JP2011521940A5 - - Google Patents

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Publication number
JP2011521940A5
JP2011521940A5 JP2011511102A JP2011511102A JP2011521940A5 JP 2011521940 A5 JP2011521940 A5 JP 2011521940A5 JP 2011511102 A JP2011511102 A JP 2011511102A JP 2011511102 A JP2011511102 A JP 2011511102A JP 2011521940 A5 JP2011521940 A5 JP 2011521940A5
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JP
Japan
Prior art keywords
composition
group
cas
exendin
obesity
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2011511102A
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English (en)
Japanese (ja)
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JP2011521940A (ja
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Priority claimed from PCT/IB2009/005659 external-priority patent/WO2009144555A1/en
Publication of JP2011521940A publication Critical patent/JP2011521940A/ja
Publication of JP2011521940A5 publication Critical patent/JP2011521940A5/ja
Withdrawn legal-status Critical Current

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JP2011511102A 2008-05-28 2009-05-18 ピラゾロスピロケトンアセチルCoAカルボキシラーゼ阻害剤 Withdrawn JP2011521940A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US5665208P 2008-05-28 2008-05-28
US61/056,652 2008-05-28
US5868908P 2008-06-04 2008-06-04
US61/058,689 2008-06-04
US17111209P 2009-04-21 2009-04-21
US61/171,112 2009-04-21
PCT/IB2009/005659 WO2009144555A1 (en) 2008-05-28 2009-05-18 Pyrazolospiroketone acetyl-coa carboxylase inhibitors

Publications (2)

Publication Number Publication Date
JP2011521940A JP2011521940A (ja) 2011-07-28
JP2011521940A5 true JP2011521940A5 (cg-RX-API-DMAC7.html) 2012-07-05

Family

ID=40974463

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011511102A Withdrawn JP2011521940A (ja) 2008-05-28 2009-05-18 ピラゾロスピロケトンアセチルCoAカルボキシラーゼ阻害剤

Country Status (5)

Country Link
US (1) US20110009443A1 (cg-RX-API-DMAC7.html)
EP (1) EP2297164A1 (cg-RX-API-DMAC7.html)
JP (1) JP2011521940A (cg-RX-API-DMAC7.html)
CA (1) CA2724603A1 (cg-RX-API-DMAC7.html)
WO (1) WO2009144555A1 (cg-RX-API-DMAC7.html)

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BR112016004118A2 (pt) 2013-09-12 2017-10-17 Pfizer uso de inibidores da acetil-coa carboxilase para tratamento de acne vulgar
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TR201809388T4 (tr) 2014-03-17 2018-07-23 Pfizer Metabolik ve ilişkili hastalıkların tedavisinde kullanılmaya yönelik diasilgliserol asiltransferaz 2 inhibitörleri.
HUE044180T2 (hu) 2014-04-04 2019-10-28 Pfizer Biciklusos kondenzált heteroaril- vagy aril-vegyületek és ezek alkalmazása IRAK4 inhibitorokként
PE20170327A1 (es) 2014-04-10 2017-04-21 Pfizer 2-AMINO-6-METIL-4,4a,5,6-TETRAHIDROPIRANO[3,4d] [1,3] TIAZIN-8a(8H)-IL-1,3-TIAZOL-4-ILAMIDAS
EP3194367B1 (en) * 2014-09-17 2021-08-18 Boehringer Ingelheim International GmbH Tetrahydroisoquinoline derivatives and pharmaceutical compositions useful for the treatment of obesity and diabetes
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JP2017538769A (ja) 2014-12-22 2017-12-28 ファイザー・インク プロスタグランジンep3受容体の拮抗薬
BR112017022340A2 (pt) 2015-05-05 2018-07-10 Pfizer 2-tiopirimidinonas
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WO2016203335A1 (en) 2015-06-18 2016-12-22 Pfizer Inc. Novel pyrido[2,3-b]pyrazinones as bet-family bromodomain inhibitors
JP2018527337A (ja) 2015-08-13 2018-09-20 ファイザー・インク 二環式縮合ヘテロアリールまたはアリール化合物
JP6804524B2 (ja) 2015-08-27 2020-12-23 ファイザー・インク Irak4モジュレーターとしての二環式縮合ヘテロアリールまたはアリール化合物
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ATE552262T1 (de) * 2006-11-29 2012-04-15 Pfizer Prod Inc Spiroketone als inhibitoren von acetyl-coa- carboxylase

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