JP2011503193A - ヒトホスファチジルイノシトール3−キナーゼδの阻害剤 - Google Patents

ヒトホスファチジルイノシトール3−キナーゼδの阻害剤 Download PDF

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JP2011503193A
JP2011503193A JP2010534149A JP2010534149A JP2011503193A JP 2011503193 A JP2011503193 A JP 2011503193A JP 2010534149 A JP2010534149 A JP 2010534149A JP 2010534149 A JP2010534149 A JP 2010534149A JP 2011503193 A JP2011503193 A JP 2011503193A
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alkylene
substituted
unsubstituted
aryl
heteroaryl
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JP2011503193A5 (https=
Inventor
スティーブン エル. ホワイト,
フーキアン ルアン,
エドワード エー. ケシキ,
ユージーン ソーセット,
フランシン ファロウズ,
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Icos Corp
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Icos Corp
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Pulmonology (AREA)
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  • Communicable Diseases (AREA)
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JP2010534149A 2007-11-13 2008-11-12 ヒトホスファチジルイノシトール3−キナーゼδの阻害剤 Pending JP2011503193A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US98772307P 2007-11-13 2007-11-13
PCT/US2008/083262 WO2009064802A2 (en) 2007-11-13 2008-11-12 Inhibitors of human phosphatidyl-inositol 3-kinase delta

Publications (2)

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JP2011503193A true JP2011503193A (ja) 2011-01-27
JP2011503193A5 JP2011503193A5 (https=) 2012-12-20

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US (1) US20110021541A1 (https=)
EP (1) EP2220089A4 (https=)
JP (1) JP2011503193A (https=)
KR (1) KR20100119745A (https=)
CN (1) CN101952292A (https=)
AU (1) AU2008321099A1 (https=)
CA (1) CA2716334A1 (https=)
EA (1) EA201070611A1 (https=)
GE (1) GEP20125635B (https=)
IL (1) IL205747A0 (https=)
NZ (1) NZ585460A (https=)
SG (1) SG185996A1 (https=)
WO (1) WO2009064802A2 (https=)

Cited By (4)

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JP2011508782A (ja) * 2008-01-04 2011-03-17 インテリカイン, インコーポレイテッド 特定の化学的実体、組成物および方法
JP2014520888A (ja) * 2011-07-19 2014-08-25 インフィニティー ファーマシューティカルズ, インコーポレイテッド 複素環式化合物及びその使用
JP2014520887A (ja) * 2011-07-19 2014-08-25 インフィニティー ファーマシューティカルズ, インコーポレイテッド 複素環式化合物及びその使用
JP2015509509A (ja) * 2012-03-06 2015-03-30 ベイジン ウェイフオン イーミーン バイオ−テクノロジー リミティドカンパニー 慢性閉塞性疾患を治療するための医薬品組成物の製造のための、ルパタジンの使用

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TWI674262B (zh) 2011-01-10 2019-10-11 美商英菲尼提製藥股份有限公司 製備異喹啉酮之方法及異喹啉酮之固體形式
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