JP2011516417A - Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 - Google Patents
Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 Download PDFInfo
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- JP2011516417A JP2011516417A JP2011501153A JP2011501153A JP2011516417A JP 2011516417 A JP2011516417 A JP 2011516417A JP 2011501153 A JP2011501153 A JP 2011501153A JP 2011501153 A JP2011501153 A JP 2011501153A JP 2011516417 A JP2011516417 A JP 2011516417A
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| PCT/EP2009/002241 WO2009118187A1 (en) | 2008-03-27 | 2009-03-26 | Methods for treating disorders using nmda nr2b-subtype selective antagonist |
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| JP2014020051A Division JP2014098018A (ja) | 2008-03-27 | 2014-02-05 | Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 |
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| JP2011516417A true JP2011516417A (ja) | 2011-05-26 |
| JP2011516417A5 JP2011516417A5 (https=) | 2012-01-05 |
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| JP2014020051A Pending JP2014098018A (ja) | 2008-03-27 | 2014-02-05 | Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 |
| JP2015236571A Pending JP2016094430A (ja) | 2008-03-27 | 2015-12-03 | Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 |
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| JP2015236571A Pending JP2016094430A (ja) | 2008-03-27 | 2015-12-03 | Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 |
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| US (1) | US20110053951A1 (https=) |
| EP (1) | EP2254580A1 (https=) |
| JP (3) | JP2011516417A (https=) |
| KR (1) | KR20100135847A (https=) |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017525700A (ja) * | 2014-08-15 | 2017-09-07 | ヤンセン ファーマシューティカルズ,インコーポレーテッド | ピラゾール類 |
| JP2019504854A (ja) * | 2016-02-10 | 2019-02-21 | ヤンセン ファーマシューティカ エヌ.ベー. | Nr2b選択的nmda調節因子としての置換1,2,3−トリアゾール |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
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| AU2013251079B2 (en) | 2012-04-20 | 2017-03-23 | Ucb Pharma S.A. | Methods for treating Parkinson's disease |
| WO2015175806A1 (en) * | 2014-05-16 | 2015-11-19 | The Trustees Of The University Of Pennsylvania | Applications of automatic anatomy recognition in medical tomographic imagery based on fuzzy anatomy models |
| WO2016025917A1 (en) * | 2014-08-15 | 2016-02-18 | Janssen Pharmaceuticals, Inc. | Triazoles as nr2b receptor inhibitors |
| BR112017025023B1 (pt) | 2015-06-01 | 2024-01-30 | Rugen Holdings (Cayman) Limited | Compostos heterocíclicos de carbamato de 3,3-difluoropiperidina, seu uso como antagonistas do receptor nmda nr2b e composição farmacêutica que os compreende |
| HRP20200410T1 (hr) | 2015-07-09 | 2020-08-21 | Janssen Pharmaceutica Nv | Supstituirani 4-azaindoli i njihova upotreba kao modulatora glun2b receptora |
| US10487055B2 (en) | 2016-06-01 | 2019-11-26 | Rhode Island Board Of Education | Diindole compounds useful in treatment of nervous system disorders |
| TW201819376A (zh) | 2016-10-06 | 2018-06-01 | 比利時商健生藥品公司 | 經取代之1H-咪唑並[4,5-b]吡啶-2(3H)-酮及其作為GLUN2B受體調節劑之用途 |
| WO2018098128A1 (en) | 2016-11-22 | 2018-05-31 | Rugen Holdings (Cayman) Limited | Treatment of autism spectrum disorders, obsessive-compulsive disorder and anxiety disorders |
| US10732235B2 (en) * | 2018-03-29 | 2020-08-04 | Siemens Healthcare Gmbh | Magnetic resonance method and apparatus using atlas-based masking for quantitative susceptibility mapping |
| WO2019193516A2 (en) | 2018-04-04 | 2019-10-10 | Janssen Pharmaceutica Nv | Substituted pyridine and pyrimidines and their use as glun2b receptor modulators |
| KR20220024403A (ko) | 2019-06-14 | 2022-03-03 | 얀센 파마슈티카 엔.브이. | 치환된 피라졸로-피라진 및 이들의 glun2b 수용체 조절제로서의 용도 |
| CN113950357A (zh) | 2019-06-14 | 2022-01-18 | 詹森药业有限公司 | 吡嗪氨基甲酸酯及其作为GluN2B受体调节剂的用途 |
| SG11202112405VA (en) | 2019-06-14 | 2021-12-30 | Janssen Pharmaceutica Nv | Substituted heteroaromatic pyrazolo-pyridines and their use as glun2b receptor modulators |
| CN113993868A (zh) | 2019-06-14 | 2022-01-28 | 詹森药业有限公司 | 取代的吡唑并吡啶酰胺以及它们作为glun2b受体调节剂的用途 |
| MX2021015508A (es) | 2019-06-14 | 2022-01-31 | Janssen Pharmaceutica Nv | Carbamatos de piridina y su uso como moduladores del receptor glun2b. |
| AU2020293642A1 (en) | 2019-06-14 | 2022-01-20 | Janssen Pharmaceutica Nv | Substituted pyrazolo[4,3-b]pyridines and their use as GluN2B receptor modulators |
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| PT885004E (pt) * | 1996-03-08 | 2002-08-30 | Hoffmann La Roche | Utilizacao de derivados de 4-fenil-3,6-di-hidro-2h-piridilo como bloqueadores dos subtipos dos receptores nmda |
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| EP1070708B1 (en) * | 1999-07-21 | 2004-01-14 | F. Hoffmann-La Roche Ag | Triazole derivatives |
| ES2225553T3 (es) * | 2000-04-20 | 2005-03-16 | F. Hoffmann-La Roche Ag | Derivados de pirrolidina y piperidina y su empleo para el tratamiento de trastornos neurodegenerativos. |
| US6432985B2 (en) * | 2000-04-25 | 2002-08-13 | Hoffmann-La Roche Inc. | Neuroprotective substituted piperidine compounds with activity as NMDA NR2B subtype selective antagonists |
| AU2001296994A1 (en) * | 2000-10-06 | 2002-04-15 | Regents Of The University Of California | Nmda receptor channel blocker with neuroprotective activity |
| CA2617104A1 (en) * | 2005-07-29 | 2007-02-08 | Regents Of The University Of Minnesota | Amyloid beta receptor and uses thereof |
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| JP2005532326A (ja) * | 2002-05-16 | 2005-10-27 | エフ.ホフマン−ラ ロシュ アーゲー | Nmdaレセプターブロッカーとしての(イミダゾール−1−イル−メチル)−ピリダジン |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017525700A (ja) * | 2014-08-15 | 2017-09-07 | ヤンセン ファーマシューティカルズ,インコーポレーテッド | ピラゾール類 |
| JP2019504854A (ja) * | 2016-02-10 | 2019-02-21 | ヤンセン ファーマシューティカ エヌ.ベー. | Nr2b選択的nmda調節因子としての置換1,2,3−トリアゾール |
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| KR20100135847A (ko) | 2010-12-27 |
| IL207835A0 (en) | 2010-12-30 |
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| CA2719749A1 (en) | 2009-10-01 |
| RU2010143864A (ru) | 2012-05-10 |
| BRPI0909378A2 (pt) | 2015-10-06 |
| NZ588698A (en) | 2012-06-29 |
| AU2009228660A1 (en) | 2009-10-01 |
| MX2010009649A (es) | 2010-12-17 |
| AU2009228660B2 (en) | 2012-11-29 |
| ZA201006587B (en) | 2012-02-29 |
| US20110053951A1 (en) | 2011-03-03 |
| JP2014098018A (ja) | 2014-05-29 |
| RU2499598C2 (ru) | 2013-11-27 |
| CN101977606A (zh) | 2011-02-16 |
| EP2254580A1 (en) | 2010-12-01 |
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