JP2012512147A5 - - Google Patents

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Publication number
JP2012512147A5
JP2012512147A5 JP2011540134A JP2011540134A JP2012512147A5 JP 2012512147 A5 JP2012512147 A5 JP 2012512147A5 JP 2011540134 A JP2011540134 A JP 2011540134A JP 2011540134 A JP2011540134 A JP 2011540134A JP 2012512147 A5 JP2012512147 A5 JP 2012512147A5
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JP
Japan
Prior art keywords
preparation according
depot preparation
depot
polymer
microparticles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2011540134A
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English (en)
Japanese (ja)
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JP5721635B2 (ja
JP2012512147A (ja
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Publication date
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Priority claimed from PCT/EP2009/067049 external-priority patent/WO2010079047A2/en
Publication of JP2012512147A publication Critical patent/JP2012512147A/ja
Publication of JP2012512147A5 publication Critical patent/JP2012512147A5/ja
Application granted granted Critical
Publication of JP5721635B2 publication Critical patent/JP5721635B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2011540134A 2008-12-15 2009-12-14 一定して高い曝露レベルを有するオクトレオチドのデポー製剤 Active JP5721635B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP08171712 2008-12-15
EP08171712.6 2008-12-15
PCT/EP2009/067049 WO2010079047A2 (en) 2008-12-15 2009-12-14 Octreotide depot formulation with constantly high exposure levels

Publications (3)

Publication Number Publication Date
JP2012512147A JP2012512147A (ja) 2012-05-31
JP2012512147A5 true JP2012512147A5 (https=) 2013-02-07
JP5721635B2 JP5721635B2 (ja) 2015-05-20

Family

ID=40520410

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011540134A Active JP5721635B2 (ja) 2008-12-15 2009-12-14 一定して高い曝露レベルを有するオクトレオチドのデポー製剤

Country Status (25)

Country Link
US (10) US20100151033A1 (https=)
EP (1) EP2376070B1 (https=)
JP (1) JP5721635B2 (https=)
KR (1) KR101708517B1 (https=)
CN (3) CN105233251A (https=)
AR (1) AR074603A1 (https=)
AU (1) AU2009336718B9 (https=)
BR (1) BRPI0922607B1 (https=)
CA (1) CA2746968C (https=)
CL (1) CL2011001438A1 (https=)
CO (1) CO6382109A2 (https=)
EC (1) ECSP11011199A (https=)
ES (1) ES2602614T3 (https=)
IL (1) IL213034A (https=)
MA (1) MA32964B1 (https=)
MX (1) MX2011006335A (https=)
MY (1) MY159789A (https=)
NZ (1) NZ592998A (https=)
PE (1) PE20110876A1 (https=)
PL (1) PL2376070T3 (https=)
PT (1) PT2376070T (https=)
RU (1) RU2526822C2 (https=)
SG (1) SG171255A1 (https=)
TN (1) TN2011000261A1 (https=)
WO (1) WO2010079047A2 (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102176900B (zh) 2008-09-17 2017-09-26 克艾思马有限公司 药物组合物和相关的给药方法
EP2851085B1 (en) * 2012-05-14 2019-06-26 Teijin Limited Protein ccomposition sterilized by radiation
JP6494657B2 (ja) * 2014-03-31 2019-04-03 ファーマシェン エス.エー. 徐放特性を持つペプチド充填plgaミクロスフェアの調製
WO2016094662A1 (en) 2014-12-10 2016-06-16 Chiasma Inc. Oral octreotide administered in combination with other therapeutic agents
HUE071943T2 (hu) 2015-02-03 2025-10-28 Amryt Endo Inc Akromegália kezelése oktreotid orális alkalmazásával
CN105963258B (zh) 2016-04-26 2021-01-22 广州帝奇医药技术有限公司 一种缓释微粒的制备方法
KR102142026B1 (ko) * 2017-05-31 2020-08-06 주식회사 대웅제약 방출제어가 용이한 서방성 약물 미립자의 제조방법
EP3681469A1 (en) * 2017-09-15 2020-07-22 Oxular Limited Ophthalmic drug compositions
US12233177B2 (en) 2019-09-16 2025-02-25 Amgen Inc. Method for external sterilization of drug delivery device
US11141457B1 (en) 2020-12-28 2021-10-12 Amryt Endo, Inc. Oral octreotide therapy and contraceptive methods

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH30995A (en) * 1989-07-07 1997-12-23 Novartis Inc Sustained release formulations of water soluble peptides.
GB9513224D0 (en) * 1995-06-29 1995-09-06 Sandoz Ltd Organic compounds
ATE418323T1 (de) * 2002-11-06 2009-01-15 Alza Corp Depot-formulierungen mit verzögerter freisetzung
US20040097419A1 (en) * 2002-11-19 2004-05-20 Holger Petersen Organic compounds
MY158342A (en) * 2003-11-14 2016-09-30 Novartis Ag Pharmaceutical composition
GB0326602D0 (en) * 2003-11-14 2003-12-17 Novartis Ag Organic compounds
US7456254B2 (en) * 2004-04-15 2008-11-25 Alkermes, Inc. Polymer-based sustained release device
AU2005316545A1 (en) * 2004-12-15 2006-06-22 Qlt Usa, Inc. Sustained delivery formulations of octreotide compounds
CA2631811C (en) * 2005-12-22 2017-06-20 Novartis Ag Sustained release formulation comprising octreotide and two or more polylactide-co-glycolide polymers

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