JP2012526850A - サイクリン依存性キナーゼ阻害剤及びその用法 - Google Patents

サイクリン依存性キナーゼ阻害剤及びその用法 Download PDF

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JP2012526850A
JP2012526850A JP2012511031A JP2012511031A JP2012526850A JP 2012526850 A JP2012526850 A JP 2012526850A JP 2012511031 A JP2012511031 A JP 2012511031A JP 2012511031 A JP2012511031 A JP 2012511031A JP 2012526850 A JP2012526850 A JP 2012526850A
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cdk4
patient
cells
cyclin
dependent kinase
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JP2012526850A5 (https=
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イー シャープレス ノーマン
ジェイ ロバーツ パトリック
ウォン クウォ−キン
リュー ヤン
ジョンソン ソレン
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University of North Carolina at Chapel Hill
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University of North Carolina at Chapel Hill
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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JP2012511031A 2009-05-13 2010-05-13 サイクリン依存性キナーゼ阻害剤及びその用法 Pending JP2012526850A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17772409P 2009-05-13 2009-05-13
US61/177,724 2009-05-13
PCT/US2010/034816 WO2010132725A2 (en) 2009-05-13 2010-05-13 Cyclin dependent kinase inhibitors and methods of use

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JP2012526850A true JP2012526850A (ja) 2012-11-01
JP2012526850A5 JP2012526850A5 (https=) 2013-06-27

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US (2) US20120100100A1 (https=)
EP (4) EP3718560A3 (https=)
JP (1) JP2012526850A (https=)
CN (1) CN102458443A (https=)
AU (1) AU2010248886A1 (https=)
CA (1) CA2761896A1 (https=)
ES (1) ES2561216T3 (https=)
IL (1) IL216315A0 (https=)
WO (1) WO2010132725A2 (https=)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016513737A (ja) * 2013-03-15 2016-05-16 ジー１、セラピューティクス、インコーポレイテッドＧ１ Ｔｈｅｒａｐｅｕｔｉｃｓ， Ｉｎｃ． 化学療法の間の正常細胞の一時的な保護
JP2017524702A (ja) * 2014-07-26 2017-08-31 サンシャイン・レイク・ファーマ・カンパニー・リミテッドＳｕｎｓｈｉｎｅ Ｌａｋｅ Ｐｈａｒｍａ Ｃｏ．，Ｌｔｄ． ＣＤＫ阻害剤としての２−アミノ−ピリド［２，３−ｄ］ピリミジン−７（８Ｈ）−オン誘導体及びその使用
JP2021523202A (ja) * 2018-05-14 2021-09-02 ファイザー・インク 経口溶液製剤

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JP2012504646A (ja) * 2008-10-01 2012-02-23 ザ ユニバーシティ オブ ノース カロライナ アット チャペル ヒル 選択的サイクリン依存性キナーゼ４／６阻害剤を用いた化学療法化合物に対する造血系の防護
JP2012526850A (ja) 2009-05-13 2012-11-01 ザ ユニバーシティ オブ ノース カロライナ アット チャペル ヒル サイクリン依存性キナーゼ阻害剤及びその用法
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Citations (4)

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