-aryl-propionamide derivatives useful as bradykinin receptor antagonists and pharmaceutical compositions containing them |
| PCT/EP2010/066324 WO2011051375A1 (en) | 2009-10-28 | 2010-10-28 | 2-aryl-propionamide derivatives useful as bradykinin receptor antagonists and pharmaceutical compositions containing them |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013509376A JP2013509376A (ja) | 2013-03-14 |
| JP2013509376A5 true JP2013509376A5 (https=) | 2013-12-19 |
Family
ID=41559661
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012535821A Pending JP2013509376A (ja) | 2009-10-28 | 2010-10-28 | ブラジキニン受容体アンタゴニストとして有用な２−アリール−プロピオンアミド誘導体およびそれらを含有する医薬組成物 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20120316169A1 (https=) |
| EP (2) | EP2316820A1 (https=) |
| JP (1) | JP2013509376A (https=) |
| KR (1) | KR20120084771A (https=) |
| CN (1) | CN102656140A (https=) |
| AU (1) | AU2010311466B2 (https=) |
| WO (1) | WO2011051375A1 (https=) |
| ZA (1) | ZA201203040B (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102701949A (zh) * | 2012-06-14 | 2012-10-03 | 山东新华制药股份有限公司 | 2-[4-(2-甲基-1-丙烯基)苯基]丙酸的制备方法 |
| CA2904052A1 (en) * | 2013-03-14 | 2014-10-02 | Shire Human Genetic Therapies, Inc. | Methods of treating b2-bradykinin receptor mediated angioedema |
| WO2019046668A1 (en) * | 2017-08-31 | 2019-03-07 | Kezar Life Sciences | AMIDE-SUBSTITUTED THIAZOLES AS INHIBITORS OF SECRETIC PROTEIN |
| CA3077659A1 (en) * | 2017-10-09 | 2019-04-18 | Ramot At Tel-Aviv University Ltd. | Modulators of potassium ion and trpv1 channels and uses thereof |
| EP4125848A1 (en) * | 2020-03-26 | 2023-02-08 | Dompe' Farmaceutici SpA | Cxcl8 inhibitors for use in the treatment of covid-19 |
| EP3884932A1 (en) * | 2020-03-26 | 2021-09-29 | Dompe' Farmaceutici S.P.A. | Cxcl8 inhibitors for use in the treatment of covid-19 |
| EP4008325A1 (en) * | 2020-12-02 | 2022-06-08 | Dompe' Farmaceutici S.P.A. | Cxcl8 inhibitors for use in the treatment of covid-19 |
| CN115403483B (zh) * | 2021-07-02 | 2024-01-26 | 河南省儿童医院郑州儿童医院 | 含二苯乙烯或二苯甲酮骨架的ca-4衍生物、药物组合物及其制备方法和应用 |
| EP4426288A4 (en) * | 2021-11-05 | 2025-12-31 | Georgiamune Inc | AKT3 MODULATORS |
| CN120093725B (zh) * | 2025-03-13 | 2025-12-16 | 江西中医药大学附属医院 | 金发藓酮e在制备治疗糖尿病视网膜病变药物中的应用 |
Family Cites Families (37)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE764238A (fr) * | 1971-03-17 | 1971-09-13 | Lilly Industries Ltd | Derives de phenylalkylamine |
| JPS6023105B2 (ja) * | 1982-10-22 | 1985-06-05 | 八洲化学工業株式会社 | α，α−ジメチルフエニル酢酸アニリド誘導体、その製造法及びそれを含有する除草剤 |
| TW253885B (https=) * | 1992-12-15 | 1995-08-11 | Ishihara Sangyo Kaisha | |
| JPH06234763A (ja) * | 1992-12-15 | 1994-08-23 | Ishihara Sangyo Kaisha Ltd | 環状アミド系化合物、それらの製造方法及びそれらを含有する除草性組成物 |
| ES2138206T3 (es) * | 1994-05-31 | 2000-01-01 | Teijin Ltd | Derivados de naftaleno. |
| FR2743562B1 (fr) | 1996-01-11 | 1998-04-03 | Sanofi Sa | Derives de n-(arylsulfonyl) aminoacides, leur preparation, les compositions pharmaceutiques en contenant |
| GB9702194D0 (en) * | 1997-02-04 | 1997-03-26 | Lilly Co Eli | Sulphonide derivatives |
| JP3752854B2 (ja) * | 1998-07-15 | 2006-03-08 | 宇部興産株式会社 | Ｎ−ベンジルカルバメイト化合物、その製法及び農園芸用の殺菌剤 |
| KR20010086461A (ko) * | 1998-12-24 | 2001-09-12 | 오흘러 로스 제이. | 인자 ｘａ 억제제로서의 치환된 (아미노이미노메틸 또는아미노메틸)벤조헤테로아릴 화합물 |
| GB9913079D0 (en) | 1999-06-04 | 1999-08-04 | Novartis Ag | Organic compounds |
| ATE250053T1 (de) | 1999-07-15 | 2003-10-15 | Pharmacopeia Inc | Bradikinin b1 rezeptor antagonisten |
| ITMI20010395A1 (it) * | 2001-02-27 | 2002-08-27 | Dompe Spa | Omega-amminoalchilammidi di acidi r-2-aril-propionici come inibitori della chemiotassi di cellule polimorfonucleate e mononucleate |
| CN1268610C (zh) | 2001-05-14 | 2006-08-09 | 诺瓦提斯公司 | 磺酰胺衍生物 |
| AU2002346048A1 (en) | 2001-06-07 | 2002-12-16 | Merck And Co., Inc. | Benzodiazepine bradykinin antagonists |
| DE10134721A1 (de) | 2001-07-17 | 2003-02-06 | Bayer Ag | Tetrahydrochinoxaline |
| AR036375A1 (es) * | 2001-08-30 | 2004-09-01 | Novartis Ag | Compuestos pirrolo [2,3-d] pirimidina -2- carbonitrilo, un proceso para su preparacion, una composicion farmaceutica y el uso de dichos compuestos para la preparacion de medicamentos |
| CA2483573A1 (en) | 2002-05-03 | 2003-11-13 | Elan Pharmaceuticals, Inc. | Sulfonylquinoxalone acetamide derivatives and related compounds as bradykinin antagonists |
| FR2840897B1 (fr) | 2002-06-14 | 2004-09-10 | Fournier Lab Sa | Nouveaux derives d'arylsulfonamides et leur utilisation en therapeutique |
| US20040034064A1 (en) | 2002-08-06 | 2004-02-19 | Kuduk Scott D. | 2-(biarylalkyl)amino-3-(alkanoylamino)pyridine derivatives |
| US20040029920A1 (en) | 2002-08-06 | 2004-02-12 | Kuduk Scott D. | 2-(biarylalkyl)amino-3-(heterocyclylcarbonylamino)-pyridine derivatives |
| US20040063761A1 (en) | 2002-08-06 | 2004-04-01 | Kuduk Scott D. | 2-(biarylalkyl)amino-3-(fluoroalkanoylamino)pyridine derivatives |
| US6908921B2 (en) | 2002-12-13 | 2005-06-21 | Merck & Co., Inc. | Quinoxalinone derivatives as bradykinin B1 antagonists |
| WO2004056744A1 (en) * | 2002-12-23 | 2004-07-08 | Janssen Pharmaceutica N.V. | Adamantyl acetamides as hydroxysteroid dehydrogenase inhibitors |
| KR100707123B1 (ko) * | 2003-07-02 | 2007-04-16 | 그뤼넨탈 게엠베하 | 바닐로이드 수용체의 길항제로서 강력한 진통효과를나타내는 4-(메틸설포닐아미노)페닐 동족체 및 이를함유하는 약학적 조성물 |
| EP1663960B1 (en) * | 2003-09-25 | 2011-08-24 | Dompe' S.P.A. | Amidines and derivatives thereof and pharmaceutical compositions containing them |
| US20050192314A1 (en) * | 2003-11-13 | 2005-09-01 | Ambit Biosciences Corporation | Urea derivatives as C-kit modulators |
| JP2005170939A (ja) * | 2003-11-20 | 2005-06-30 | Takeda Chem Ind Ltd | 糖尿病の予防・治療剤 |
| ATE444286T1 (de) * | 2004-03-23 | 2009-10-15 | Dompe Pha R Ma Spa Res & Mfg | 2-phenylpropionsäurederivate und diese enthaltende pharmazeutische zusammensetzung |
| US20080039609A1 (en) | 2004-07-09 | 2008-02-14 | Mitsui Chemicals, Inc. | Thermoplastic Resin |
| US7456194B2 (en) * | 2004-11-12 | 2008-11-25 | Bristol-Myers Squibb Company | Imidazo-fused oxazolo [4,5-b]pyridine and imidazo-fused thiazolo[4,5-b]pyridine based tricyclic compounds and pharmaceutical compositions comprising same |
| US20060111392A1 (en) * | 2004-11-23 | 2006-05-25 | Wood Michael R | Substituted biaryl-carboxylate derivatives |
| NZ555502A (en) * | 2004-12-15 | 2010-12-24 | Dompe Pha R Ma Spa Res & Mfg | 2-arylpropionic acid derivatives and pharmaceutical compositions containing them |
| TW200715993A (en) * | 2005-06-15 | 2007-05-01 | Senomyx Inc | Bis-aromatic amides and their uses as sweet flavor modifiers, tastants, and taste enhancers |
| PT2094638E (pt) * | 2006-12-19 | 2012-11-20 | Dompe Spa | Ácidos 2-aril-fluoropropanóicos e derivados e composições farmacêuticas que os contêm |
| WO2009001127A1 (en) * | 2007-06-26 | 2008-12-31 | Astrazeneca Ab | Cyanocyclopropylcarboxamides as cathepsin inhibitors |
| AU2008335709A1 (en) * | 2007-12-13 | 2009-06-18 | Amgen Inc. | Gamma secretase modulators |
| AU2010244685B2 (en) * | 2009-05-07 | 2016-02-18 | Medifron Dbt Inc. | Substituted phenylureas and phenylamides as vanilloid receptor ligands |
-
2009
- 2009-10-28 EP EP09174390A patent/EP2316820A1/en not_active Withdrawn
-
2010
- 2010-10-28 EP EP10775775A patent/EP2493846A1/en not_active Withdrawn
- 2010-10-28 WO PCT/EP2010/066324 patent/WO2011051375A1/en not_active Ceased
- 2010-10-28 AU AU2010311466A patent/AU2010311466B2/en not_active Expired - Fee Related
- 2010-10-28 JP JP2012535821A patent/JP2013509376A/ja active Pending
- 2010-10-28 US US13/504,535 patent/US20120316169A1/en not_active Abandoned
- 2010-10-28 CN CN201080053832XA patent/CN102656140A/zh active Pending
- 2010-10-28 KR KR1020127013707A patent/KR20120084771A/ko not_active Ceased
-
2012
- 2012-04-25 ZA ZA2012/03040A patent/ZA201203040B/en unknown
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