JP2019131544A5 - - Google Patents

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JP2019131544A5
JP2019131544A5 JP2019013745A JP2019013745A JP2019131544A5 JP 2019131544 A5 JP2019131544 A5 JP 2019131544A5 JP 2019013745 A JP2019013745 A JP 2019013745A JP 2019013745 A JP2019013745 A JP 2019013745A JP 2019131544 A5 JP2019131544 A5 JP 2019131544A5
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JP
Japan
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pharmaceutically acceptable
formula
acceptable salt
diabetes
compound represented
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JP2019013745A
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English (en)
Japanese (ja)
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JP2019131544A (ja
JP7241556B2 (ja
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Publication of JP2019131544A publication Critical patent/JP2019131544A/ja
Publication of JP2019131544A5 publication Critical patent/JP2019131544A5/ja
Priority to JP2023034806A priority Critical patent/JP2023071925A/ja
Application granted granted Critical
Publication of JP7241556B2 publication Critical patent/JP7241556B2/ja
Priority to JP2024094812A priority patent/JP2024116307A/ja
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JP2019013745A 2018-02-01 2019-01-30 含窒素複素環アミド化合物及びその医薬用途 Active JP7241556B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2023034806A JP2023071925A (ja) 2018-02-01 2023-03-07 含窒素複素環アミド化合物及びその医薬用途
JP2024094812A JP2024116307A (ja) 2018-02-01 2024-06-12 含窒素複素環アミド化合物及びその医薬用途

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2018016328 2018-02-01
JP2018016328 2018-02-01

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023034806A Division JP2023071925A (ja) 2018-02-01 2023-03-07 含窒素複素環アミド化合物及びその医薬用途

Publications (3)

Publication Number Publication Date
JP2019131544A JP2019131544A (ja) 2019-08-08
JP2019131544A5 true JP2019131544A5 (https=) 2022-02-03
JP7241556B2 JP7241556B2 (ja) 2023-03-17

Family

ID=67479787

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2019013745A Active JP7241556B2 (ja) 2018-02-01 2019-01-30 含窒素複素環アミド化合物及びその医薬用途
JP2023034806A Ceased JP2023071925A (ja) 2018-02-01 2023-03-07 含窒素複素環アミド化合物及びその医薬用途
JP2024094812A Pending JP2024116307A (ja) 2018-02-01 2024-06-12 含窒素複素環アミド化合物及びその医薬用途

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2023034806A Ceased JP2023071925A (ja) 2018-02-01 2023-03-07 含窒素複素環アミド化合物及びその医薬用途
JP2024094812A Pending JP2024116307A (ja) 2018-02-01 2024-06-12 含窒素複素環アミド化合物及びその医薬用途

Country Status (21)

Country Link
US (4) US10800784B2 (https=)
EP (1) EP3747888A4 (https=)
JP (3) JP7241556B2 (https=)
KR (1) KR102725118B1 (https=)
CN (1) CN111655692B (https=)
AR (1) AR114237A1 (https=)
AU (1) AU2019214048B2 (https=)
BR (1) BR112020014177A2 (https=)
CA (1) CA3090219A1 (https=)
CL (1) CL2020002003A1 (https=)
CO (1) CO2020009420A2 (https=)
IL (1) IL276386B2 (https=)
MX (1) MX2020008126A (https=)
MY (1) MY205011A (https=)
PE (1) PE20211273A1 (https=)
PH (1) PH12020500613A1 (https=)
SA (1) SA520412473B1 (https=)
SG (1) SG11202006916SA (https=)
TW (1) TWI803570B (https=)
WO (1) WO2019151274A1 (https=)
ZA (1) ZA202004548B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20220362215A1 (en) 2018-09-11 2022-11-17 Japan Tobacco Inc. Therapeutic or prophylactic agent for chronic kidney disease containing pyrazole-amide compound
CN110407744A (zh) * 2019-08-13 2019-11-05 上海毕得医药科技有限公司 一种1-(4-氨基吡啶-2-基)乙酮的合成方法
CN119841865A (zh) 2020-02-07 2025-04-18 加舒布鲁姆生物公司 杂环glp-1激动剂
PL4116301T3 (pl) * 2020-03-04 2026-02-16 Japan Tobacco Inc. Skondensowany związek tricykliczny i jego zastosowanie medyczne
EP4211139A4 (en) * 2020-09-10 2024-12-18 Gasherbrum Bio, Inc. HETEROCYCLIC GLP-1 AGONISTS
JP7599039B2 (ja) * 2021-03-23 2024-12-12 上海海雁医薬科技有限公司 複素環置換ケトン類誘導体、その組成物および医薬における使用
CN117897382A (zh) * 2021-09-01 2024-04-16 日本烟草产业株式会社 含氮三环化合物及其药物用途
AU2024222719A1 (en) 2023-02-16 2025-08-21 Gasherbrum Bio, Inc. Heterocyclic glp-1 agonists

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US7943617B2 (en) * 2006-11-27 2011-05-17 Bristol-Myers Squibb Company Heterobicyclic compounds useful as kinase inhibitors
WO2008132162A1 (en) 2007-04-26 2008-11-06 Boehringer Ingelheim International Gmbh 3- (sulphonylamino) -phenyl-2 -hydroxy-ethylamino derivatives useful as beta-agonists, processes for preparing them and their use as medicaments
MX2009013130A (es) * 2007-06-01 2010-01-15 Schering Corp Moduladores de gamma secretasa.
EP2090576A1 (en) * 2008-02-01 2009-08-19 Merz Pharma GmbH & Co.KGaA 6-halo-pyrazolo[1,5-a]pyridines, a process for their preparation and their use as metabotropic glutamate receptor (mGluR) modulators
AR074797A1 (es) * 2008-10-10 2011-02-16 Japan Tobacco Inc Compuesto de fluoreno , composiciones farmaceuticas , inhibidores de pdhk y pdhk2 , metodos de tratamiento , usos de los mismos y kit comercial
BR112013033098B8 (pt) 2011-06-27 2021-03-23 Alectos Therapeutics Inc inibidores de glicosidade seletivos e usos dos mesmos
AU2012339870B2 (en) * 2011-11-15 2017-06-29 Merck Sharp & Dohme Corp. Substituted cyclopropyl compounds useful as GPR119 agonists
PT2858986T (pt) * 2012-06-12 2019-11-29 Chong Kun Dang Pharmaceutical Corp Derivados de piperidina como agonistas de gpr119
CN103570725B (zh) 2012-08-01 2017-03-22 中国科学院上海药物研究所 哌嗪并三唑类化合物及其制备方法和用途
MY182884A (en) * 2013-03-15 2021-02-05 Japan Tobacco Inc Pyrazole-amide compound and medicinal uses therefor
JP2015028009A (ja) * 2013-07-01 2015-02-12 日本たばこ産業株式会社 ピラゾール−アルコール化合物およびその医薬用途
TW201536748A (zh) * 2013-07-01 2015-10-01 Japan Tobacco Inc 茀-醯胺化合物及其醫藥用途
GB201316823D0 (en) * 2013-09-23 2013-11-06 R & D Vernalis Ltd New Chemical Entities
SG11201604940VA (en) 2013-12-17 2016-07-28 Merck Patent Gmbh N1-(3,3,3-trifluoro-2-hydroxo-2-methylpropionyl)-piperidine derivatives as inhibitors of pyruvate dehydrogenase kinase
CA2994027C (en) 2015-07-31 2023-10-10 Merck Patent Gmbh Bicyclic heterocyclic derivatives
JP6923551B2 (ja) 2016-03-29 2021-08-18 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung ピルバートデヒドロゲナーゼキナーゼのインヒビターとしてのn1−(3,3,3−トリフルオロ−2−ヒドロキシ−2−メチルプロピオニル)−ピペリジン誘導体
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RU2019109039A (ru) 2016-10-28 2020-11-30 Х. Лундбекк А/С Комбинированные средства для лечения, предусматривающего введение имидазопиразинонов, предназначенные для лечения психических и/или когнитивных расстройств
PL4116301T3 (pl) * 2020-03-04 2026-02-16 Japan Tobacco Inc. Skondensowany związek tricykliczny i jego zastosowanie medyczne
CN117897382A (zh) * 2021-09-01 2024-04-16 日本烟草产业株式会社 含氮三环化合物及其药物用途

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