EA201070611A1 - Ингибиторы человеческой фосфатидилинозитол-3-киназы дельта - Google Patents

Ингибиторы человеческой фосфатидилинозитол-3-киназы дельта

Info

Publication number
EA201070611A1
EA201070611A1 EA201070611A EA201070611A EA201070611A1 EA 201070611 A1 EA201070611 A1 EA 201070611A1 EA 201070611 A EA201070611 A EA 201070611A EA 201070611 A EA201070611 A EA 201070611A EA 201070611 A1 EA201070611 A1 EA 201070611A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pi3kδ
kinase delta
delta inhibitors
human phosphatidylinositol
activity
Prior art date
Application number
EA201070611A
Other languages
English (en)
Russian (ru)
Inventor
Стефен Л. Уайт
Фуцян Жуань
Эдвард А. Кесицки
Юджин Торсетт
Франсин Фару
Original Assignee
Айкос Корпорейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Айкос Корпорейшн filed Critical Айкос Корпорейшн
Publication of EA201070611A1 publication Critical patent/EA201070611A1/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Communicable Diseases (AREA)
  • Otolaryngology (AREA)
  • Biomedical Technology (AREA)
  • Transplantation (AREA)
EA201070611A 2007-11-13 2008-11-12 Ингибиторы человеческой фосфатидилинозитол-3-киназы дельта EA201070611A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US98772307P 2007-11-13 2007-11-13
PCT/US2008/083262 WO2009064802A2 (en) 2007-11-13 2008-11-12 Inhibitors of human phosphatidyl-inositol 3-kinase delta

Publications (1)

Publication Number Publication Date
EA201070611A1 true EA201070611A1 (ru) 2010-12-30

Family

ID=40639422

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201070611A EA201070611A1 (ru) 2007-11-13 2008-11-12 Ингибиторы человеческой фосфатидилинозитол-3-киназы дельта

Country Status (13)

Country Link
US (1) US20110021541A1 (https=)
EP (1) EP2220089A4 (https=)
JP (1) JP2011503193A (https=)
KR (1) KR20100119745A (https=)
CN (1) CN101952292A (https=)
AU (1) AU2008321099A1 (https=)
CA (1) CA2716334A1 (https=)
EA (1) EA201070611A1 (https=)
GE (1) GEP20125635B (https=)
IL (1) IL205747A0 (https=)
NZ (1) NZ585460A (https=)
SG (1) SG185996A1 (https=)
WO (1) WO2009064802A2 (https=)

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