JP2013136631A5 - - Google Patents
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- Publication number
- JP2013136631A5 JP2013136631A5 JP2013055494A JP2013055494A JP2013136631A5 JP 2013136631 A5 JP2013136631 A5 JP 2013136631A5 JP 2013055494 A JP2013055494 A JP 2013055494A JP 2013055494 A JP2013055494 A JP 2013055494A JP 2013136631 A5 JP2013136631 A5 JP 2013136631A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- alkyl
- aryl
- compound
- deoxorapamycin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0601406.2 | 2006-01-24 | ||
| GBGB0601406.2A GB0601406D0 (en) | 2006-01-24 | 2006-01-24 | Organic Compounds |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008551707A Division JP5416412B2 (ja) | 2006-01-24 | 2007-01-22 | ラパマイシン誘導体の製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013136631A JP2013136631A (ja) | 2013-07-11 |
| JP2013136631A5 true JP2013136631A5 (enExample) | 2013-10-03 |
Family
ID=36060760
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008551707A Expired - Fee Related JP5416412B2 (ja) | 2006-01-24 | 2007-01-22 | ラパマイシン誘導体の製造方法 |
| JP2013055494A Pending JP2013136631A (ja) | 2006-01-24 | 2013-03-18 | ラパマイシン誘導体の製造方法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008551707A Expired - Fee Related JP5416412B2 (ja) | 2006-01-24 | 2007-01-22 | ラパマイシン誘導体の製造方法 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US8138344B2 (enExample) |
| EP (1) | EP1979359A1 (enExample) |
| JP (2) | JP5416412B2 (enExample) |
| KR (1) | KR101423343B1 (enExample) |
| CN (2) | CN104211716A (enExample) |
| AU (1) | AU2007209569B2 (enExample) |
| BR (1) | BRPI0707330A2 (enExample) |
| CA (1) | CA2637075A1 (enExample) |
| GB (1) | GB0601406D0 (enExample) |
| RU (1) | RU2448970C2 (enExample) |
| WO (1) | WO2007085400A1 (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0601406D0 (en) * | 2006-01-24 | 2006-03-08 | Novartis Ag | Organic Compounds |
| JP6378192B2 (ja) * | 2012-11-13 | 2018-08-22 | エルジー エレクトロニクス インコーポレイティド | データ送信方法及び装置、並びにデータ送信方法及び装置 |
| CN108864149B (zh) | 2013-03-15 | 2022-04-05 | 生物传感器国际集团有限公司 | 雷帕霉素衍生物的纯化 |
| EP3109250A1 (en) * | 2015-06-23 | 2016-12-28 | Synbias Pharma AG | Method for the synthesis of rapamycin derivatives |
| UY37900A (es) | 2017-09-26 | 2019-04-30 | Novartis Ag | Nuevos derivados de rapamicina |
| LT3898637T (lt) | 2018-12-18 | 2025-03-10 | Novartis Ag | Rapamicino dariniai |
| CA3127448C (en) | 2019-01-22 | 2024-06-04 | Aeovian Pharmaceuticals, Inc. | Mtorc modulators and uses thereof |
| KR20260115158A (ko) | 2019-03-26 | 2026-07-23 | 노파르티스 아게 | 이소티아졸리딘 1,1-디옥시드 및 1,4-부탄 술톤 함유 라파마이신 유도체 및 이의 용도 |
| CN115776907B (zh) | 2020-03-27 | 2025-02-25 | 艾奥维安制药公司 | Mtorc1调节剂及其用途 |
| WO2026080482A1 (en) * | 2024-10-07 | 2026-04-16 | Tornado Therapeutics, Inc. | Rapamycin derivatives and uses thereof |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5256790A (en) * | 1992-08-13 | 1993-10-26 | American Home Products Corporation | 27-hydroxyrapamycin and derivatives thereof |
| GB9221220D0 (en) * | 1992-10-09 | 1992-11-25 | Sandoz Ag | Organic componds |
| DE69624921T2 (de) * | 1995-06-09 | 2003-09-11 | Novartis Ag, Basel | Rapamycinderivate |
| IL150524A0 (en) * | 2000-01-07 | 2003-02-12 | Transform Pharmaceuticals Inc | High-throughput formation, identification, and analysis of diverse solid-forms |
| GB0601406D0 (en) * | 2006-01-24 | 2006-03-08 | Novartis Ag | Organic Compounds |
-
2006
- 2006-01-24 GB GBGB0601406.2A patent/GB0601406D0/en not_active Ceased
-
2007
- 2007-01-22 JP JP2008551707A patent/JP5416412B2/ja not_active Expired - Fee Related
- 2007-01-22 RU RU2008134424/04A patent/RU2448970C2/ru not_active IP Right Cessation
- 2007-01-22 CN CN201410391783.0A patent/CN104211716A/zh active Pending
- 2007-01-22 BR BRPI0707330-5A patent/BRPI0707330A2/pt not_active IP Right Cessation
- 2007-01-22 AU AU2007209569A patent/AU2007209569B2/en not_active Ceased
- 2007-01-22 CN CNA2007800034190A patent/CN101374847A/zh active Pending
- 2007-01-22 KR KR1020087018088A patent/KR101423343B1/ko not_active Expired - Fee Related
- 2007-01-22 US US12/160,110 patent/US8138344B2/en not_active Expired - Fee Related
- 2007-01-22 CA CA002637075A patent/CA2637075A1/en not_active Abandoned
- 2007-01-22 EP EP07702931A patent/EP1979359A1/en not_active Withdrawn
- 2007-01-22 WO PCT/EP2007/000514 patent/WO2007085400A1/en not_active Ceased
-
2013
- 2013-03-18 JP JP2013055494A patent/JP2013136631A/ja active Pending
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