JP2013503161A5 - - Google Patents

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Publication number
JP2013503161A5
JP2013503161A5 JP2012526732A JP2012526732A JP2013503161A5 JP 2013503161 A5 JP2013503161 A5 JP 2013503161A5 JP 2012526732 A JP2012526732 A JP 2012526732A JP 2012526732 A JP2012526732 A JP 2012526732A JP 2013503161 A5 JP2013503161 A5 JP 2013503161A5
Authority
JP
Japan
Prior art keywords
pyridin
methyl
ethyl
tetrahydro
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2012526732A
Other languages
English (en)
Japanese (ja)
Other versions
JP2013503161A (ja
JP5746698B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2010/002360 external-priority patent/WO2011025541A1/en
Publication of JP2013503161A publication Critical patent/JP2013503161A/ja
Publication of JP2013503161A5 publication Critical patent/JP2013503161A5/ja
Application granted granted Critical
Publication of JP5746698B2 publication Critical patent/JP5746698B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2012526732A 2009-08-28 2010-08-27 カンナビノイド受容体モジュレーター Expired - Fee Related JP5746698B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US27550609P 2009-08-28 2009-08-28
US61/275,506 2009-08-28
US39658810P 2010-05-28 2010-05-28
US61/396,588 2010-05-28
US40014610P 2010-07-22 2010-07-22
US61/400,146 2010-07-22
PCT/US2010/002360 WO2011025541A1 (en) 2009-08-28 2010-08-27 Cannabinoid receptor modulators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015095753A Division JP2015145423A (ja) 2009-08-28 2015-05-08 カンナビノイド受容体モジュレーター

Publications (3)

Publication Number Publication Date
JP2013503161A JP2013503161A (ja) 2013-01-31
JP2013503161A5 true JP2013503161A5 (https=) 2013-10-10
JP5746698B2 JP5746698B2 (ja) 2015-07-08

Family

ID=43127457

Family Applications (5)

Application Number Title Priority Date Filing Date
JP2012526732A Expired - Fee Related JP5746698B2 (ja) 2009-08-28 2010-08-27 カンナビノイド受容体モジュレーター
JP2015095753A Withdrawn JP2015145423A (ja) 2009-08-28 2015-05-08 カンナビノイド受容体モジュレーター
JP2017207036A Withdrawn JP2018021074A (ja) 2009-08-28 2017-10-26 カンナビノイド受容体モジュレーター
JP2019221000A Withdrawn JP2020033387A (ja) 2009-08-28 2019-12-06 カンナビノイド受容体モジュレーター
JP2021173078A Withdrawn JP2022009408A (ja) 2009-08-28 2021-10-22 カンナビノイド受容体モジュレーター

Family Applications After (4)

Application Number Title Priority Date Filing Date
JP2015095753A Withdrawn JP2015145423A (ja) 2009-08-28 2015-05-08 カンナビノイド受容体モジュレーター
JP2017207036A Withdrawn JP2018021074A (ja) 2009-08-28 2017-10-26 カンナビノイド受容体モジュレーター
JP2019221000A Withdrawn JP2020033387A (ja) 2009-08-28 2019-12-06 カンナビノイド受容体モジュレーター
JP2021173078A Withdrawn JP2022009408A (ja) 2009-08-28 2021-10-22 カンナビノイド受容体モジュレーター

Country Status (19)

Country Link
US (6) US8778950B2 (https=)
EP (4) EP3363788A1 (https=)
JP (5) JP5746698B2 (https=)
KR (6) KR102682216B1 (https=)
CN (2) CN103539785B (https=)
AR (1) AR077991A1 (https=)
AU (1) AU2010286988B2 (https=)
BR (1) BR112012008159A2 (https=)
CA (1) CA2770866C (https=)
EA (1) EA023586B1 (https=)
HK (1) HK1259082A1 (https=)
IL (1) IL218130A (https=)
IN (1) IN2012DN02474A (https=)
MX (1) MX2012002499A (https=)
NZ (1) NZ598288A (https=)
SG (3) SG178907A1 (https=)
TW (1) TWI503316B (https=)
WO (1) WO2011025541A1 (https=)
ZA (1) ZA202205142B (https=)

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EP2803668A1 (en) 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles
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WO2015095953A1 (en) 2013-12-27 2015-07-02 The Centre For Drug Research And Development Sulfonamide-containing linkage systems for drug conjugates
ES2905569T3 (es) 2014-09-17 2022-04-11 Zymeworks Inc Compuestos citotóxicos y antimitóticos y métodos para utilizarlos
WO2016085941A1 (en) * 2014-11-25 2016-06-02 Arena Pharmaceuticals, Inc. Processes for the preparation of cannabinoid receptor modulators
US10172786B2 (en) 2014-12-16 2019-01-08 Axim Biotechnologies, Inc. Oral care composition comprising cannabinoids
AU2017249211A1 (en) * 2016-04-10 2018-11-22 Arena Pharmaceuticals, Inc. Methods of treatment with selective CB2 receptor agonists
CN109689045A (zh) 2016-05-04 2019-04-26 因美制药公司 大麻素的局部制剂在治疗大疱性表皮松解症和相关结缔组织病症中的用途
WO2018208847A1 (en) 2017-05-08 2018-11-15 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of pain from inflammatory bowel disease
US20200078358A1 (en) 2017-05-08 2020-03-12 Arena Pharmaceuticals, Inc. Compounds and Methods for Treatment of Visceral Pain
WO2019043635A1 (en) 2017-09-01 2019-03-07 Richter Gedeon Nyrt. COMPOUNDS INHIBITING THE ACTIVITY OF D-AMINO ACID OXIDASE
US12357604B2 (en) 2017-09-22 2025-07-15 Inmed Pharmaceuticals Inc. Topical formulations of cannabinoids and use thereof in the treatment of pain
EP3886845B1 (en) 2018-11-28 2024-09-04 Merck Sharp & Dohme LLC Novel substituted piperazine amide compounds as indoleamine 2, 3-dioxygenase (ido) inhibitors
WO2021047583A1 (zh) * 2019-09-12 2021-03-18 四川海思科制药有限公司 一种三环吡唑衍生物及其制备
WO2021047581A1 (zh) * 2019-09-12 2021-03-18 四川海思科制药有限公司 一种六氢化苯并吡唑衍生物及其制备
JP7620024B2 (ja) 2020-09-24 2025-01-22 富士フイルム株式会社 複合パターンの製造方法、樹脂組成物、積層体の製造方法、及び、半導体デバイスの製造方法
CN115536648B (zh) * 2021-06-29 2024-09-17 深圳开悦生命科技有限公司 一类抑制rna解旋酶dhx33的多环化合物及其应用
CN114736173B (zh) * 2022-05-24 2024-06-11 无锡捷化医药科技有限公司 一种3-（二氟甲基）氧杂环丁烷-3-胺盐酸盐的制备方法
WO2025090133A1 (en) 2023-10-23 2025-05-01 Inmed Pharmaceuticals Inc. Compositions and methods for use of cannabinol compounds in neuroprotection
WO2025090587A1 (en) 2023-10-23 2025-05-01 Inmed Pharmaceuticals Inc. Cannabinoids compounds and their use in the treatment of neuronal disorders

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EP2678330A1 (en) * 2011-02-25 2014-01-01 Arena Pharmaceuticals, Inc. Crystalline forms and processes for the preparation of condensed azacycles ( cannabinoid receptor modulators)

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