JP2011510928A5 - - Google Patents
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- Publication number
- JP2011510928A5 JP2011510928A5 JP2010544413A JP2010544413A JP2011510928A5 JP 2011510928 A5 JP2011510928 A5 JP 2011510928A5 JP 2010544413 A JP2010544413 A JP 2010544413A JP 2010544413 A JP2010544413 A JP 2010544413A JP 2011510928 A5 JP2011510928 A5 JP 2011510928A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- independently
- haloalkyl
- alkoxy
- cyano
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 125000000217 alkyl group Chemical group 0.000 claims 57
- 125000003545 alkoxy group Chemical group 0.000 claims 33
- -1 cyano, hydroxy Chemical group 0.000 claims 33
- 125000001188 haloalkyl group Chemical group 0.000 claims 29
- 229910052736 halogen Inorganic materials 0.000 claims 23
- 150000002367 halogens Chemical class 0.000 claims 23
- 125000004183 alkoxy alkyl group Chemical group 0.000 claims 19
- 229910052799 carbon Inorganic materials 0.000 claims 19
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims 17
- 125000004438 haloalkoxy group Chemical group 0.000 claims 17
- 125000004448 alkyl carbonyl group Chemical group 0.000 claims 16
- 125000004432 carbon atoms Chemical group C* 0.000 claims 16
- 125000003342 alkenyl group Chemical group 0.000 claims 15
- 125000000262 haloalkenyl group Chemical group 0.000 claims 15
- 125000001424 substituent group Chemical group 0.000 claims 15
- 125000000753 cycloalkyl group Chemical group 0.000 claims 14
- 125000000232 haloalkynyl group Chemical group 0.000 claims 14
- 125000003282 alkyl amino group Chemical group 0.000 claims 13
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 claims 13
- 125000004414 alkyl thio group Chemical group 0.000 claims 13
- 125000000304 alkynyl group Chemical group 0.000 claims 13
- 125000004093 cyano group Chemical group *C#N 0.000 claims 13
- 125000005347 halocycloalkyl group Chemical group 0.000 claims 12
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 12
- 125000006350 alkyl thio alkyl group Chemical group 0.000 claims 11
- 125000004663 dialkyl amino group Chemical group 0.000 claims 11
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims 10
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 claims 10
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims 10
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 claims 10
- 229910052739 hydrogen Inorganic materials 0.000 claims 10
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 10
- 125000004665 trialkylsilyl group Chemical group 0.000 claims 10
- 125000005119 alkyl cycloalkyl group Chemical group 0.000 claims 9
- 125000000278 alkyl amino alkyl group Chemical group 0.000 claims 8
- 125000005120 alkyl cycloalkyl alkyl group Chemical group 0.000 claims 8
- 125000004687 alkyl sulfinyl alkyl group Chemical group 0.000 claims 8
- 125000004688 alkyl sulfonyl alkyl group Chemical group 0.000 claims 8
- 150000001875 compounds Chemical class 0.000 claims 8
- 125000004994 halo alkoxy alkyl group Chemical group 0.000 claims 8
- 125000005203 haloalkylcarbonyloxy group Chemical group 0.000 claims 8
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 claims 8
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 7
- 125000004995 haloalkylthio group Chemical group 0.000 claims 7
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 7
- 150000002829 nitrogen Chemical group 0.000 claims 7
- 229910052760 oxygen Inorganic materials 0.000 claims 7
- 125000002813 thiocarbonyl group Chemical group *C(*)=S 0.000 claims 7
- 125000005078 alkoxycarbonylalkyl group Chemical group 0.000 claims 6
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 claims 6
- 125000004390 alkyl sulfonyl group Chemical group 0.000 claims 6
- 125000004985 dialkyl amino alkyl group Chemical group 0.000 claims 6
- 125000001624 naphthyl group Chemical group 0.000 claims 6
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims 6
- 125000005083 alkoxyalkoxy group Chemical group 0.000 claims 5
- 125000005081 alkoxyalkoxyalkyl group Chemical group 0.000 claims 5
- 125000004122 cyclic group Chemical group 0.000 claims 5
- 125000000000 cycloalkoxy group Chemical group 0.000 claims 5
- 125000004858 cycloalkoxyalkyl group Chemical group 0.000 claims 5
- 125000006310 cycloalkyl amino group Chemical group 0.000 claims 5
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims 4
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 4
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 4
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 4
- 125000005130 alkyl carbonyl thio group Chemical group 0.000 claims 4
- 125000004644 alkyl sulfinyl group Chemical group 0.000 claims 4
- OKTJSMMVPCPJKN-UHFFFAOYSA-N carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 4
- 125000005112 cycloalkylalkoxy group Chemical group 0.000 claims 4
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 claims 4
- 125000004992 haloalkylamino group Chemical group 0.000 claims 4
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 claims 4
- 125000004461 halocycloalkylalkyl group Chemical group 0.000 claims 4
- 229910052717 sulfur Inorganic materials 0.000 claims 4
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims 3
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 3
- 125000003302 alkenyloxy group Chemical group 0.000 claims 3
- 125000004656 alkyl sulfonylamino group Chemical group 0.000 claims 3
- 125000005133 alkynyloxy group Chemical group 0.000 claims 3
- 125000003118 aryl group Chemical group 0.000 claims 3
- 125000002619 bicyclic group Chemical group 0.000 claims 3
- 125000006254 cycloalkyl carbonyl group Chemical group 0.000 claims 3
- 125000006448 cycloalkyl cycloalkyl group Chemical group 0.000 claims 3
- 125000005167 cycloalkylaminocarbonyl group Chemical group 0.000 claims 3
- 125000005201 cycloalkylcarbonyloxy group Chemical group 0.000 claims 3
- 125000005366 cycloalkylthio group Chemical group 0.000 claims 3
- 125000005291 haloalkenyloxy group Chemical group 0.000 claims 3
- 125000004664 haloalkylsulfonylamino group Chemical group 0.000 claims 3
- 125000005292 haloalkynyloxy group Chemical group 0.000 claims 3
- 125000006769 halocycloalkoxy group Chemical group 0.000 claims 3
- 125000005842 heteroatoms Chemical group 0.000 claims 3
- 125000000623 heterocyclic group Chemical group 0.000 claims 3
- 125000002768 hydroxyalkyl group Chemical group 0.000 claims 3
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims 3
- 125000002757 morpholinyl group Chemical group 0.000 claims 3
- 125000003386 piperidinyl group Chemical group 0.000 claims 3
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 3
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims 2
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims 2
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims 2
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims 2
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 2
- 125000006771 (C1-C6) haloalkylthio group Chemical group 0.000 claims 2
- 125000006766 (C2-C6) alkynyloxy group Chemical group 0.000 claims 2
- 125000006765 (C2-C6) haloalkenyloxy group Chemical group 0.000 claims 2
- 125000002853 C1-C4 hydroxyalkyl group Chemical group 0.000 claims 2
- 125000003320 C2-C6 alkenyloxy group Chemical group 0.000 claims 2
- 125000004648 C2-C8 alkenyl group Chemical group 0.000 claims 2
- 125000004649 C2-C8 alkynyl group Chemical group 0.000 claims 2
- 125000006615 aromatic heterocyclic group Chemical group 0.000 claims 2
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims 2
- 125000000392 cycloalkenyl group Chemical group 0.000 claims 2
- 125000005144 cycloalkylsulfonyl group Chemical group 0.000 claims 2
- 125000005221 halo alkyl carbonyl amino group Chemical group 0.000 claims 2
- 125000001160 methoxycarbonyl group Chemical group [H]C([H])([H])OC(*)=O 0.000 claims 2
- 229910052757 nitrogen Inorganic materials 0.000 claims 2
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 2
- 125000000719 pyrrolidinyl group Chemical group 0.000 claims 2
- 125000006729 (C2-C5) alkenyl group Chemical group 0.000 claims 1
- 125000006825 (C2-C5) haloalkyl group Chemical group 0.000 claims 1
- 125000006767 (C2-C6) haloalkynyloxy group Chemical group 0.000 claims 1
- 125000004198 2-fluorophenyl group Chemical group [H]C1=C([H])C(F)=C(*)C([H])=C1[H] 0.000 claims 1
- MHHBHSAYGWOQIM-UHFFFAOYSA-N N'-(2,5-dimethylphenyl)-4-[4-(5-phenyl-4,5-dihydro-1,2-oxazol-3-yl)-1,3-thiazol-2-yl]piperidine-1-carboximidamide Chemical compound CC1=CC=C(C)C(NC(=N)N2CCC(CC2)C=2SC=C(N=2)C=2CC(ON=2)C=2C=CC=CC=2)=C1 MHHBHSAYGWOQIM-UHFFFAOYSA-N 0.000 claims 1
- 150000001204 N-oxides Chemical class 0.000 claims 1
- 241000233654 Oomycetes Species 0.000 claims 1
- 125000004450 alkenylene group Chemical group 0.000 claims 1
- 125000004702 alkoxy alkyl carbonyl group Chemical group 0.000 claims 1
- 125000006466 alkoxy alkyl cycloalkyl group Chemical group 0.000 claims 1
- 125000005082 alkoxyalkenyl group Chemical group 0.000 claims 1
- 125000000033 alkoxyamino group Chemical group 0.000 claims 1
- 125000005085 alkoxycarbonylalkoxy group Chemical group 0.000 claims 1
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 claims 1
- 125000004949 alkyl amino carbonyl amino group Chemical group 0.000 claims 1
- 125000004471 alkyl aminosulfonyl group Chemical group 0.000 claims 1
- 125000004947 alkyl aryl amino group Chemical group 0.000 claims 1
- 125000002947 alkylene group Chemical group 0.000 claims 1
- 125000005038 alkynylalkyl group Chemical group 0.000 claims 1
- 125000004103 aminoalkyl group Chemical group 0.000 claims 1
- 230000000844 anti-bacterial Effects 0.000 claims 1
- 125000004429 atoms Chemical group 0.000 claims 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims 1
- 125000004966 cyanoalkyl group Chemical group 0.000 claims 1
- 125000004465 cycloalkenyloxy group Chemical group 0.000 claims 1
- 125000005149 cycloalkylsulfinyl group Chemical group 0.000 claims 1
- 125000004983 dialkoxyalkyl group Chemical group 0.000 claims 1
- 125000004472 dialkylaminosulfonyl group Chemical group 0.000 claims 1
- 201000010099 disease Diseases 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 230000002538 fungal Effects 0.000 claims 1
- 125000004443 haloalkoxycarbonylamino group Chemical group 0.000 claims 1
- 125000005843 halogen group Chemical group 0.000 claims 1
- 125000000842 isoxazolyl group Chemical group 0.000 claims 1
- AGYVSBQQNSDGIS-UHFFFAOYSA-N methyl N-(2,5-dimethylphenyl)-4-[4-[5-(2-oxo-1,3-benzoxazol-3-yl)-4,5-dihydro-1,2-oxazol-3-yl]-1,3-thiazol-2-yl]piperidine-1-carboximidate Chemical compound C1CC(C=2SC=C(N=2)C=2CC(ON=2)N2C(OC3=CC=CC=C32)=O)CCN1C(OC)=NC1=CC(C)=CC=C1C AGYVSBQQNSDGIS-UHFFFAOYSA-N 0.000 claims 1
- 125000004674 methylcarbonyl group Chemical group CC(=O)* 0.000 claims 1
- 125000006574 non-aromatic ring group Chemical group 0.000 claims 1
- 230000001717 pathogenic Effects 0.000 claims 1
- 244000052769 pathogens Species 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 239000011780 sodium chloride Substances 0.000 claims 1
- FZWLAAWBMGSTSO-UHFFFAOYSA-N thiazole Chemical group C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 claims 1
- XCJZAEBHRKDWQG-UHFFFAOYSA-N CC(C1)=NOC1c(c(OC)cc(OC)c1)c1OC Chemical compound CC(C1)=NOC1c(c(OC)cc(OC)c1)c1OC XCJZAEBHRKDWQG-UHFFFAOYSA-N 0.000 description 1
- 0 CC(C1)=NOC1c1c(C)cc(*)cc1C Chemical compound CC(C1)=NOC1c1c(C)cc(*)cc1C 0.000 description 1
- KPHATKPOJFGEAO-UHFFFAOYSA-N CC(C1)=NOC1c1ccccc1 Chemical compound CC(C1)=NOC1c1ccccc1 KPHATKPOJFGEAO-UHFFFAOYSA-N 0.000 description 1
- WCKLKDXFQHATPQ-UHFFFAOYSA-N CC(C1)=NOC1c1ccccc1C(OC)=O Chemical compound CC(C1)=NOC1c1ccccc1C(OC)=O WCKLKDXFQHATPQ-UHFFFAOYSA-N 0.000 description 1
- REDZCUVHHXAOGE-GFCCVEGCSA-N CC(C1)=NO[C@]1(c(cccc1)c1N1CI)C1=O Chemical compound CC(C1)=NO[C@]1(c(cccc1)c1N1CI)C1=O REDZCUVHHXAOGE-GFCCVEGCSA-N 0.000 description 1
- LBZIXNGCDVMNGZ-GFCCVEGCSA-N CC(C1)=NO[C@]1(c1c2cccc1)N(C)C2=O Chemical compound CC(C1)=NO[C@]1(c1c2cccc1)N(C)C2=O LBZIXNGCDVMNGZ-GFCCVEGCSA-N 0.000 description 1
- KBCUKLBCFHQJRI-NSHDSACASA-N CC(C1)=NO[C@]1(c1ccccc1)C#N Chemical compound CC(C1)=NO[C@]1(c1ccccc1)C#N KBCUKLBCFHQJRI-NSHDSACASA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6239508P | 2008-01-25 | 2008-01-25 | |
| US61/062,395 | 2008-01-25 | ||
| PCT/US2009/031686 WO2009094445A2 (en) | 2008-01-25 | 2009-01-22 | Fungicidal hetercyclic compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011510928A JP2011510928A (ja) | 2011-04-07 |
| JP2011510928A5 true JP2011510928A5 (US06653308-20031125-C00173.png) | 2012-02-23 |
| JP5529044B2 JP5529044B2 (ja) | 2014-06-25 |
Family
ID=40791139
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010544413A Expired - Fee Related JP5529044B2 (ja) | 2008-01-25 | 2009-01-22 | 殺菌性複素環化合物 |
Country Status (9)
Families Citing this family (60)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9090604B2 (en) | 2006-07-27 | 2015-07-28 | E I Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| WO2008013622A2 (en) | 2006-07-27 | 2008-01-31 | E. I. Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| US9643922B2 (en) | 2008-08-18 | 2017-05-09 | Yale University | MIF modulators |
| US9540322B2 (en) | 2008-08-18 | 2017-01-10 | Yale University | MIF modulators |
| WO2010021693A2 (en) * | 2008-08-18 | 2010-02-25 | Yale University | Mif modulators |
| UY32285A (es) | 2008-12-02 | 2010-06-30 | Du Pont | Compuestos heterocíclicos fungicidas |
| WO2010066353A1 (de) | 2008-12-11 | 2010-06-17 | Bayer Cropscience Ag | Thiazolyoximether und -hydrazone asl pflanzenschutzmittel |
| US20100267706A1 (en) * | 2009-04-20 | 2010-10-21 | Institute For Oneworld Health | Compounds, Compositions and Methods Comprising Pyridazine Derivatives |
| US8927551B2 (en) | 2009-05-18 | 2015-01-06 | Infinity Pharmaceuticals, Inc. | Isoxazolines as inhibitors of fatty acid amide hydrolase |
| AR076687A1 (es) * | 2009-05-18 | 2011-06-29 | Infinity Pharmaceuticals Inc | Isoxazolinas como inhibidores de la amidahidrolasa de acidos grasos y com-posiciones farmaceuticas que los contienen |
| US9149465B2 (en) | 2009-05-18 | 2015-10-06 | Infinity Pharmaceuticals, Inc. | Isoxazolines as inhibitors of fatty acid amide hydrolase |
| US8557821B2 (en) * | 2009-08-12 | 2013-10-15 | Syngenta Crop Protection, Llc | Microbiocidal heterocycles |
| WO2011051244A1 (de) | 2009-10-30 | 2011-05-05 | Bayer Cropscience Ag | Heteroarylpiperidin und -piperazin derivate |
| CA2780905A1 (en) * | 2009-12-11 | 2011-06-16 | E.I. Du Pont De Nemours And Company | Azocyclic inhibitors of fatty acid amide hydrolase |
| MX2012007200A (es) | 2009-12-21 | 2012-07-10 | Bayer Cropscience Ag | Bis(difluorometil)pirazoles como fungicidas. |
| ES2534516T3 (es) * | 2010-01-07 | 2015-04-23 | E.I. Du Pont De Nemours And Company | Compuestos heterocíclicos fungicidas |
| EP2563786B1 (de) | 2010-04-28 | 2016-11-02 | Bayer Intellectual Property GmbH | Ketoheteroarylpiperidin und -piperazin Derivate als Fungizide |
| US8815775B2 (en) | 2010-05-18 | 2014-08-26 | Bayer Cropscience Ag | Bis(difluoromethyl)pyrazoles as fungicides |
| EP2571866A1 (en) * | 2010-05-20 | 2013-03-27 | E.I. Du Pont De Nemours And Company | Fungicidal oximes and hydrazones |
| BR112012030184A2 (pt) | 2010-05-27 | 2015-12-29 | Bayer Cropscience Ag | derivados de ácido piridinilcarboxílico como fungicidas |
| US20120122928A1 (en) | 2010-08-11 | 2012-05-17 | Bayer Cropscience Ag | Heteroarylpiperidine and -Piperazine Derivatives as Fungicides |
| AU2015261660B2 (en) * | 2010-08-25 | 2017-01-05 | Bayer Cropscience Aktiengesellschaft | Heteroarylpiperidine and -piperazine derivatives as fungicides |
| EP2423210A1 (de) | 2010-08-25 | 2012-02-29 | Bayer CropScience AG | Heteroarylpiperidin- und -piperazinderivate als Fungizide |
| US8759527B2 (en) | 2010-08-25 | 2014-06-24 | Bayer Cropscience Ag | Heteroarylpiperidine and -piperazine derivatives as fungicides |
| WO2012055837A1 (de) | 2010-10-27 | 2012-05-03 | Bayer Cropscience Ag | Heteroarylpiperidin und -piperazinderivate als fungizide |
| JP5695397B2 (ja) * | 2010-11-25 | 2015-04-01 | 日本エンバイロケミカルズ株式会社 | 防カビ剤、それを用いる防カビ方法、生育阻止剤およびそれを用いる生育阻止方法 |
| AU2011344161A1 (en) * | 2010-12-17 | 2013-06-20 | E. I. Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| CN104987330B (zh) | 2011-02-01 | 2019-04-05 | 拜耳知识产权有限责任公司 | 作为杀真菌剂的杂芳基哌啶和杂芳基哌嗪衍生物 |
| EP2532233A1 (en) | 2011-06-07 | 2012-12-12 | Bayer CropScience AG | Active compound combinations |
| MX355824B (es) | 2011-09-15 | 2018-05-02 | Bayer Ip Gmbh | Piperidinpirazoles como fungicidas. |
| DK2797899T3 (en) | 2011-12-27 | 2016-04-04 | Bayer Ip Gmbh | Heteroarylpiperidin and -piperazinderivater as fungicides |
| EA027595B1 (ru) | 2012-02-02 | 2017-08-31 | Актелион Фармасьютиклз Лтд. | 4-(бензоимидазол-2-ил)тиазольные соединения и родственные азапроизводные |
| BR112014020898B1 (pt) | 2012-02-27 | 2020-08-11 | Bayer Intellectual Property Gmbh | Combinação, método para controle de fungos fitopatogênicos prejudiciais compreendendo a referida combinação e seu uso |
| AU2013277673A1 (en) | 2012-06-22 | 2015-01-22 | E. I. Du Pont De Nemours And Company | Fungicidal heterocyclic compounds |
| US9145370B2 (en) | 2012-08-30 | 2015-09-29 | Bayer Cropscience Ag | Procedure for the decarboxylation of 3,5-bis(haloalkyl)-pyrazole-4-carboxylic acid derivatives |
| EP2801575A1 (en) | 2013-05-07 | 2014-11-12 | Bayer CropScience AG | Heteroaryldihydropyridine derivatives as fungicides |
| CN105473585B (zh) | 2013-06-24 | 2018-04-13 | 拜耳作物科学股份公司 | 作为杀真菌剂的哌啶羧酸衍生物 |
| WO2015011099A1 (en) | 2013-07-22 | 2015-01-29 | Actelion Pharmaceuticals Ltd | 1-(piperazin-1-yl)-2-([1,2,4]triazol-1-yl)-ethanone derivatives |
| WO2015028457A1 (en) * | 2013-08-28 | 2015-03-05 | Bayer Cropscience Ag | Malonic ester derivatives of heteroarylpiperidines and -piperazines as fungicides |
| AU2015238574B2 (en) | 2014-03-24 | 2019-02-21 | Bayer Cropscience Aktiengesellschaft | Phenylpiperidinecarboxamide derivatives as fungicides |
| AR099789A1 (es) | 2014-03-24 | 2016-08-17 | Actelion Pharmaceuticals Ltd | Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina |
| TWI665192B (zh) * | 2014-05-28 | 2019-07-11 | 德商拜耳作物科學股份有限公司 | 製備二氫異唑衍生物之方法 |
| CN106414437B (zh) * | 2014-05-28 | 2019-06-21 | 拜耳作物科学股份公司 | 制备噻唑衍生物的方法 |
| WO2016024350A1 (ja) | 2014-08-13 | 2016-02-18 | 株式会社エス・ディー・エス バイオテック | 縮合１１員環化合物及びそれらを含有する農園芸用殺菌剤 |
| EP3766871A1 (en) * | 2014-08-13 | 2021-01-20 | Nippon Soda Co., Ltd. | Diarylimidazole compound and pest control agent |
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| AR103399A1 (es) | 2015-01-15 | 2017-05-10 | Actelion Pharmaceuticals Ltd | Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3 |
| WO2016202761A1 (en) | 2015-06-17 | 2016-12-22 | Bayer Cropscience Aktiengesellschaft | Active compound combinations |
| CN105541830B (zh) * | 2015-12-14 | 2018-04-27 | 北京迪尔乐农业高新技术研发中心 | 一种杀菌化合物、制备方法及其应用 |
| ES2895047T3 (es) | 2016-02-08 | 2022-02-17 | Gowan Crop Prot Limited | Proceso para la preparación del compuesto 1,2-bencenodimetanol |
| JP6649967B2 (ja) * | 2016-02-08 | 2020-02-19 | 株式会社エス・ディー・エス バイオテック | 殺菌性組成物 |
| WO2018193387A1 (en) | 2017-04-19 | 2018-10-25 | Pi Industries Ltd. | Heterocyclic compounds with microbiocidal properties |
| WO2019048988A1 (en) * | 2017-09-08 | 2019-03-14 | Pi Industries Ltd. | NOVEL FUNGICIDE HETEROCYCLIC COMPOUNDS |
| BR112020004356A2 (pt) * | 2017-09-08 | 2020-12-01 | Pi Industries Ltd. | novos compostos heterocíclicos fungicidas |
| CN109516962A (zh) * | 2018-12-13 | 2019-03-26 | 天津雅奥泰克科技有限公司 | 一种合成2,6-二氟苯基-1-(4,5-二氢异恶唑)-3-乙基酮的新方法 |
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| AR125834A1 (es) | 2021-05-15 | 2023-08-16 | Pi Industries Ltd | Composición agroquímica que comprende compuestos de piperidin-tiazol |
| CN113480489A (zh) * | 2021-08-19 | 2021-10-08 | 贵州大学 | 异噁唑联苯类化合物及其制备方法和应用 |
| CN117624158A (zh) * | 2022-08-26 | 2024-03-01 | 江苏中旗科技股份有限公司 | 含链状羧酸酰胺结构的化合物及其制备方法和应用、杀菌剂 |
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2009
- 2009-01-22 EP EP11007851.6A patent/EP2402332A3/en not_active Withdrawn
- 2009-01-22 EP EP09704518A patent/EP2260032A2/en not_active Withdrawn
- 2009-01-22 JP JP2010544413A patent/JP5529044B2/ja not_active Expired - Fee Related
- 2009-01-22 BR BRPI0905759-5A patent/BRPI0905759A2/pt not_active Application Discontinuation
- 2009-01-22 KR KR1020157014513A patent/KR20150065958A/ko not_active Application Discontinuation
- 2009-01-22 WO PCT/US2009/031686 patent/WO2009094445A2/en active Application Filing
- 2009-01-22 CN CN201410221847.2A patent/CN103965187A/zh active Pending
- 2009-01-22 KR KR1020107018519A patent/KR20100119552A/ko not_active Application Discontinuation
- 2009-01-22 CN CN200980105521.0A patent/CN101970432B/zh not_active Expired - Fee Related
- 2009-01-22 US US12/863,875 patent/US8349870B2/en not_active Expired - Fee Related
- 2009-01-22 MX MX2010008102A patent/MX2010008102A/es active IP Right Grant
- 2009-01-22 AU AU2009206468A patent/AU2009206468B2/en not_active Ceased
