JP2011500537A5 - - Google Patents
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- Publication number
- JP2011500537A5 JP2011500537A5 JP2010528414A JP2010528414A JP2011500537A5 JP 2011500537 A5 JP2011500537 A5 JP 2011500537A5 JP 2010528414 A JP2010528414 A JP 2010528414A JP 2010528414 A JP2010528414 A JP 2010528414A JP 2011500537 A5 JP2011500537 A5 JP 2011500537A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- pyrrolidinyl
- chlorophenyl
- alkyl
- compound according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US97910507P | 2007-10-11 | 2007-10-11 | |
| PCT/EP2008/063642 WO2009047336A1 (en) | 2007-10-11 | 2008-10-10 | Phthalazine and pyrido [3,4-d] pyridaz ine compounds as h1 receptor antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011500537A JP2011500537A (ja) | 2011-01-06 |
| JP2011500537A5 true JP2011500537A5 (enExample) | 2011-12-01 |
Family
ID=40104668
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010528414A Ceased JP2011500537A (ja) | 2007-10-11 | 2008-10-10 | Ｈ１受容体アンタゴニストとしてのフタラジンおよびピリド［３，４−ｄ］ピリダジン化合物 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20100216799A1 (enExample) |
| EP (1) | EP2215082B1 (enExample) |
| JP (1) | JP2011500537A (enExample) |
| AT (1) | ATE525370T1 (enExample) |
| ES (1) | ES2369320T3 (enExample) |
| WO (1) | WO2009047336A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006115221A1 (ja) * | 2005-04-21 | 2006-11-02 | Nippon Shinyaku Co., Ltd. | フタラジノン誘導体及びその医薬 |
| UA97506C2 (xx) * | 2006-12-28 | 2012-02-27 | Эбботт Лаборетриз | Інгібітори полі(adp-рибозо)полімерази$ингибиторы поли(adp-рибозо)полимеразы |
| CA2685219C (en) * | 2007-05-04 | 2012-06-19 | Amgen Inc. | Diazaquinolones that inhibit prolyl hydroxylase activity |
| CN115135315B (zh) | 2019-12-20 | 2024-11-26 | 米拉蒂治疗股份有限公司 | Sos1抑制剂 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3813384A (en) * | 1972-01-17 | 1974-05-28 | Asta Werke Ag Chem Fab | Basically substituted benzyl phthalazone derivatives,acid salts thereof and process for the production thereof |
| PH23995A (en) * | 1984-01-09 | 1990-02-09 | Janssen Pharmaceutica Nv | 4((bicycle heterocyclyl)-methyl and hetero)piperidines |
| DE3575135D1 (de) * | 1984-09-14 | 1990-02-08 | Asta Pharma Ag | Substituierte benzylphthalazinon-derivate. |
| DE3634942A1 (de) * | 1985-11-11 | 1987-05-14 | Asta Werke Ag Chem Fab | Neue 4-benzyl-1-(2h)-phthalazinon-derivate |
| ATE60598T1 (de) * | 1985-11-11 | 1991-02-15 | Asta Pharma Ag | 4-benzyl-1-(2h)-phthalazinon-derivate. |
| EP0289939A1 (de) * | 1987-05-08 | 1988-11-09 | ASTA Pharma AG | Neue 4-Benzyl-1-(2H)-phthalazinon-Derivate mit einem Aminosäurerest |
| CZ199593A3 (en) * | 1992-10-02 | 1994-04-13 | Asta Medica Ag | Phthalazinone derivatives exhibiting anti-arrhythmic and analgesic activity and eliminating resistance to a plurality of medicaments (mdr) |
| US6180629B1 (en) * | 1998-08-14 | 2001-01-30 | Cell Pathways, Inc. | [4,5]-Fused-1,3-disubstituted-1,2-diazine-6-one derivatives with nitrogen containing substitutents in position one for the treatment of neoplasia |
| ES2209337T3 (es) * | 1998-08-14 | 2004-06-16 | Pfizer Inc. | Agentes antitromboticos. |
| US20030073692A1 (en) * | 2001-08-07 | 2003-04-17 | Pharmacia & Upjohn S.P.A. | Amino-phthalazinone derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them |
| CA2519220A1 (en) * | 2003-03-18 | 2004-09-30 | Merck & Co., Inc. | Amino cyclobutylamide modulators of chemokine receptor activity |
| JP4735261B2 (ja) * | 2003-06-27 | 2011-07-27 | Ｍｓｄ株式会社 | ヘテロアリールオキシ含窒素飽和ヘテロ環誘導体 |
| ES2341813T3 (es) * | 2006-12-20 | 2010-06-28 | Glaxo Group Limited | 4-bencil-1 (2h)-ftalazinonas como antagonistas del receptor h1. |
-
2008
- 2008-10-10 EP EP08805231A patent/EP2215082B1/en not_active Not-in-force
- 2008-10-10 JP JP2010528414A patent/JP2011500537A/ja not_active Ceased
- 2008-10-10 WO PCT/EP2008/063642 patent/WO2009047336A1/en not_active Ceased
- 2008-10-10 US US12/681,945 patent/US20100216799A1/en not_active Abandoned
- 2008-10-10 ES ES08805231T patent/ES2369320T3/es active Active
- 2008-10-10 AT AT08805231T patent/ATE525370T1/de not_active IP Right Cessation
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