JP2011507941A5 - - Google Patents

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Publication number
JP2011507941A5
JP2011507941A5 JP2010540175A JP2010540175A JP2011507941A5 JP 2011507941 A5 JP2011507941 A5 JP 2011507941A5 JP 2010540175 A JP2010540175 A JP 2010540175A JP 2010540175 A JP2010540175 A JP 2010540175A JP 2011507941 A5 JP2011507941 A5 JP 2011507941A5
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JP
Japan
Prior art keywords
group
iii
hydroxy
aryl
optionally substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010540175A
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English (en)
Japanese (ja)
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JP2011507941A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/GB2008/051221 external-priority patent/WO2009081208A1/en
Publication of JP2011507941A publication Critical patent/JP2011507941A/ja
Publication of JP2011507941A5 publication Critical patent/JP2011507941A5/ja
Pending legal-status Critical Current

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JP2010540175A 2007-12-26 2008-12-19 プレガバリンの製造方法 Pending JP2011507941A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1729KO2007 2007-12-26
PCT/GB2008/051221 WO2009081208A1 (en) 2007-12-26 2008-12-19 Processes to pregabalin

Publications (2)

Publication Number Publication Date
JP2011507941A JP2011507941A (ja) 2011-03-10
JP2011507941A5 true JP2011507941A5 (enExample) 2012-02-16

Family

ID=40474656

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010540175A Pending JP2011507941A (ja) 2007-12-26 2008-12-19 プレガバリンの製造方法

Country Status (7)

Country Link
US (1) US20100324139A1 (enExample)
EP (1) EP2222630A1 (enExample)
JP (1) JP2011507941A (enExample)
CN (1) CN101965328A (enExample)
AU (1) AU2008339583A1 (enExample)
CA (1) CA2710152A1 (enExample)
WO (1) WO2009081208A1 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA019285B1 (ru) * 2008-05-21 2014-02-28 Сандоз Аг Способ стереоселективного ферментативного гидролиза эфира 5-метил-3-нитрометилгексановой кислоты
US9545415B2 (en) * 2012-01-06 2017-01-17 Skyview Enterprise Ltd. Anti-inflammatory compounds in combination with hydrogen for the treatment of inflammation
JP6482465B2 (ja) 2012-11-07 2019-03-13 ハイカル リミテッド プレガバリンの調製方法
WO2015189068A1 (en) 2014-06-12 2015-12-17 Siegfried Ltd. Method for the preparation of beta-substituted gamma-amino carboxylic acids
CN107673967A (zh) * 2016-08-01 2018-02-09 上海朴颐化学科技有限公司 一种α‑氟代丙酰乙酸酯的制备方法
CN108373411A (zh) * 2017-12-16 2018-08-07 山东新华制药股份有限公司 高纯度4-氯-3-羟基丁酸乙酯的制备方法
CN108218649B (zh) * 2017-12-29 2021-07-30 联化科技股份有限公司 普瑞巴林及其中间体的合成方法
CN110407715A (zh) * 2019-07-01 2019-11-05 陕西师范大学 一种普瑞巴林中间体的合成方法
CN110803994B (zh) * 2019-11-19 2023-06-30 陕西科技大学 一种普瑞巴林中间体3-硝基亚甲基-5-甲基-己酸乙酯的合成方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3856816B2 (ja) * 1992-05-20 2006-12-13 ノースウェスターン ユニヴァーシティ 抗発作治療用のｇａｂａ及びｌ−グルタミン酸類縁体
US5637767A (en) * 1995-06-07 1997-06-10 Warner-Lambert Company Method of making (S)-3-(aminomethyl)-5-methylhexanoic acid
SK287303B6 (sk) * 2000-01-27 2010-06-07 Warner-Lambert Company Spôsob prípravy derivátu (S)-3-kyano-5-metyl-hexánovej kyseliny, spôsob a medziprodukt na prípravu pregabalínu
DE10203122A1 (de) * 2002-01-25 2003-07-31 Gruenenthal Gmbh Verfahren zur Herstellung von substituierten Acrylsäureestern bzw. deren Einsatz zur Herstellung von substituierten gamma-Aminosäuren
US6903233B2 (en) * 2002-03-11 2005-06-07 Takasago International Corporation Process for producing optically active 3-halogenocarboxylic acid ester and 3-azidocarboxylic acid ester
JP4043810B2 (ja) * 2002-03-11 2008-02-06 高砂香料工業株式会社 光学活性３−クロロカルボン酸エステルの製造方法
US20030225149A1 (en) * 2002-04-30 2003-12-04 Blazecka Peter G. Process for preparing highly functionalized gamma-butyrolactams and gamma-amino acids
RS51210B (sr) * 2004-06-21 2010-12-31 Warner-Lambert Company Llc. Dobijanje pregaballina i srodnih jedinjenja
US20070066846A1 (en) * 2005-04-11 2007-03-22 Asher Maymon Process for making (S)-Pregabalin

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