JP2011516417A5 - - Google Patents

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Publication number
JP2011516417A5
JP2011516417A5 JP2011501153A JP2011501153A JP2011516417A5 JP 2011516417 A5 JP2011516417 A5 JP 2011516417A5 JP 2011501153 A JP2011501153 A JP 2011501153A JP 2011501153 A JP2011501153 A JP 2011501153A JP 2011516417 A5 JP2011516417 A5 JP 2011516417A5
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JP
Japan
Prior art keywords
pain
disease
pharmaceutical composition
composition according
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011501153A
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English (en)
Japanese (ja)
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JP2011516417A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2009/002241 external-priority patent/WO2009118187A1/en
Publication of JP2011516417A publication Critical patent/JP2011516417A/ja
Publication of JP2011516417A5 publication Critical patent/JP2011516417A5/ja
Pending legal-status Critical Current

Links

JP2011501153A 2008-03-27 2009-03-26 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法 Pending JP2011516417A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4008708P 2008-03-27 2008-03-27
US61/040,087 2008-03-27
PCT/EP2009/002241 WO2009118187A1 (en) 2008-03-27 2009-03-26 Methods for treating disorders using nmda nr2b-subtype selective antagonist

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014020051A Division JP2014098018A (ja) 2008-03-27 2014-02-05 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法

Publications (2)

Publication Number Publication Date
JP2011516417A JP2011516417A (ja) 2011-05-26
JP2011516417A5 true JP2011516417A5 (https=) 2012-01-05

Family

ID=40910288

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011501153A Pending JP2011516417A (ja) 2008-03-27 2009-03-26 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法
JP2014020051A Pending JP2014098018A (ja) 2008-03-27 2014-02-05 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法
JP2015236571A Pending JP2016094430A (ja) 2008-03-27 2015-12-03 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2014020051A Pending JP2014098018A (ja) 2008-03-27 2014-02-05 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法
JP2015236571A Pending JP2016094430A (ja) 2008-03-27 2015-12-03 Nmdanr2b−サブタイプ選択的アンタゴニストを使用する障害の処置方法

Country Status (14)

Country Link
US (1) US20110053951A1 (https=)
EP (1) EP2254580A1 (https=)
JP (3) JP2011516417A (https=)
KR (1) KR20100135847A (https=)
CN (1) CN101977606A (https=)
AU (1) AU2009228660B2 (https=)
BR (1) BRPI0909378A2 (https=)
CA (1) CA2719749A1 (https=)
IL (1) IL207835A0 (https=)
MX (1) MX2010009649A (https=)
NZ (1) NZ588698A (https=)
RU (1) RU2499598C2 (https=)
WO (1) WO2009118187A1 (https=)
ZA (1) ZA201006587B (https=)

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AU2013251079B2 (en) 2012-04-20 2017-03-23 Ucb Pharma S.A. Methods for treating Parkinson's disease
WO2015175806A1 (en) * 2014-05-16 2015-11-19 The Trustees Of The University Of Pennsylvania Applications of automatic anatomy recognition in medical tomographic imagery based on fuzzy anatomy models
ES2791252T3 (es) * 2014-08-15 2020-11-03 Janssen Pharmaceuticals Inc Pirazoles
WO2016025917A1 (en) * 2014-08-15 2016-02-18 Janssen Pharmaceuticals, Inc. Triazoles as nr2b receptor inhibitors
BR112017025023B1 (pt) 2015-06-01 2024-01-30 Rugen Holdings (Cayman) Limited Compostos heterocíclicos de carbamato de 3,3-difluoropiperidina, seu uso como antagonistas do receptor nmda nr2b e composição farmacêutica que os compreende
HRP20200410T1 (hr) 2015-07-09 2020-08-21 Janssen Pharmaceutica Nv Supstituirani 4-azaindoli i njihova upotreba kao modulatora glun2b receptora
BR112018016329A2 (pt) 2016-02-10 2018-12-18 Janssen Pharmaceutica Nv 1,2,3-triazóis substituídos como moduladores de nmda seletivos para nr2b
US10487055B2 (en) 2016-06-01 2019-11-26 Rhode Island Board Of Education Diindole compounds useful in treatment of nervous system disorders
TW201819376A (zh) 2016-10-06 2018-06-01 比利時商健生藥品公司 經取代之1H-咪唑並[4,5-b]吡啶-2(3H)-酮及其作為GLUN2B受體調節劑之用途
WO2018098128A1 (en) 2016-11-22 2018-05-31 Rugen Holdings (Cayman) Limited Treatment of autism spectrum disorders, obsessive-compulsive disorder and anxiety disorders
US10732235B2 (en) * 2018-03-29 2020-08-04 Siemens Healthcare Gmbh Magnetic resonance method and apparatus using atlas-based masking for quantitative susceptibility mapping
WO2019193516A2 (en) 2018-04-04 2019-10-10 Janssen Pharmaceutica Nv Substituted pyridine and pyrimidines and their use as glun2b receptor modulators
KR20220024403A (ko) 2019-06-14 2022-03-03 얀센 파마슈티카 엔.브이. 치환된 피라졸로-피라진 및 이들의 glun2b 수용체 조절제로서의 용도
CN113950357A (zh) 2019-06-14 2022-01-18 詹森药业有限公司 吡嗪氨基甲酸酯及其作为GluN2B受体调节剂的用途
SG11202112405VA (en) 2019-06-14 2021-12-30 Janssen Pharmaceutica Nv Substituted heteroaromatic pyrazolo-pyridines and their use as glun2b receptor modulators
CN113993868A (zh) 2019-06-14 2022-01-28 詹森药业有限公司 取代的吡唑并吡啶酰胺以及它们作为glun2b受体调节剂的用途
MX2021015508A (es) 2019-06-14 2022-01-31 Janssen Pharmaceutica Nv Carbamatos de piridina y su uso como moduladores del receptor glun2b.
AU2020293642A1 (en) 2019-06-14 2022-01-20 Janssen Pharmaceutica Nv Substituted pyrazolo[4,3-b]pyridines and their use as GluN2B receptor modulators
JP7667097B2 (ja) 2019-06-14 2025-04-22 ヤンセン ファーマシューティカ エヌ.ベー. 置換ピラゾロ-ピリジンアミド及びglun2b受容体調節因子としてのその使用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT885004E (pt) * 1996-03-08 2002-08-30 Hoffmann La Roche Utilizacao de derivados de 4-fenil-3,6-di-hidro-2h-piridilo como bloqueadores dos subtipos dos receptores nmda
US5985936A (en) * 1997-12-18 1999-11-16 Forbes Medi-Tech, Inc. Method of preventing and delaying onset of Alzheimer's disease and composition therefor
US6015824A (en) * 1998-02-10 2000-01-18 Hoffmann-La Roche Ag Pyrrolidine and piperidine derivatives and treatment of neurodegenerative disorders
TWI254043B (en) * 1999-06-08 2006-05-01 Hoffmann La Roche Ethanesulfonyl-piperidine derivatives having good affinity to N-methyl-D-aspartate (NMDA) receptor
EP1070708B1 (en) * 1999-07-21 2004-01-14 F. Hoffmann-La Roche Ag Triazole derivatives
ES2225553T3 (es) * 2000-04-20 2005-03-16 F. Hoffmann-La Roche Ag Derivados de pirrolidina y piperidina y su empleo para el tratamiento de trastornos neurodegenerativos.
US6432985B2 (en) * 2000-04-25 2002-08-13 Hoffmann-La Roche Inc. Neuroprotective substituted piperidine compounds with activity as NMDA NR2B subtype selective antagonists
AU2001296994A1 (en) * 2000-10-06 2002-04-15 Regents Of The University Of California Nmda receptor channel blocker with neuroprotective activity
US7005432B2 (en) * 2002-05-16 2006-02-28 Hoffman-La Roche Inc. Substituted imidazol-pyridazine derivatives
CA2617104A1 (en) * 2005-07-29 2007-02-08 Regents Of The University Of Minnesota Amyloid beta receptor and uses thereof

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