JP2011530604A5 - - Google Patents

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Publication number
JP2011530604A5
JP2011530604A5 JP2011523042A JP2011523042A JP2011530604A5 JP 2011530604 A5 JP2011530604 A5 JP 2011530604A5 JP 2011523042 A JP2011523042 A JP 2011523042A JP 2011523042 A JP2011523042 A JP 2011523042A JP 2011530604 A5 JP2011530604 A5 JP 2011530604A5
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JP
Japan
Prior art keywords
linear
branched alkyl
disease
group
branched
Prior art date
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Application number
JP2011523042A
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English (en)
Japanese (ja)
Other versions
JP5529131B2 (ja
JP2011530604A (ja
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Publication date
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Priority claimed from PCT/US2009/052773 external-priority patent/WO2010019417A2/en
Publication of JP2011530604A publication Critical patent/JP2011530604A/ja
Publication of JP2011530604A5 publication Critical patent/JP2011530604A5/ja
Application granted granted Critical
Publication of JP5529131B2 publication Critical patent/JP5529131B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2011523042A 2008-08-13 2009-08-05 キマーゼ阻害薬 Active JP5529131B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8855108P 2008-08-13 2008-08-13
US61/088,551 2008-08-13
PCT/US2009/052773 WO2010019417A2 (en) 2008-08-13 2009-08-05 Chymase inhibitors

Publications (3)

Publication Number Publication Date
JP2011530604A JP2011530604A (ja) 2011-12-22
JP2011530604A5 true JP2011530604A5 (https=) 2012-09-20
JP5529131B2 JP5529131B2 (ja) 2014-06-25

Family

ID=41507988

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011523042A Active JP5529131B2 (ja) 2008-08-13 2009-08-05 キマーゼ阻害薬

Country Status (5)

Country Link
US (1) US8969348B2 (https=)
EP (1) EP2323991B1 (https=)
JP (1) JP5529131B2 (https=)
CA (1) CA2733128C (https=)
WO (1) WO2010019417A2 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2784180C (en) 2009-12-25 2014-03-11 Daiichi Sankyo Company, Limited Seven-membered ring compound and pharmaceutical use therefor

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3813384A (en) * 1972-01-17 1974-05-28 Asta Werke Ag Chem Fab Basically substituted benzyl phthalazone derivatives,acid salts thereof and process for the production thereof
GB8610018D0 (en) * 1986-04-24 1986-05-29 Fujisawa Pharmaceutical Co Phthalazine derivatives
DE3813531A1 (de) 1987-05-02 1988-11-10 Asta Pharma Ag Neue 2-aminoalkyl-4-benzyl-1-(2h)-phthalazinon-derivate
ZA882639B (en) * 1987-05-02 1988-09-30 Asta-Pharma Aktiengesellschaft New 2-aminoalkyl-4-benzyl-1(2h)-phthalazinone derivatives
US5380721A (en) * 1990-09-10 1995-01-10 Sterling Winthrop Inc. Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents
TW245719B (https=) 1990-09-10 1995-04-21 Sterling Winthrop Inc
DE4207234A1 (de) * 1992-03-07 1993-09-09 Asta Medica Ag Neue aminocarbonsaeure-derivate mit antiallergischer/antiasthmatischer wirkung und verfahren zu deren herstellung
CA2104060A1 (en) 1992-11-10 1994-05-11 Robert Ed Johnson Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents
ITMI981670A1 (it) * 1998-07-21 2000-01-21 Zambon Spa Derivati ftalazinici inibitori della fosfodiesterasi 4
NZ522882A (en) 2000-06-05 2004-07-30 Altana Pharma Bv Pyridazinone compounds effective as beta-2-adrenoreceptor agonists as well as PDE4-inhibitors
WO2008023357A1 (en) * 2006-08-22 2008-02-28 Technion Research And Development Foundation Ltd. Heterocyclic derivatives binding to the peripheral-type benzodiazepine receptor (pbr)
ATE459358T1 (de) * 2006-12-20 2010-03-15 Glaxo Group Ltd 4-benzyl-1(2h)-phthalazinone als h1-rezeptor- antagonisten

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