JP2011517455A - Ｃ（１０）エチルエステルおよびｃ（１０）シクロプロピルエステル置換タキサン - Google Patents

Ｃ（１０）エチルエステルおよびｃ（１０）シクロプロピルエステル置換タキサン Download PDF

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Publication number
JP2011517455A
JP2011517455A JP2011503034A JP2011503034A JP2011517455A JP 2011517455 A JP2011517455 A JP 2011517455A JP 2011503034 A JP2011503034 A JP 2011503034A JP 2011503034 A JP2011503034 A JP 2011503034A JP 2011517455 A JP2011517455 A JP 2011517455A
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pharmaceutical composition
taxane
cancer
tumor
compound
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Japanese (ja)
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JP2011517455A5 (cg-RX-API-DMAC7.html
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フォン・ブ
ロバート・エイ・ホルトン
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Florida State University Research Foundation Inc
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Florida State University Research Foundation Inc
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Publication of JP2011517455A publication Critical patent/JP2011517455A/ja
Publication of JP2011517455A5 publication Critical patent/JP2011517455A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
JP2011503034A 2008-03-31 2009-03-24 Ｃ（１０）エチルエステルおよびｃ（１０）シクロプロピルエステル置換タキサン Pending JP2011517455A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4101708P 2008-03-31 2008-03-31
US61/041,017 2008-03-31
PCT/US2009/038119 WO2009145981A1 (en) 2008-03-31 2009-03-24 C(10) ethyl ester and c(10) cyclopropyl ester substituted taxanes

Publications (2)

Publication Number Publication Date
JP2011517455A true JP2011517455A (ja) 2011-06-09
JP2011517455A5 JP2011517455A5 (cg-RX-API-DMAC7.html) 2012-05-17

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JP2011503034A Pending JP2011517455A (ja) 2008-03-31 2009-03-24 Ｃ（１０）エチルエステルおよびｃ（１０）シクロプロピルエステル置換タキサン

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US (1) US8242166B2 (cg-RX-API-DMAC7.html)
EP (1) EP2276755A4 (cg-RX-API-DMAC7.html)
JP (1) JP2011517455A (cg-RX-API-DMAC7.html)
CA (1) CA2718567A1 (cg-RX-API-DMAC7.html)
WO (1) WO2009145981A1 (cg-RX-API-DMAC7.html)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
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WO2009002425A2 (en) * 2007-06-22 2008-12-31 Scidose Llc Solubilized formulation of docetaxel without tween 80
JP2011514349A (ja) * 2008-03-07 2011-05-06 サイドース・エルエルシー フルベストラント配合物
US8541465B2 (en) * 2009-10-19 2013-09-24 Scidose, Llc Docetaxel formulations with lipoic acid and/or dihydrolipoic acid
US7772274B1 (en) 2009-10-19 2010-08-10 Scidose, Llc Docetaxel formulations with lipoic acid
US20110092579A1 (en) * 2009-10-19 2011-04-21 Scidose Llc Solubilized formulation of docetaxel
US8476310B2 (en) 2009-10-19 2013-07-02 Scidose Llc Docetaxel formulations with lipoic acid
US8912228B2 (en) 2009-10-19 2014-12-16 Scidose Llc Docetaxel formulations with lipoic acid
US11179468B2 (en) 2012-04-09 2021-11-23 Eagle Pharmaceuticals, Inc. Fulvestrant formulations

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JP5571380B2 (ja) * 2006-07-24 2014-08-13 ルミナス バイオサイエンシズ，インコーポレイテッド オストワルド熟成を減少させた水不溶性の医薬品物質の固体ナノ粒子処方物

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JPH07503477A (ja) * 1992-02-07 1995-04-13 ローン−プーラン・ロレ・ソシエテ・アノニム バッカチン３および１０‐デアセチルバッカチン３の新規誘導体，それらの製造およびそれらを含有する医薬組成物
WO1999014209A1 (en) * 1997-09-17 1999-03-25 Kabushiki Kaisha Yakult Honsha New taxane derivatives
WO1999032473A1 (en) * 1997-12-19 1999-07-01 Kabushiki Kaisha Yakult Honsha Taxane derivatives
JP2003521545A (ja) * 2000-02-02 2003-07-15 フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド 改良された溶解性を有するタキサン製剤
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JPN6013049957; ＳＡＭＰＡＴＨ，Ｄ．　ｅｔ　ａｌ: Ｃｌｉｎｉｃａｌ　Ｃａｎｃｅｒ　Ｒｅｓｅａｒｃｈ Ｖｏｌ．１２，　Ｎｏ．１１, 2006, ｐ．３４５９-３４６９ *

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EP2276755A1 (en) 2011-01-26
US20090318543A1 (en) 2009-12-24
US8242166B2 (en) 2012-08-14
EP2276755A4 (en) 2011-05-04
WO2009145981A1 (en) 2009-12-03
CA2718567A1 (en) 2009-12-03

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